JP2021185200A5 - - Google Patents

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Publication number
JP2021185200A5
JP2021185200A5 JP2021146090A JP2021146090A JP2021185200A5 JP 2021185200 A5 JP2021185200 A5 JP 2021185200A5 JP 2021146090 A JP2021146090 A JP 2021146090A JP 2021146090 A JP2021146090 A JP 2021146090A JP 2021185200 A5 JP2021185200 A5 JP 2021185200A5
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JP
Japan
Prior art keywords
pyridinylmethoxy
anilino
quinolinyl
ethoxy
cyano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021146090A
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English (en)
Japanese (ja)
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JP2021185200A (ja
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Publication date
Priority claimed from JP2020070281A external-priority patent/JP2020111606A/ja
Application filed filed Critical
Publication of JP2021185200A publication Critical patent/JP2021185200A/ja
Publication of JP2021185200A5 publication Critical patent/JP2021185200A5/ja
Priority to JP2023160192A priority Critical patent/JP2023164747A/ja
Priority to JP2025124961A priority patent/JP2025137789A/ja
Pending legal-status Critical Current

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JP2021146090A 2007-10-17 2021-09-08 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態 Pending JP2021185200A (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2023160192A JP2023164747A (ja) 2007-10-17 2023-09-25 （ｅ）－ｎ－｛４－［３－クロロ－４－（２－ピリジニルメトキシ）アニリノ］－３－シアノ－７－エトキシ－６－キノリニル｝－４－（ジメチルアミノ）－２－ブテンアミドのマレイン酸塩およびその結晶形態
JP2025124961A JP2025137789A (ja) 2007-10-17 2025-07-25 （ｅ）－ｎ－｛４－［３－クロロ－４－（２－ピリジニルメトキシ）アニリノ］－３－シアノ－７－エトキシ－６－キノリニル｝－４－（ジメチルアミノ）－２－ブテンアミドのマレイン酸塩およびその結晶形態

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US12479607P 2007-10-17 2007-10-17
US61/124,796 2007-10-17
JP2020070281A JP2020111606A (ja) 2007-10-17 2020-04-09 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態

Related Parent Applications (1)

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JP2020070281A Division JP2020111606A (ja) 2007-10-17 2020-04-09 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023160192A Division JP2023164747A (ja) 2007-10-17 2023-09-25 （ｅ）－ｎ－｛４－［３－クロロ－４－（２－ピリジニルメトキシ）アニリノ］－３－シアノ－７－エトキシ－６－キノリニル｝－４－（ジメチルアミノ）－２－ブテンアミドのマレイン酸塩およびその結晶形態

Publications (2)

Publication Number Publication Date
JP2021185200A JP2021185200A (ja) 2021-12-09
JP2021185200A5 true JP2021185200A5 (https=) 2022-06-08

Family

ID=40347915

Family Applications (11)

Application Number Title Priority Date Filing Date
JP2010530105A Pending JP2011500712A (ja) 2007-10-17 2008-10-16 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2010258729A Withdrawn JP2011063610A (ja) 2007-10-17 2010-11-19 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2011289220A Active JP5965640B2 (ja) 2007-10-17 2011-12-28 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2012279650A Pending JP2013053170A (ja) 2007-10-17 2012-12-21 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2015080748A Pending JP2015127352A (ja) 2007-10-17 2015-04-10 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2016238151A Active JP6412090B2 (ja) 2007-10-17 2016-12-08 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2018079067A Withdrawn JP2018109071A (ja) 2007-10-17 2018-04-17 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2020070281A Withdrawn JP2020111606A (ja) 2007-10-17 2020-04-09 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2021146090A Pending JP2021185200A (ja) 2007-10-17 2021-09-08 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2023160192A Withdrawn JP2023164747A (ja) 2007-10-17 2023-09-25 （ｅ）－ｎ－｛４－［３－クロロ－４－（２－ピリジニルメトキシ）アニリノ］－３－シアノ－７－エトキシ－６－キノリニル｝－４－（ジメチルアミノ）－２－ブテンアミドのマレイン酸塩およびその結晶形態
JP2025124961A Pending JP2025137789A (ja) 2007-10-17 2025-07-25 （ｅ）－ｎ－｛４－［３－クロロ－４－（２－ピリジニルメトキシ）アニリノ］－３－シアノ－７－エトキシ－６－キノリニル｝－４－（ジメチルアミノ）－２－ブテンアミドのマレイン酸塩およびその結晶形態

Family Applications Before (8)

