CR20140332A - Inhibidores de bromodominios - Google Patents

Inhibidores de bromodominios

Info

Publication number
CR20140332A
CR20140332A CR20140332A CR20140332A CR20140332A CR 20140332 A CR20140332 A CR 20140332A CR 20140332 A CR20140332 A CR 20140332A CR 20140332 A CR20140332 A CR 20140332A CR 20140332 A CR20140332 A CR 20140332A
Authority
CR
Costa Rica
Prior art keywords
bromodominium
inhibitors
compounds
formula
pharmaceutically acceptable
Prior art date
Application number
CR20140332A
Other languages
English (en)
Spanish (es)
Inventor
Le Wang
John K Pratt
Keith F Mcdaniel
Yujia Dai
Steven D Fidanze
Lisa Hasvold
James H Holms
Warren M Kati
Dachun Liu
Robert A Mantei
William J Mcclellan
George S Sheppard
Carol K Wada
Original Assignee
Abbvie Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbvie Inc filed Critical Abbvie Inc
Publication of CR20140332A publication Critical patent/CR20140332A/es

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Classifications

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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  • Virology (AREA)
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CR20140332A 2011-12-30 2014-07-10 Inhibidores de bromodominios CR20140332A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/CN2011/002224 WO2013097052A1 (en) 2011-12-30 2011-12-30 Bromodomain inhibitors
PCT/CN2012/086357 WO2013097601A1 (en) 2011-12-30 2012-12-11 Bromodomain inhibitors

Publications (1)

Publication Number Publication Date
CR20140332A true CR20140332A (es) 2014-11-10

Family

ID=48696151

Family Applications (1)

Application Number Title Priority Date Filing Date
CR20140332A CR20140332A (es) 2011-12-30 2014-07-10 Inhibidores de bromodominios

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