AP762A - Substituted 6,5-hetero-bicyclic derivatives. - Google Patents
Substituted 6,5-hetero-bicyclic derivatives. Download PDFInfo
- Publication number
- AP762A AP762A APAP/P/1997/001077A AP9701077A AP762A AP 762 A AP762 A AP 762A AP 9701077 A AP9701077 A AP 9701077A AP 762 A AP762 A AP 762A
- Authority
- AP
- ARIPO
- Prior art keywords
- alkyl
- phenyl
- trimethyl
- methyl
- ethyl
- Prior art date
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
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- Public Health (AREA)
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- Biomedical Technology (AREA)
- Diabetes (AREA)
- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Addiction (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Reproductive Health (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Pulmonology (AREA)
- Virology (AREA)
- Pregnancy & Childbirth (AREA)
- Gynecology & Obstetrics (AREA)
- Dermatology (AREA)
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2503996P | 1996-08-28 | 1996-08-28 |
Publications (2)
Publication Number | Publication Date |
---|---|
AP9701077A0 AP9701077A0 (en) | 1997-10-31 |
AP762A true AP762A (en) | 1999-09-13 |
Family
ID=21823717
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
APAP/P/1997/001077A AP762A (en) | 1996-08-28 | 1997-08-21 | Substituted 6,5-hetero-bicyclic derivatives. |
Country Status (36)
Country | Link |
---|---|
EP (1) | EP0923582B1 (es) |
JP (2) | JP3621706B2 (es) |
KR (1) | KR20000035934A (es) |
CN (1) | CN1227554A (es) |
AP (1) | AP762A (es) |
AR (1) | AR015103A1 (es) |
AT (1) | ATE340176T1 (es) |
AU (1) | AU735401B2 (es) |
BG (1) | BG103189A (es) |
BR (1) | BR9711970A (es) |
CA (1) | CA2263566C (es) |
CO (1) | CO4600634A1 (es) |
CZ (1) | CZ68199A3 (es) |
DE (1) | DE69736711T2 (es) |
DZ (1) | DZ2300A1 (es) |
EA (1) | EA002769B1 (es) |
ES (1) | ES2273369T3 (es) |
GT (1) | GT199700095A (es) |
HR (1) | HRP970454B1 (es) |
HU (1) | HUP9903965A3 (es) |
ID (1) | ID18249A (es) |
IL (1) | IL127566A0 (es) |
IS (1) | IS4963A (es) |
MA (1) | MA26438A1 (es) |
NO (1) | NO313636B1 (es) |
NZ (1) | NZ333302A (es) |
OA (1) | OA10977A (es) |
PA (1) | PA8436201A1 (es) |
PE (1) | PE108898A1 (es) |
PL (1) | PL332040A1 (es) |
SK (1) | SK23399A3 (es) |
TN (1) | TNSN97145A1 (es) |
TR (1) | TR199900389T2 (es) |
TW (1) | TW575573B (es) |
WO (1) | WO1998008847A1 (es) |
ZA (1) | ZA977687B (es) |
Families Citing this family (147)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2194756A1 (en) | 1995-05-12 | 1996-11-14 | Jun Yuan | Novel deazapurine derivatives; a new class of crf1 specific ligands |
US6191131B1 (en) | 1997-07-23 | 2001-02-20 | Dupont Pharmaceuticals Company | Azolo triazines and pyrimidines |
US6313124B1 (en) | 1997-07-23 | 2001-11-06 | Dupont Pharmaceuticals Company | Tetrazine bicyclic compounds |
US6124289A (en) * | 1996-07-24 | 2000-09-26 | Dupont Pharmaceuticals Co. | Azolo triazines and pyrimidines |
US7094782B1 (en) | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
US6060478A (en) * | 1996-07-24 | 2000-05-09 | Dupont Pharmaceuticals | Azolo triazines and pyrimidines |
EP0970082A2 (en) | 1997-02-18 | 2000-01-12 | Neurocrine Biosciences, Inc. | Biazacyclic crf antagonists |
JP2002501493A (ja) | 1997-04-22 | 2002-01-15 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | Crfアンタゴニストのチオフェノピリジン類 |
EP0994877A1 (en) * | 1997-07-03 | 2000-04-26 | Du Pont Pharmaceuticals Company | Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders |
NZ505079A (en) * | 1998-01-28 | 2003-08-29 | Du Pont Pharm Co | Pyrazolotriazines and pyrazolopyrimidines useful as corticotropin releasing factor antagonists |
US6187777B1 (en) * | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
CA2326319A1 (en) | 1998-04-02 | 1999-10-14 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-tetrahydro-9h pyrimidino[2,3-b]indole and 5,6,7,8-tetrahydro-9h-pyrimidino[4,5-b]indole derivatives: crf1 specific ligands |
US6472402B1 (en) | 1998-04-02 | 2002-10-29 | Neurogen Corporation | Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives |
CA2326884A1 (en) * | 1998-04-03 | 1999-10-14 | Dupont Pharmaceuticals Company | Thiazolo¬4,5-d|pyrimidines and pyridines as corticotropin releasing factor (crf) antagonists |
AU4556999A (en) | 1998-06-09 | 1999-12-30 | Neurogen Corporation | Pyrido[2,3-b]indolizine derivatives and aza analogues thereof; crf1 specific ligands |
US6509338B1 (en) | 1998-06-22 | 2003-01-21 | Bristol-Myers Squibb Company | Pyrazolo[1,5-A]triazine corticotropin releasing factor antagonists |
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- 1997-08-25 GT GT199700095A patent/GT199700095A/es unknown
- 1997-08-25 TW TW086112194A patent/TW575573B/zh active
- 1997-08-26 ID IDP972962A patent/ID18249A/id unknown
- 1997-08-26 AR ARP970103861A patent/AR015103A1/es not_active Application Discontinuation
- 1997-08-27 MA MA24779A patent/MA26438A1/fr unknown
- 1997-08-27 ZA ZA977687A patent/ZA977687B/xx unknown
- 1997-08-27 TN TNTNSN97145A patent/TNSN97145A1/fr unknown
- 1997-08-27 DZ DZ970150A patent/DZ2300A1/fr active
- 1997-08-28 CO CO97049895A patent/CO4600634A1/es unknown
-
1999
- 1999-01-29 IS IS4963A patent/IS4963A/is unknown
- 1999-02-17 OA OA9900035A patent/OA10977A/en unknown
- 1999-02-22 BG BG103189A patent/BG103189A/xx unknown
- 1999-02-26 NO NO19990927A patent/NO313636B1/no not_active IP Right Cessation
-
2004
- 2004-09-21 JP JP2004273978A patent/JP2005047930A/ja not_active Withdrawn
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1995033750A1 (en) * | 1994-06-08 | 1995-12-14 | Pfizer Inc. | Corticotropin releasing factor antagonists |
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