AR089527A1 - Inhibidores de bromodominios - Google Patents

Inhibidores de bromodominios

Info

Publication number
AR089527A1
AR089527A1 ARP120105053A ARP120105053A AR089527A1 AR 089527 A1 AR089527 A1 AR 089527A1 AR P120105053 A ARP120105053 A AR P120105053A AR P120105053 A ARP120105053 A AR P120105053A AR 089527 A1 AR089527 A1 AR 089527A1
Authority
AR
Argentina
Prior art keywords
alkylene
alkyl
haloalkyl
independently
hydrogen
Prior art date
Application number
ARP120105053A
Other languages
English (en)
Spanish (es)
Inventor
F Mdaniel Keith
A Mantei Robert
S Sheppard George
K Wada Carol
Wang Le
Dai Yujia
D Fidanze Steven
Hasvold Lisa
H Holms James
K Pratt John
J Mclellan William
M Kati Warren
Liu Dachun
Original Assignee
Abbvie Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbvie Inc filed Critical Abbvie Inc
Publication of AR089527A1 publication Critical patent/AR089527A1/es

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
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ARP120105053A 2011-12-30 2012-12-28 Inhibidores de bromodominios AR089527A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/CN2011/002224 WO2013097052A1 (en) 2011-12-30 2011-12-30 Bromodomain inhibitors

Publications (1)

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AR089527A1 true AR089527A1 (es) 2014-08-27

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ARP120105053A AR089527A1 (es) 2011-12-30 2012-12-28 Inhibidores de bromodominios
ARP220100723A AR125222A2 (es) 2011-12-30 2022-03-25 Inhibidores de bromodominios

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ARP220100723A AR125222A2 (es) 2011-12-30 2022-03-25 Inhibidores de bromodominios

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