DK2797918T3 - BROMDOMAIN INHIBITORS - Google Patents

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Publication number
DK2797918T3
DK2797918T3 DK12863599.2T DK12863599T DK2797918T3 DK 2797918 T3 DK2797918 T3 DK 2797918T3 DK 12863599 T DK12863599 T DK 12863599T DK 2797918 T3 DK2797918 T3 DK 2797918T3
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Prior art keywords
methyl
dihydro
pyridin
phenyl
pyrrol
Prior art date
Application number
DK12863599.2T
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Danish (da)
English (en)
Inventor
Le Wang
John K Pratt
Keith F Mcdaniel
Yujia Dai
Steven D Fidanze
Lisa Hasvold
James H Holms
Warren M Kati
Dachun Liu
Robert A Mantei
William J Mcclellan
George S Sheppard
Carol K Wada
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Abbvie Inc
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Publication of DK2797918T3 publication Critical patent/DK2797918T3/en

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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  • Veterinary Medicine (AREA)
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  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Dermatology (AREA)
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  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
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DK12863599.2T 2011-12-30 2012-12-11 BROMDOMAIN INHIBITORS DK2797918T3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/CN2011/002224 WO2013097052A1 (en) 2011-12-30 2011-12-30 Bromodomain inhibitors
PCT/CN2012/086357 WO2013097601A1 (en) 2011-12-30 2012-12-11 Bromodomain inhibitors

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DK2797918T3 true DK2797918T3 (en) 2018-03-12

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