TR199900389T2 - �kame edilmi� 6,5-hetero-bisiklik t�revleri. - Google Patents
�kame edilmi� 6,5-hetero-bisiklik t�revleri.Info
- Publication number
- TR199900389T2 TR199900389T2 TR1999/00389T TR9900389T TR199900389T2 TR 199900389 T2 TR199900389 T2 TR 199900389T2 TR 1999/00389 T TR1999/00389 T TR 1999/00389T TR 9900389 T TR9900389 T TR 9900389T TR 199900389 T2 TR199900389 T2 TR 199900389T2
- Authority
- TR
- Turkey
- Prior art keywords
- nitrogen
- hetero
- substituted
- carbon
- formula
- Prior art date
Links
- IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 10
- 229910052757 nitrogen Inorganic materials 0.000 abstract 5
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 2
- 229910052799 carbon Inorganic materials 0.000 abstract 2
- -1 C = S Chemical compound 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 230000003042 antagnostic effect Effects 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 239000011593 sulfur Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Addiction (AREA)
- Endocrinology (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychiatry (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Cardiology (AREA)
- Rheumatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Reproductive Health (AREA)
- Obesity (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Communicable Diseases (AREA)
- Psychology (AREA)
- Oncology (AREA)
- Pregnancy & Childbirth (AREA)
- Virology (AREA)
- Gynecology & Obstetrics (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2503996P | 1996-08-28 | 1996-08-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR199900389T2 true TR199900389T2 (xx) | 2000-06-21 |
Family
ID=21823717
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR1999/00389T TR199900389T2 (xx) | 1996-08-28 | 1997-07-25 | �kame edilmi� 6,5-hetero-bisiklik t�revleri. |
Country Status (36)
Families Citing this family (152)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH10506126A (ja) | 1995-05-12 | 1998-06-16 | ニューロゲン コーポレイション | 新規なデアザプリン誘導体;crf1特異性リガンドの新規なクラス |
| US6313124B1 (en) | 1997-07-23 | 2001-11-06 | Dupont Pharmaceuticals Company | Tetrazine bicyclic compounds |
| US6124289A (en) * | 1996-07-24 | 2000-09-26 | Dupont Pharmaceuticals Co. | Azolo triazines and pyrimidines |
| US6191131B1 (en) | 1997-07-23 | 2001-02-20 | Dupont Pharmaceuticals Company | Azolo triazines and pyrimidines |
| US6060478A (en) * | 1996-07-24 | 2000-05-09 | Dupont Pharmaceuticals | Azolo triazines and pyrimidines |
| US7094782B1 (en) | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
| JP2001511813A (ja) | 1997-02-18 | 2001-08-14 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | Crfレセプターアンタゴニストおよびそれらに関連する方法 |
| NZ335823A (en) | 1997-04-22 | 2001-06-29 | Neurocrine Biosciences Inc | Thiophenopyridines, preparation as CRF receptor antagonists |
| JP2002507996A (ja) * | 1997-07-03 | 2002-03-12 | デュポン ファーマシューティカルズ カンパニー | 神経学的障害を治療するためのイミダゾピリミジン類およびイミダゾピリジン類 |
| IL137019A0 (en) * | 1998-01-28 | 2001-06-14 | Du Pont Pharm Co | Azolo triazines and pyrimidines |
| US6187777B1 (en) * | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
| EP1068205A1 (en) | 1998-04-02 | 2001-01-17 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-tetrahydro-9h pyrimidino 2,3-b]indole and 5,6,7,8-tetrahydro-9h-pyrimidino 4,5-b]indole derivatives: crf1 specific ligands |
