TW201932456A - 適用作pim激酶抑制劑之噻唑甲醯胺及吡啶甲醯胺化合物 - Google Patents

適用作pim激酶抑制劑之噻唑甲醯胺及吡啶甲醯胺化合物 Download PDF

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TW201932456A
TW201932456A TW108116840A TW108116840A TW201932456A TW 201932456 A TW201932456 A TW 201932456A TW 108116840 A TW108116840 A TW 108116840A TW 108116840 A TW108116840 A TW 108116840A TW 201932456 A TW201932456 A TW 201932456A
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Taiwan
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amino
pyridin
carboxamide
compound
pharmaceutically acceptable
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TW108116840A
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English (en)
Chinese (zh)
Inventor
楚標 薛
裕隆 李
馮皓
淳 潘
王安來
克 張
文清 姚
張豐雷
金聰 卓
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美商英塞特控股公司
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Publication of TW201932456A publication Critical patent/TW201932456A/zh

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4355—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having oxygen as a ring hetero atom
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TW108116840A 2013-01-15 2014-01-14 適用作pim激酶抑制劑之噻唑甲醯胺及吡啶甲醯胺化合物 TW201932456A (zh)

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US201361752897P 2013-01-15 2013-01-15
US61/752,897 2013-01-15
US201361790952P 2013-03-15 2013-03-15
US61/790,952 2013-03-15
US201361859118P 2013-07-26 2013-07-26
US61/859,118 2013-07-26

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TW103101314A TWI662030B (zh) 2013-01-15 2014-01-14 適用作ｐｉｍ激酶抑制劑之噻唑甲醯胺及吡啶甲醯胺化合物

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