DOP2014000152A - Inhibidores de bromodominios - Google Patents

Inhibidores de bromodominios

Info

Publication number
DOP2014000152A
DOP2014000152A DO2014000152A DO2014000152A DOP2014000152A DO P2014000152 A DOP2014000152 A DO P2014000152A DO 2014000152 A DO2014000152 A DO 2014000152A DO 2014000152 A DO2014000152 A DO 2014000152A DO P2014000152 A DOP2014000152 A DO P2014000152A
Authority
DO
Dominican Republic
Prior art keywords
bromodominium
inhibitors
compounds
formula
diseases
Prior art date
Application number
DO2014000152A
Other languages
English (en)
Spanish (es)
Inventor
Le Wang
John K Pratt
Warren M Kati
Keith F Mcdaniel
Lisa Hasvold
William J Mcclellan
Yujia Dai
Robert A Mantei
Steven D Fidanze
James H Holms
Dachun Liu
George S Sheppard
Carol K Wada
Original Assignee
Abbvie Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbvie Inc filed Critical Abbvie Inc
Publication of DOP2014000152A publication Critical patent/DOP2014000152A/es

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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DO2014000152A 2011-12-30 2014-06-26 Inhibidores de bromodominios DOP2014000152A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/CN2011/002224 WO2013097052A1 (en) 2011-12-30 2011-12-30 Bromodomain inhibitors

Publications (1)

Publication Number Publication Date
DOP2014000152A true DOP2014000152A (es) 2014-08-31

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DO2014000152A DOP2014000152A (es) 2011-12-30 2014-06-26 Inhibidores de bromodominios

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