ATE114657T1 - Cephalosporin-verbindungen. - Google Patents
Cephalosporin-verbindungen.Info
- Publication number
- ATE114657T1 ATE114657T1 AT87900286T AT87900286T ATE114657T1 AT E114657 T1 ATE114657 T1 AT E114657T1 AT 87900286 T AT87900286 T AT 87900286T AT 87900286 T AT87900286 T AT 87900286T AT E114657 T1 ATE114657 T1 AT E114657T1
- Authority
- AT
- Austria
- Prior art keywords
- lower alkyl
- carbamoyl
- amino
- substd
- carboxy
- Prior art date
Links
- -1 CEPHALOSPORIN COMPOUNDS Chemical class 0.000 title abstract 3
- 229930186147 Cephalosporin Natural products 0.000 title abstract 2
- 229940124587 cephalosporin Drugs 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 6
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 3
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 2
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 2
- IKWLIQXIPRUIDU-ZCFIWIBFSA-N (6r)-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid Chemical compound OC(=O)C1=CCS[C@@H]2CC(=O)N12 IKWLIQXIPRUIDU-ZCFIWIBFSA-N 0.000 abstract 1
- 125000003282 alkyl amino group Chemical group 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 150000001780 cephalosporins Chemical class 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 238000010511 deprotection reaction Methods 0.000 abstract 1
- 125000004005 formimidoyl group Chemical group [H]\N=C(/[H])* 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000003396 thiol group Chemical class [H]S* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP29183685 | 1985-12-26 | ||
| JP61037449A JPH0717654B2 (ja) | 1986-02-24 | 1986-02-24 | ７−チアジアゾリルアセトアミド−３−セフエム誘導体 |
| JP61233356A JPS6388187A (ja) | 1986-10-02 | 1986-10-02 | ３−アンモニオプロペニルセフエム誘導体 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE114657T1 true ATE114657T1 (de) | 1994-12-15 |
Family
ID=27289474
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT87900286T ATE114657T1 (de) | 1985-12-26 | 1986-12-26 | Cephalosporin-verbindungen. |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP0329785B1 (de) |
| AT (1) | ATE114657T1 (de) |
| DE (1) | DE3650157T2 (de) |
| WO (1) | WO1987003875A1 (de) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5373000A (en) * | 1985-12-26 | 1994-12-13 | Eisai Co., Ltd. | 7Beta-(thiadiazolyl)-2-iminoacetamido-3cephem compounds |
| DE68928174T2 (de) * | 1988-03-16 | 1997-12-18 | Eisai Co., Ltd., Tokio/Tokyo | Verfahren zur Herstellung von Cephemderivaten |
| FR2663332B1 (fr) * | 1990-06-15 | 1997-11-07 | Roussel Uclaf | Nouvelles cephalosporines comportant en position 3 un radical propenyle substitue par un ammonium quaternaire, leur procede de preparation, leur application comme medicaments, les compositions les renfermant et les nouveaux intermediaires obtenus. |
| US5143911A (en) * | 1990-08-23 | 1992-09-01 | Bristol-Myers Squibb Company | Antibiotic c-3 di-hydroxyphenyl substituted cephalosporin compounds, compositions and method of use thereof |
| US5126336A (en) * | 1990-08-23 | 1992-06-30 | Bristol-Myers Squibb Company | Antibiotic c-3 catechol-substituted cephalosporin compounds, compositions and method of use thereof |
| AT396108B (de) * | 1991-08-21 | 1993-06-25 | Biochemie Gmbh | Neues verfahren und neue zwischenprodukte zur herstellung von 7-aminocephalosporansaeurederivaten |
| JPH07173168A (ja) * | 1993-07-14 | 1995-07-11 | Sumitomo Chem Co Ltd | セフェム系化合物、その製法、およびそれのセフェム系抗生物質製造への利用 |
| KR100248851B1 (ko) * | 1994-08-16 | 2000-04-01 | 이치로 키타사토 | 신규 세펨 유도체 |
| KR0174117B1 (ko) * | 1995-12-28 | 1999-02-01 | 윤원영 | 새로운 세팔로스포린 유도체 및 그 제조방법 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3247613A1 (de) * | 1982-12-23 | 1984-07-05 | Hoechst Ag, 6230 Frankfurt | Cephalosporinderivate und verfahren zu ihrer herstellung |
| US4486586A (en) * | 1983-02-10 | 1984-12-04 | Bristol-Myers Company | Cephalosporin derivatives |
| CA1276929C (en) * | 1984-04-09 | 1990-11-27 | Masahisa Oka | Cephalosporin antibacterial agents |
| JPH0697983A (ja) * | 1992-09-10 | 1994-04-08 | Toshiba Corp | ネットワークシステム |
-
1986
- 1986-12-26 WO PCT/JP1986/000655 patent/WO1987003875A1/ja not_active Ceased
- 1986-12-26 EP EP87900286A patent/EP0329785B1/de not_active Expired - Lifetime
- 1986-12-26 DE DE3650157T patent/DE3650157T2/de not_active Expired - Fee Related
- 1986-12-26 AT AT87900286T patent/ATE114657T1/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| EP0329785A4 (de) | 1990-02-06 |
| DE3650157D1 (de) | 1995-01-12 |
| EP0329785A1 (de) | 1989-08-30 |
| EP0329785B1 (de) | 1994-11-30 |
| DE3650157T2 (de) | 1995-05-04 |
| WO1987003875A1 (fr) | 1987-07-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |