RU2056425C1 - Производные цефалоспорина или их фармацевтически приемлемые кислотно-аддитивные соли и способы их получения - Google Patents

Производные цефалоспорина или их фармацевтически приемлемые кислотно-аддитивные соли и способы их получения Download PDF

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RU2056425C1
RU2056425C1 SU853878102A SU3878102A RU2056425C1 RU 2056425 C1 RU2056425 C1 RU 2056425C1 SU 853878102 A SU853878102 A SU 853878102A SU 3878102 A SU3878102 A SU 3878102A RU 2056425 C1 RU2056425 C1 RU 2056425C1
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Russia
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amino
doublet
mixture
max
group
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SU853878102A
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English (en)
Russian (ru)
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Ока Масахиса
Ямасита Харухиро
Наито Такаюки
Окумура Юн
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Бристоль-Мейерз Компани
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/08—1,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/78—Separation; Purification; Stabilisation; Use of additives
    • C07C45/79—Separation; Purification; Stabilisation; Use of additives by solid-liquid treatment; by chemisorption

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SU853878102A 1984-04-09 1985-04-08 Производные цефалоспорина или их фармацевтически приемлемые кислотно-аддитивные соли и способы их получения RU2056425C1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59794184A 1984-04-09 1984-04-09
US597941 1984-04-09

Publications (1)

Publication Number Publication Date
RU2056425C1 true RU2056425C1 (ru) 1996-03-20

Family

ID=24393575

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Application Number Title Priority Date Filing Date
SU853878102A RU2056425C1 (ru) 1984-04-09 1985-04-08 Производные цефалоспорина или их фармацевтически приемлемые кислотно-аддитивные соли и способы их получения

Country Status (31)

Country Link
JP (4) JPS615084A (xx)
KR (1) KR870002166B1 (xx)
AR (1) AR244694A1 (xx)
AT (1) AT388735B (xx)
AU (2) AU580990B2 (xx)
BE (1) BE902148A (xx)
CA (3) CA1276929C (xx)
CH (1) CH669197A5 (xx)
DD (3) DD249024A5 (xx)
DE (1) DE3512225A1 (xx)
DK (1) DK155985A (xx)
ES (4) ES8607318A1 (xx)
FI (1) FI84830C (xx)
FR (1) FR2563832B1 (xx)
GB (3) GB2157293B (xx)
GR (1) GR850883B (xx)
HU (2) HU204277B (xx)
IE (2) IE58408B1 (xx)
IL (1) IL74826A (xx)
IT (1) IT1190353B (xx)
LU (1) LU85840A1 (xx)
MY (1) MY101940A (xx)
NL (1) NL192925C (xx)
NZ (1) NZ211659A (xx)
OA (1) OA07985A (xx)
PT (1) PT80246B (xx)
RU (1) RU2056425C1 (xx)
SE (4) SE466205B (xx)
SU (4) SU1436882A3 (xx)
YU (2) YU46151B (xx)
ZA (1) ZA852236B (xx)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS61145186A (ja) * 1984-12-20 1986-07-02 Meiji Seika Kaisha Ltd 新規セフエム化合物及びその製造法
US4708955A (en) * 1985-06-24 1987-11-24 Bristol-Myers Company 3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof
ATE114657T1 (de) * 1985-12-26 1994-12-15 Eisai Co Ltd Cephalosporin-verbindungen.
AU614723B2 (en) * 1986-10-13 1991-09-12 Eisai Co. Ltd. 3-propenylcephem derivative
IL84128A (en) * 1986-10-13 1992-12-01 Eisai Co Ltd 3-propenylcephem derivatives, their preparation and pharmaceutical compositions containing them
JPH085897B2 (ja) * 1986-11-06 1996-01-24 エーザイ株式会社 ３−プロペニルセフェム誘導体
FR2622585B1 (fr) * 1987-11-03 1991-04-19 Roussel Uclaf Nouvelles cephalosporines comportant en position 3 un radical vinyle substitue, leur procede de preparation, leur application comme medicaments, les compositions les renfermant et les nouveaux intermediaires obtenus
CA1339738C (en) * 1988-03-16 1998-03-17 Takashi Kamiya Process for the preparation of cephem derivatives and entermediates therefor
JPH0699449B2 (ja) * 1988-03-16 1994-12-07 エーザイ株式会社 セフェム誘導体の合成中間体
FR2655042B1 (fr) * 1989-11-29 1994-01-21 Adir Cie Nouvelles benzothiazolinones substituees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
FR2663332B1 (fr) * 1990-06-15 1997-11-07 Roussel Uclaf Nouvelles cephalosporines comportant en position 3 un radical propenyle substitue par un ammonium quaternaire, leur procede de preparation, leur application comme medicaments, les compositions les renfermant et les nouveaux intermediaires obtenus.
US5126336A (en) * 1990-08-23 1992-06-30 Bristol-Myers Squibb Company Antibiotic c-3 catechol-substituted cephalosporin compounds, compositions and method of use thereof
AT396108B (de) * 1991-08-21 1993-06-25 Biochemie Gmbh Neues verfahren und neue zwischenprodukte zur herstellung von 7-aminocephalosporansaeurederivaten
JPH0741484A (ja) * 1993-07-29 1995-02-10 Katayama Seiyakushiyo:Kk セフェム化合物及び抗菌剤
KR100248851B1 (ko) * 1994-08-16 2000-04-01 이치로 키타사토 신규 세펨 유도체
WO1999067255A1 (en) 1998-06-22 1999-12-29 F. Hoffmann-La Roche Ag Propenyl cephalosporin derivatives
WO2005026176A1 (ja) 2003-09-09 2005-03-24 Nippon Chemical Industrial Co.,Ltd. ３−クロロメチル-３-セフェム誘導体の製造方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1342241A (en) * 1970-01-23 1974-01-03 Glaxo Lab Ltd Cephalosporin compounds
US4390534A (en) * 1978-12-29 1983-06-28 Fujisawa Pharmaceutical Co., Ltd. Cephem and cepham compounds
EP0025017A1 (de) * 1979-08-28 1981-03-11 Ciba-Geigy Ag Polyazathiaverbindungen, Verfahren zu ihrer Herstellung, pharmazeutische Präparate enthaltend solche Verbindungen und Verwendung von letzteren
US4409214A (en) * 1979-11-19 1983-10-11 Fujisawa Pharmaceutical, Co., Ltd. 7-Acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
GR75644B (xx) * 1980-06-18 1984-08-02 Fujisawa Pharmaceutical Co
GR78245B (xx) * 1980-09-12 1984-09-26 Ciba Geigy Ag
US4521413A (en) * 1981-09-14 1985-06-04 Fujisawa Pharmaceutical Co., Ltd. Cephem compounds
US4486586A (en) * 1983-02-10 1984-12-04 Bristol-Myers Company Cephalosporin derivatives

