CL2014001752A1 - Compuestos biciclicos sustituidos; composicion farmaceutica que los comprende; y uso en el tratamiento de enfermedades tales como cancer, alzheimer, sida, entre otras. - Google Patents
Compuestos biciclicos sustituidos; composicion farmaceutica que los comprende; y uso en el tratamiento de enfermedades tales como cancer, alzheimer, sida, entre otras.Info
- Publication number
- CL2014001752A1 CL2014001752A1 CL2014001752A CL2014001752A CL2014001752A1 CL 2014001752 A1 CL2014001752 A1 CL 2014001752A1 CL 2014001752 A CL2014001752 A CL 2014001752A CL 2014001752 A CL2014001752 A CL 2014001752A CL 2014001752 A1 CL2014001752 A1 CL 2014001752A1
- Authority
- CL
- Chile
- Prior art keywords
- alzheimer
- aids
- cancer
- diseases
- treatment
- Prior art date
Links
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/541—Non-condensed thiazines containing further heterocyclic rings
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
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- Diabetes (AREA)
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- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Oncology (AREA)
- Dermatology (AREA)
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- Communicable Diseases (AREA)
- Urology & Nephrology (AREA)
- Virology (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
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- Heart & Thoracic Surgery (AREA)
- Molecular Biology (AREA)
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- Reproductive Health (AREA)
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/CN2011/002224 WO2013097052A1 (en) | 2011-12-30 | 2011-12-30 | Bromodomain inhibitors |
Publications (1)
Publication Number | Publication Date |
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CL2014001752A1 true CL2014001752A1 (es) | 2014-10-10 |
Family
ID=48696151
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2014001752A CL2014001752A1 (es) | 2011-12-30 | 2014-06-27 | Compuestos biciclicos sustituidos; composicion farmaceutica que los comprende; y uso en el tratamiento de enfermedades tales como cancer, alzheimer, sida, entre otras. |
Country Status (39)
Country | Link |
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US (5) | US9296741B2 (es) |
EP (2) | EP3360874A1 (es) |
JP (3) | JP6117238B2 (es) |
KR (1) | KR102008975B1 (es) |
CN (2) | CN104136435B (es) |
AR (2) | AR089527A1 (es) |
AU (3) | AU2012361967B2 (es) |
BR (1) | BR112014016233B1 (es) |
CA (1) | CA2859619C (es) |
CL (1) | CL2014001752A1 (es) |
CO (1) | CO7020912A2 (es) |
CR (1) | CR20140332A (es) |
CY (1) | CY1120287T1 (es) |
DK (1) | DK2797918T3 (es) |
DO (1) | DOP2014000152A (es) |
EC (1) | ECSP14011359A (es) |
ES (1) | ES2665890T3 (es) |
GT (1) | GT201400133A (es) |
HK (3) | HK1203508A1 (es) |
HR (1) | HRP20180357T1 (es) |
HU (1) | HUE038391T2 (es) |
IL (1) | IL233454A (es) |
LT (1) | LT2797918T (es) |
ME (1) | ME03028B (es) |
MX (1) | MX341740B (es) |
NO (1) | NO2797918T3 (es) |
PE (1) | PE20142340A1 (es) |
PH (1) | PH12014501469A1 (es) |
PL (1) | PL2797918T3 (es) |
PT (1) | PT2797918T (es) |
RS (1) | RS56978B1 (es) |
RU (3) | RU2647592C2 (es) |
SG (1) | SG11201403717WA (es) |
SI (1) | SI2797918T1 (es) |
TW (1) | TWI602815B (es) |
UA (1) | UA111770C2 (es) |
UY (2) | UY34559A (es) |
WO (2) | WO2013097052A1 (es) |
ZA (1) | ZA201404616B (es) |
Families Citing this family (128)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR101857599B1 (ko) | 2010-05-14 | 2018-05-14 | 다나-파버 캔서 인스티튜트 인크. | 종양형성, 염증성 질환 및 다른 장애를 치료하기 위한 조성물 및 방법 |
WO2011143660A2 (en) | 2010-05-14 | 2011-11-17 | Dana-Farber Cancer Institute, Inc. | Compositions and methods for treating leukemia |
US9301962B2 (en) | 2010-05-14 | 2016-04-05 | Baylor College Of Medicine | Male contraceptive compositions and methods of use |
US9115096B2 (en) | 2011-05-10 | 2015-08-25 | Gilead Sciences, Inc. | Fused heterocyclic compounds as ion channel modulators |
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