CY2007002I1 - Ω-καρβοξυαρυλυποκατεστημενες διφαινυλουριες σαν αναστολεις της raf κινασης - Google Patents

Ω-καρβοξυαρυλυποκατεστημενες διφαινυλουριες σαν αναστολεις της raf κινασης

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Publication number
CY2007002I1
CY2007002I1 CY200700002C CY2007002C CY2007002I1 CY 2007002 I1 CY2007002 I1 CY 2007002I1 CY 200700002 C CY200700002 C CY 200700002C CY 2007002 C CY2007002 C CY 2007002C CY 2007002 I1 CY2007002 I1 CY 2007002I1
Authority
CY
Cyprus
Prior art keywords
carboxyarylipocutated
bifinylureas
kinase inhibitors
raf kinase
raf
Prior art date
Application number
CY200700002C
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English (en)
Other versions
CY2007002I2 (el
Original Assignee
Bayer Pharmaceuticals Corporation
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=56290111&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY2007002(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Pharmaceuticals Corporation filed Critical Bayer Pharmaceuticals Corporation
Publication of CY2007002I1 publication Critical patent/CY2007002I1/el
Publication of CY2007002I2 publication Critical patent/CY2007002I2/el

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    • C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
    • C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C275/36—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring with at least one of the oxygen atoms further bound to a carbon atom of a six-membered aromatic ring, e.g. N-aryloxyphenylureas
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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CY200700002C 1999-01-13 2007-01-18 Ω-καρβοξυαρυλυποκατεστημενες διφαινυλουριες σαν αναστολεις της raf κινασης CY2007002I2 (el)

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US20010011136A1 (en) 2001-08-02
US20010016659A1 (en) 2001-08-23
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CY1105286T1 (el) 2010-03-03
US20020042517A1 (en) 2002-04-11
WO2000042012A1 (en) 2000-07-20
EP1140840B1 (en) 2006-03-22
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