Application Number Title Priority Date Filing Date
JP2010530105A Pending JP2011500712A (ja) 2007-10-17 2008-10-16 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2010258729A Withdrawn JP2011063610A (ja) 2007-10-17 2010-11-19 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2011289220A Active JP5965640B2 (ja) 2007-10-17 2011-12-28 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2012279650A Pending JP2013053170A (ja) 2007-10-17 2012-12-21 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2015080748A Pending JP2015127352A (ja) 2007-10-17 2015-04-10 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2016238151A Active JP6412090B2 (ja) 2007-10-17 2016-12-08 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2018079067A Withdrawn JP2018109071A (ja) 2007-10-17 2018-04-17 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態
JP2020070281A Withdrawn JP2020111606A (ja) 2007-10-17 2020-04-09 （ｅ）−ｎ−｛４−［３−クロロ−４−（２−ピリジニルメトキシ）アニリノ］−３−シアノ−７−エトキシ−６−キノリニル｝−４−（ジメチルアミノ）−２−ブテンアミドのマレイン酸塩およびその結晶形態

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2023160192A Withdrawn JP2023164747A (ja) 2007-10-17 2023-09-25 （ｅ）－ｎ－｛４－［３－クロロ－４－（２－ピリジニルメトキシ）アニリノ］－３－シアノ－７－エトキシ－６－キノリニル｝－４－（ジメチルアミノ）－２－ブテンアミドのマレイン酸塩およびその結晶形態
JP2025124961A Pending JP2025137789A (ja) 2007-10-17 2025-07-25 （ｅ）－ｎ－｛４－［３－クロロ－４－（２－ピリジニルメトキシ）アニリノ］－３－シアノ－７－エトキシ－６－キノリニル｝－４－（ジメチルアミノ）－２－ブテンアミドのマレイン酸塩およびその結晶形態

Country Status (20)

Country Link
US (7) US8022216B2 (https=)
EP (6) EP2212311A2 (https=)
JP (11) JP2011500712A (https=)
KR (5) KR101208301B1 (https=)
CN (7) CN101918390B (https=)
AR (2) AR068932A1 (https=)
AU (1) AU2008312474B2 (https=)
BR (2) BR122019023745B8 (https=)
CA (2) CA2702930C (https=)
CL (1) CL2008003088A1 (https=)
ES (3) ES2602123T3 (https=)
IL (3) IL308687A (https=)
IN (1) IN2015DN01135A (https=)
MX (5) MX2010004173A (https=)
NZ (3) NZ600349A (https=)
PA (1) PA8800701A1 (https=)
RU (2) RU2463300C2 (https=)
SG (2) SG10201900175TA (https=)
TW (1) TW200934761A (https=)
WO (1) WO2009052264A2 (https=)

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CN107698563B (zh) * 2017-11-23 2020-10-30 江苏创诺制药有限公司 制备马来酸来那替尼晶型的方法
CN108299394A (zh) * 2018-02-28 2018-07-20 江苏创诺制药有限公司 来那替尼二马来酸盐晶型及其制备方法
CN110357855A (zh) * 2018-03-26 2019-10-22 江苏创诺制药有限公司 一种来那替尼盐酸盐晶型及其制备方法
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CN109053702A (zh) * 2018-08-13 2018-12-21 扬子江药业集团有限公司 一种阿法替尼类似物及其制备方法和用途
CN109503479A (zh) * 2018-12-03 2019-03-22 四川自豪时代药业有限公司 一种磷酸萘酚喹工艺杂质及其合成方法
CN111848581B (zh) * 2020-08-19 2021-08-10 昆明学院 3-氰基-4-苯胺基-6-氨基喹啉衍生物的制备方法
CN111943933B (zh) * 2020-09-02 2021-05-28 重庆医科大学 一种来那替尼杂质d的制备方法
CN111995618B (zh) * 2020-09-02 2021-06-11 重庆医科大学 一种来那替尼杂质g的制备方法
CN114380745A (zh) * 2020-10-19 2022-04-22 江苏苏中药业集团股份有限公司 一种取代丁烯酰胺颗粒混合物及晶型ii制备方法与应用
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KR101190953B1 (ko) 2009-08-25 2012-10-12 한올바이오파마주식회사 메트포르민 타우린염, 그의 제조방법, 그를 포함하는 약학 조성물 및 그를 포함하는 복합제제
KR20110021691A (ko) 2009-08-25 2011-03-04 한올바이오파마주식회사 메트포르민 메탄설폰산염, 그의 제조방법, 그를 포함하는 약학 조성물 및 그를 포함하는 복합제제
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