| US6472402B1 (en) | 1998-04-02 | 2002-10-29 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives |
| WO1999051608A1 (en) * | 1998-04-03 | 1999-10-14 | Du Pont Pharmaceuticals Company | THIAZOLO[4,5-d]PYRIMIDINES AND PYRIDINES AS CORTICOTROPIN RELEASING FACTOR (CRF) ANTAGONISTS |
| AU4556999A (en) * | 1998-06-09 | 1999-12-30 | Neurogen Corporation | Pyrido[2,3-b]indolizine derivatives and aza analogues thereof; crf1 specific ligands |
| US6509338B1 (en) | 1998-06-22 | 2003-01-21 | Bristol-Myers Squibb Company | Pyrazolo[1,5-A]triazine corticotropin releasing factor antagonists |
| CA2339188A1 (en) * | 1998-08-21 | 2000-03-02 | Dupont Pharmaceuticals Company | Isoxazolo¬4,5-d|pyrimidines as crf antagonists |
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- 1997-07-25 PL PL97332040A patent/PL332040A1/xx unknown
- 1997-07-25 DE DE69736711T patent/DE69736711T2/de not_active Expired - Fee Related
- 1997-07-25 CZ CZ99681A patent/CZ68199A3/cs unknown
- 1997-07-25 SK SK233-99A patent/SK23399A3/sk unknown
- 1997-07-25 CA CA002263566A patent/CA2263566C/en not_active Expired - Fee Related
- 1997-07-25 NZ NZ333302A patent/NZ333302A/xx unknown
- 1997-07-25 AT AT97930697T patent/ATE340176T1/de not_active IP Right Cessation
- 1997-07-25 EA EA199900165A patent/EA002769B1/ru not_active IP Right Cessation
- 1997-07-25 ES ES97930697T patent/ES2273369T3/es not_active Expired - Lifetime
- 1997-07-25 JP JP51142998A patent/JP3621706B2/ja not_active Expired - Fee Related
- 1997-07-25 AU AU34561/97A patent/AU735401B2/en not_active Ceased
- 1997-07-25 TR TR1999/00389T patent/TR199900389T2/xx unknown
- 1997-07-25 BR BR9711970A patent/BR9711970A/pt not_active Application Discontinuation
- 1997-07-25 HU HU9903965A patent/HUP9903965A3/hu unknown
- 1997-07-25 EP EP97930697A patent/EP0923582B1/en not_active Revoked
- 1997-07-25 IL IL12756697A patent/IL127566A0/xx unknown
- 1997-07-25 WO PCT/IB1997/000922 patent/WO1998008847A1/en not_active Ceased
- 1997-07-25 KR KR1019997001674A patent/KR20000035934A/ko not_active Ceased
- 1997-07-25 CN CN97197027A patent/CN1227554A/zh active Pending
- 1997-08-12 PA PA19978436201A patent/PA8436201A1/es unknown
- 1997-08-21 AP APAP/P/1997/001077A patent/AP762A/en active
- 1997-08-22 HR HR970454A patent/HRP970454B1/xx not_active IP Right Cessation
- 1997-08-25 TW TW086112194A patent/TW575573B/zh active
- 1997-08-25 PE PE1997000756A patent/PE108898A1/es not_active Application Discontinuation
- 1997-08-25 GT GT199700095A patent/GT199700095A/es unknown
- 1997-08-26 AR ARP970103861A patent/AR015103A1/es not_active Application Discontinuation
- 1997-08-26 ID IDP972962A patent/ID18249A/id unknown
- 1997-08-27 DZ DZ970150A patent/DZ2300A1/fr active
- 1997-08-27 TN TNTNSN97145A patent/TNSN97145A1/fr unknown
- 1997-08-27 MA MA24779A patent/MA26438A1/fr unknown
- 1997-08-27 ZA ZA977687A patent/ZA977687B/xx unknown
- 1997-08-28 CO CO97049895A patent/CO4600634A1/es unknown
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1999
- 1999-01-29 IS IS4963A patent/IS4963A/is unknown
- 1999-02-17 OA OA9900035A patent/OA10977A/en unknown
- 1999-02-22 BG BG103189A patent/BG103189A/xx unknown
- 1999-02-26 NO NO19990927A patent/NO313636B1/no not_active IP Right Cessation
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2004
- 2004-09-21 JP JP2004273978A patent/JP2005047930A/ja not_active Withdrawn
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