ZA966044B - Crystalline [R-(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino) carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1). - Google Patents

Crystalline [R-(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino) carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1).

Info

Publication number
ZA966044B
ZA966044B ZA9606044A ZA966044A ZA966044B ZA 966044 B ZA966044 B ZA 966044B ZA 9606044 A ZA9606044 A ZA 9606044A ZA 966044 A ZA966044 A ZA 966044A ZA 966044 B ZA966044 B ZA 966044B
Authority
ZA
South Africa
Prior art keywords
phenylamino
methylethyl
fluorophenyl
pyrrole
dihydroxy
Prior art date
Application number
ZA9606044A
Other languages
English (en)
Inventor
Christopher A Briggs
Robert A Wade
Shigeru Ichikawa
Shinsuke Nakagawa
Rex Allen Jennings
Kikuko Harasawa
Kazuo Minohara
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21696090&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA966044(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of ZA966044B publication Critical patent/ZA966044B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ZA9606044A 1995-07-17 1996-07-16 Crystalline [R-(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino) carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1). ZA966044B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US145295P 1995-07-17 1995-07-17

Publications (1)

Publication Number Publication Date
ZA966044B true ZA966044B (en) 1997-02-03

Family

ID=21696090

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9606044A ZA966044B (en) 1995-07-17 1996-07-16 Crystalline [R-(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino) carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1).

Country Status (38)

Country Link
US (1) US5969156A (es)
EP (2) EP1148049B1 (es)
JP (4) JP3296564B2 (es)
KR (2) KR100431038B1 (es)
CN (1) CN1087288C (es)
AR (2) AR003459A1 (es)
AT (3) ATE208375T1 (es)
AU (1) AU725424B2 (es)
BG (1) BG63630B1 (es)
BR (1) BR9609872A (es)
CA (1) CA2220018C (es)
CO (1) CO4700443A1 (es)
CY (1) CY2358B1 (es)
CZ (3) CZ294695B6 (es)
DE (2) DE69616808T2 (es)
DK (2) DK0848705T3 (es)
EA (1) EA000474B1 (es)
EE (1) EE03606B1 (es)
ES (2) ES2233526T3 (es)
GE (1) GEP20002029B (es)
HK (1) HK1018052A1 (es)
HR (1) HRP960339B1 (es)
HU (1) HU223599B1 (es)
IL (7) IL128862A (es)
MX (1) MX9709099A (es)
NO (1) NO309898B1 (es)
NZ (1) NZ312907A (es)
PE (1) PE1898A1 (es)
PL (1) PL193479B1 (es)
PT (2) PT1148049E (es)
RO (1) RO120070B1 (es)
SI (2) SI1148049T1 (es)
SK (1) SK284202B6 (es)
TW (1) TW486467B (es)
UA (1) UA51661C2 (es)
UY (2) UY24285A1 (es)
WO (1) WO1997003959A1 (es)
ZA (1) ZA966044B (es)

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