UA77303C2 - Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use - Google Patents
Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use Download PDFInfo
- Publication number
- UA77303C2 UA77303C2 UA20041210250A UA20041210250A UA77303C2 UA 77303 C2 UA77303 C2 UA 77303C2 UA 20041210250 A UA20041210250 A UA 20041210250A UA 20041210250 A UA20041210250 A UA 20041210250A UA 77303 C2 UA77303 C2 UA 77303C2
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- UA
- Ukraine
- Prior art keywords
- alkyl
- compound
- aryl
- indole
- carboxylic acid
- Prior art date
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Ophthalmology & Optometry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US38911002P | 2002-06-14 | 2002-06-14 | |
PCT/IB2003/002393 WO2003106462A1 (en) | 2002-06-14 | 2003-06-04 | Benzofused heteroaryl amide derivatives of thienopyridines useful as therapeutic agents, pharmaceutical compositions including the same, and methods for their use |
Publications (1)
Publication Number | Publication Date |
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UA77303C2 true UA77303C2 (en) | 2006-11-15 |
Family
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Family Applications (1)
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UA20041210250A UA77303C2 (en) | 2002-06-14 | 2003-04-06 | Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use |
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US (3) | US6869962B2 (zh) |
EP (1) | EP1515975B1 (zh) |
JP (1) | JP2005534669A (zh) |
KR (2) | KR100714545B1 (zh) |
CN (1) | CN1671714A (zh) |
AP (1) | AP2004003184A0 (zh) |
AR (1) | AR039673A1 (zh) |
AT (1) | ATE373665T1 (zh) |
AU (1) | AU2003233134A1 (zh) |
BR (1) | BR0311806A (zh) |
CA (1) | CA2489466A1 (zh) |
CO (1) | CO5631447A2 (zh) |
DE (1) | DE60316440T2 (zh) |
EA (1) | EA008255B1 (zh) |
EC (1) | ECSP045483A (zh) |
ES (1) | ES2290460T3 (zh) |
GE (1) | GEP20074033B (zh) |
GT (1) | GT200300129A (zh) |
HN (1) | HN2003000182A (zh) |
HR (1) | HRP20041173A2 (zh) |
IL (1) | IL165591A0 (zh) |
IS (1) | IS7552A (zh) |
MA (1) | MA27596A1 (zh) |
MX (1) | MXPA04011637A (zh) |
NO (1) | NO20045103L (zh) |
NZ (1) | NZ537140A (zh) |
OA (1) | OA12865A (zh) |
PA (1) | PA8575401A1 (zh) |
PE (1) | PE20050123A1 (zh) |
PL (1) | PL374542A1 (zh) |
RS (1) | RS107504A (zh) |
TN (1) | TNSN04246A1 (zh) |
TW (1) | TW200404070A (zh) |
UA (1) | UA77303C2 (zh) |
WO (1) | WO2003106462A1 (zh) |
ZA (1) | ZA200409862B (zh) |
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2003
- 2003-04-06 UA UA20041210250A patent/UA77303C2/uk unknown
- 2003-06-04 KR KR1020067019988A patent/KR100714545B1/ko not_active IP Right Cessation
- 2003-06-04 MX MXPA04011637A patent/MXPA04011637A/es unknown
- 2003-06-04 NZ NZ537140A patent/NZ537140A/en unknown
- 2003-06-04 EP EP03727888A patent/EP1515975B1/en not_active Expired - Lifetime
- 2003-06-04 CN CNA038181096A patent/CN1671714A/zh active Pending
- 2003-06-04 AT AT03727888T patent/ATE373665T1/de not_active IP Right Cessation
- 2003-06-04 RS YU107504A patent/RS107504A/sr unknown
- 2003-06-04 JP JP2004513293A patent/JP2005534669A/ja not_active Withdrawn
- 2003-06-04 ES ES03727888T patent/ES2290460T3/es not_active Expired - Lifetime
- 2003-06-04 EA EA200500018A patent/EA008255B1/ru unknown
- 2003-06-04 BR BR0311806-1A patent/BR0311806A/pt not_active IP Right Cessation
- 2003-06-04 WO PCT/IB2003/002393 patent/WO2003106462A1/en active IP Right Grant
- 2003-06-04 CA CA002489466A patent/CA2489466A1/en not_active Abandoned
- 2003-06-04 AU AU2003233134A patent/AU2003233134A1/en not_active Abandoned
- 2003-06-04 AP AP2004003184A patent/AP2004003184A0/xx unknown
- 2003-06-04 KR KR1020047020286A patent/KR100671632B1/ko not_active IP Right Cessation
- 2003-06-04 OA OA1200400325A patent/OA12865A/en unknown
- 2003-06-04 PL PL03374542A patent/PL374542A1/xx not_active Application Discontinuation
- 2003-06-04 GE GEAP8535A patent/GEP20074033B/en unknown
- 2003-06-04 DE DE60316440T patent/DE60316440T2/de not_active Expired - Fee Related
- 2003-06-11 PE PE2003000579A patent/PE20050123A1/es not_active Application Discontinuation
- 2003-06-11 US US10/460,010 patent/US6869962B2/en not_active Expired - Fee Related
- 2003-06-12 PA PA20038575401A patent/PA8575401A1/es unknown
- 2003-06-12 GT GT200300129A patent/GT200300129A/es unknown
- 2003-06-13 AR ARP030102121A patent/AR039673A1/es not_active Application Discontinuation
- 2003-06-13 TW TW092116098A patent/TW200404070A/zh unknown
- 2003-06-13 HN HN2003000182A patent/HN2003000182A/es unknown
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2004
- 2004-03-09 US US10/796,226 patent/US7045528B2/en not_active Expired - Fee Related
- 2004-11-24 NO NO20045103A patent/NO20045103L/no not_active Application Discontinuation
- 2004-11-25 IS IS7552A patent/IS7552A/is unknown
- 2004-12-06 IL IL16559104A patent/IL165591A0/xx unknown
- 2004-12-06 ZA ZA200409862A patent/ZA200409862B/xx unknown
- 2004-12-08 MA MA27986A patent/MA27596A1/fr unknown
- 2004-12-09 CO CO04123221A patent/CO5631447A2/es not_active Application Discontinuation
- 2004-12-09 HR HR20041173A patent/HRP20041173A2/hr not_active Application Discontinuation
- 2004-12-09 EC EC2004005483A patent/ECSP045483A/es unknown
- 2004-12-13 TN TNP2004000246A patent/TNSN04246A1/fr unknown
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2005
- 2005-10-21 US US11/256,477 patent/US20060079548A1/en not_active Abandoned
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