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
1. Европейская заявка N 0062321, кл. C 07D 501/46, 1982. 2. Европейская заявка N 0074653, кл. C 07D 501/46, 1983. 3. Заявка Японии Kokai N 57-112396, кл. C 07D 501/46, 1982. *

Also Published As

Publication number Publication date
ES8706694A1 (es) 1987-07-01
GR850883B (xx) 1985-11-25
NZ211659A (en) 1988-11-29
IL74826A (en) 1990-01-18
SE8501680D0 (sv) 1985-04-03
JPS61143387A (ja) 1986-07-01
GB2157293B (en) 1988-10-05
AU610278B2 (en) 1991-05-16
JPS61143391A (ja) 1986-07-01
IE58408B1 (en) 1993-09-22
JPS615084A (ja) 1986-01-10
JPH0351716B2 (xx) 1991-08-07
ES8706155A1 (es) 1987-06-01
FI84830C (fi) 1992-01-27
AT388735B (de) 1989-08-25
NL192925C (nl) 1998-05-07
JPH0262557B2 (xx) 1990-12-26
JPH0357106B2 (xx) 1991-08-30
AR244694A1 (es) 1993-11-30
KR850007424A (ko) 1985-12-04
SE8901226D0 (sv) 1989-04-06
SE466205B (sv) 1992-01-13
AU4086285A (en) 1985-10-17
YU60085A (en) 1987-12-31
NL192925B (nl) 1998-01-05
ES551550A0 (es) 1987-06-01
ES551551A0 (es) 1987-07-01
CH669197A5 (de) 1989-02-28
CA1340638C (en) 1999-07-06
ES8607318A1 (es) 1986-06-16
GB2194789A (en) 1988-03-16
SE8901224L (sv) 1989-04-06
IL74826A0 (en) 1985-07-31
IT8520267A0 (it) 1985-04-05
OA07985A (fr) 1987-01-31
GB2194790A (en) 1988-03-16
SE8901225L (sv) 1989-04-06
FI84830B (fi) 1991-10-15
GB2157293A (en) 1985-10-23
SE8901224D0 (sv) 1989-04-06
HUT37622A (en) 1986-01-23
ATA103985A (de) 1989-01-15
HU204277B (en) 1991-12-30
IE58403B1 (en) 1993-09-22
GB2194790B (en) 1988-10-05
ES8800949A1 (es) 1987-12-01
DD249024A5 (de) 1987-08-26
DD236735A5 (de) 1986-06-18
SE8901226L (sv) 1989-04-06
YU118987A (en) 1988-10-31
FR2563832A1 (fr) 1985-11-08
MY101940A (en) 1992-02-15
GB8508846D0 (en) 1985-05-09
DK155985D0 (da) 1985-04-03
JPS61143390A (ja) 1986-07-01
BE902148A (fr) 1985-10-09
SE470259B (sv) 1993-12-20
HU193750B (en) 1987-11-30
FI851379L (fi) 1985-10-10
AU580990B2 (en) 1989-02-09
NL8501002A (nl) 1985-11-01
ES557060A0 (es) 1987-12-01
GB8721347D0 (en) 1987-10-14
SU1375140A3 (ru) 1988-02-15
GB8721346D0 (en) 1987-10-14
DE3512225C2 (xx) 1990-02-22
LU85840A1 (fr) 1985-12-16
KR870002166B1 (ko) 1987-12-14
YU46213B (sh) 1993-05-28
GB2194789B (en) 1988-10-12
CA1276929C (en) 1990-11-27
ZA852236B (en) 1985-11-27
DK155985A (da) 1985-10-10
SE470260B (sv) 1993-12-20
SU1367858A3 (ru) 1988-01-15
FI851379A0 (fi) 1985-04-04
PT80246B (pt) 1987-10-20
FR2563832B1 (fr) 1989-08-18
YU46151B (sh) 1993-05-28
IE850866L (en) 1985-10-09
SE8501680L (sv) 1985-10-10
AU2504188A (en) 1989-03-02
SU1436882A3 (ru) 1988-11-07
IT1190353B (it) 1988-02-16
DD251752A5 (de) 1987-11-25
SE505256C2 (sv) 1997-07-21
JPH0350754B2 (xx) 1991-08-02
ES542013A0 (es) 1986-06-16
SU1487814A3 (ru) 1989-06-15
PT80246A (en) 1985-05-01
DE3512225A1 (de) 1985-10-17
CA1340672C (en) 1999-07-20
SE8901225D0 (sv) 1989-04-06

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