CN105473581B - 作为溴结构域抑制剂的新取代的双环化合物 - Google Patents
作为溴结构域抑制剂的新取代的双环化合物 Download PDFInfo
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- CN105473581B CN105473581B CN201480045603.1A CN201480045603A CN105473581B CN 105473581 B CN105473581 B CN 105473581B CN 201480045603 A CN201480045603 A CN 201480045603A CN 105473581 B CN105473581 B CN 105473581B
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Abstract
Description
实施例化合物 | 体内活性 |
实施例9 | 活性 |
实施例化合物 | 体内活性 |
实施例9 | 活性 |
实施例化合物 | 体内活性 |
实施例9 | 活性 |
实施例化合物 | 体内活性 |
实施例9 | 活性 |
Claims (23)
Applications Claiming Priority (5)
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US201361837830P | 2013-06-21 | 2013-06-21 | |
US61/837,830 | 2013-06-21 | ||
US201361911668P | 2013-12-04 | 2013-12-04 | |
US61/911,668 | 2013-12-04 | ||
PCT/IB2014/002240 WO2015004534A2 (en) | 2013-06-21 | 2014-06-20 | Novel substituted bicyclic compounds as bromodomain inhibitors |
Publications (2)
Publication Number | Publication Date |
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CN105473581A CN105473581A (zh) | 2016-04-06 |
CN105473581B true CN105473581B (zh) | 2019-04-23 |
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CN201480045605.0A Active CN105492439B (zh) | 2013-06-21 | 2014-06-20 | 作为溴结构域抑制剂的取代的双环化合物 |
CN201480045603.1A Active CN105473581B (zh) | 2013-06-21 | 2014-06-20 | 作为溴结构域抑制剂的新取代的双环化合物 |
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CN201480045605.0A Active CN105492439B (zh) | 2013-06-21 | 2014-06-20 | 作为溴结构域抑制剂的取代的双环化合物 |
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CA (2) | CA2915561C (zh) |
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