OA10977A - Substituted 6,5-hetero-bicyclic derivatives - Google Patents
Substituted 6,5-hetero-bicyclic derivatives Download PDFInfo
- Publication number
- OA10977A OA10977A OA9900035A OA9900035A OA10977A OA 10977 A OA10977 A OA 10977A OA 9900035 A OA9900035 A OA 9900035A OA 9900035 A OA9900035 A OA 9900035A OA 10977 A OA10977 A OA 10977A
- Authority
- OA
- OAPI
- Prior art keywords
- phenyl
- trimethyl
- stress
- compounds
- ethyl
- Prior art date
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P11/06—Antiasthmatics
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2503996P | 1996-08-28 | 1996-08-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
OA10977A true OA10977A (en) | 2001-11-02 |
Family
ID=21823717
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
OA9900035A OA10977A (en) | 1996-08-28 | 1999-02-17 | Substituted 6,5-hetero-bicyclic derivatives |
Country Status (36)
Country | Link |
---|---|
EP (1) | EP0923582B1 (es) |
JP (2) | JP3621706B2 (es) |
KR (1) | KR20000035934A (es) |
CN (1) | CN1227554A (es) |
AP (1) | AP762A (es) |
AR (1) | AR015103A1 (es) |
AT (1) | ATE340176T1 (es) |
AU (1) | AU735401B2 (es) |
BG (1) | BG103189A (es) |
BR (1) | BR9711970A (es) |
CA (1) | CA2263566C (es) |
CO (1) | CO4600634A1 (es) |
CZ (1) | CZ68199A3 (es) |
DE (1) | DE69736711T2 (es) |
DZ (1) | DZ2300A1 (es) |
EA (1) | EA002769B1 (es) |
ES (1) | ES2273369T3 (es) |
GT (1) | GT199700095A (es) |
HR (1) | HRP970454B1 (es) |
HU (1) | HUP9903965A3 (es) |
ID (1) | ID18249A (es) |
IL (1) | IL127566A0 (es) |
IS (1) | IS4963A (es) |
MA (1) | MA26438A1 (es) |
NO (1) | NO313636B1 (es) |
NZ (1) | NZ333302A (es) |
OA (1) | OA10977A (es) |
PA (1) | PA8436201A1 (es) |
PE (1) | PE108898A1 (es) |
PL (1) | PL332040A1 (es) |
SK (1) | SK23399A3 (es) |
TN (1) | TNSN97145A1 (es) |
TR (1) | TR199900389T2 (es) |
TW (1) | TW575573B (es) |
WO (1) | WO1998008847A1 (es) |
ZA (1) | ZA977687B (es) |
Families Citing this family (147)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE182148T1 (de) | 1995-05-12 | 1999-07-15 | Neurogen Corp | Neue deazapurinderivate; eine neue klasse von crf1-spezifischen liganden |
US7094782B1 (en) | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
US6191131B1 (en) | 1997-07-23 | 2001-02-20 | Dupont Pharmaceuticals Company | Azolo triazines and pyrimidines |
US6060478A (en) * | 1996-07-24 | 2000-05-09 | Dupont Pharmaceuticals | Azolo triazines and pyrimidines |
US6124289A (en) * | 1996-07-24 | 2000-09-26 | Dupont Pharmaceuticals Co. | Azolo triazines and pyrimidines |
US6313124B1 (en) | 1997-07-23 | 2001-11-06 | Dupont Pharmaceuticals Company | Tetrazine bicyclic compounds |
AU6279598A (en) | 1997-02-18 | 1998-09-08 | Neurocrine Biosciences, Inc. | Biazacyclic CRF antagonists |
US6211195B1 (en) | 1997-04-22 | 2001-04-03 | Neurocrine Biosciences, Inc. | CRF antagonistic thiophenopyridines |
SK179899A3 (en) | 1997-07-03 | 2001-12-03 | Du Pont Pharm Co | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
JP4228332B2 (ja) * | 1998-01-28 | 2009-02-25 | ブリストル−マイヤーズ スクイブ ファーマ カンパニー | アゾロトリアジン類およびアゾロピリミジン類 |
US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
US6472402B1 (en) | 1998-04-02 | 2002-10-29 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives |
WO1999051597A1 (en) | 1998-04-02 | 1999-10-14 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-tetrahydro-9h pyrimidino[2,3-b]indole and 5,6,7,8-tetrahydro-9h-pyrimidino[4,5-b]indole derivatives: crf1 specific ligands |
AU3213699A (en) * | 1998-04-03 | 1999-10-25 | Du Pont Pharmaceuticals Company | Thiazolo(4,5-d)pyrimidines and pyridines as corticotropin releasing factor (CRF)antagonists |
EP1086103B1 (en) | 1998-06-09 | 2003-05-02 | Neurogen Corporation | Pyrido 2,3-b]indolizine derivatives and aza analogues thereof; crf 1 specific ligands |
US6509338B1 (en) | 1998-06-22 | 2003-01-21 | Bristol-Myers Squibb Company | Pyrazolo[1,5-A]triazine corticotropin releasing factor antagonists |
EP1105394A1 (en) * | 1998-08-21 | 2001-06-13 | Du Pont Pharmaceuticals Company | ISOXAZOLO 4,5-d]PYRIMIDINES AS CRF ANTAGONISTS |
US6531475B1 (en) * | 1998-11-12 | 2003-03-11 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods relating thereto |
DE69903333T2 (de) * | 1998-11-12 | 2003-08-07 | Neurocrine Biosciences Inc | Crf rezeptor-antagonisten und darauf bezogene methoden |
DK1129096T3 (da) | 1998-11-12 | 2003-09-15 | Neurocrine Biosciences Inc | CRF-receptorantagonister og fremgangsmåder, der er relateret dertil |
WO2000044754A1 (fr) * | 1999-01-29 | 2000-08-03 | Sumitomo Chemical Company, Limited | Agents inhibiteurs d'accumulation de graisse |
EP1040831A3 (en) * | 1999-04-02 | 2003-05-02 | Pfizer Products Inc. | Use of corticotropin releasing factor (CRF) antagonists to prevent sudden death |
WO2000059908A2 (en) * | 1999-04-06 | 2000-10-12 | Du Pont Pharmaceuticals Company | Pyrazolopyrimidines as crf antagonists |
AU4331500A (en) | 1999-04-06 | 2000-10-23 | Du Pont Pharmaceuticals Company | Pyrazolotriazines as crf antagonists |
US6982265B1 (en) | 1999-05-21 | 2006-01-03 | Bristol Myers Squibb Company | Pyrrolotriazine inhibitors of kinases |
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