JP2022523368A5 - - Google Patents

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Publication number
JP2022523368A5
JP2022523368A5 JP2021549407A JP2021549407A JP2022523368A5 JP 2022523368 A5 JP2022523368 A5 JP 2022523368A5 JP 2021549407 A JP2021549407 A JP 2021549407A JP 2021549407 A JP2021549407 A JP 2021549407A JP 2022523368 A5 JP2022523368 A5 JP 2022523368A5
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JP
Japan
Application number
JP2021549407A
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Japanese (ja)
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JP2022523368A (ja
JPWO2020169736A5 (https=
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Publication date
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Priority claimed from PCT/EP2020/054485 external-priority patent/WO2020169736A1/en
Publication of JP2022523368A publication Critical patent/JP2022523368A/ja
Publication of JP2022523368A5 publication Critical patent/JP2022523368A5/ja
Publication of JPWO2020169736A5 publication Critical patent/JPWO2020169736A5/ja
Pending legal-status Critical Current

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JP2021549407A 2019-02-22 2020-02-20 1-(1-オキソ-1,2-ジヒドロイソキノリン-5-イル)-5-(トリフルオロメチル)-n-[2-(トリフルオロメチル)ピリジン-4-イル]-1h-ピラゾール-4-カルボキサミド一水和物の結晶形態 Pending JP2022523368A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CNPCT/CN2019/075834 2019-02-22
CN2019075834 2019-02-22
PCT/EP2020/054485 WO2020169736A1 (en) 2019-02-22 2020-02-20 Crystalline form of 1-(1-oxo-1,2-dihydroisoquinolin-5-yl)-5-(trifluoromethyl)-n-(2-(trifluoromethyl)pyridin-4-yl)-1h-pyrazole-4-carboxamide monohydrate

Publications (3)

Publication Number Publication Date
JP2022523368A JP2022523368A (ja) 2022-04-22
JP2022523368A5 true JP2022523368A5 (https=) 2023-02-28
JPWO2020169736A5 JPWO2020169736A5 (https=) 2023-02-28

Family

ID=69723907

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021549407A Pending JP2022523368A (ja) 2019-02-22 2020-02-20 1-(1-オキソ-1,2-ジヒドロイソキノリン-5-イル)-5-(トリフルオロメチル)-n-[2-(トリフルオロメチル)ピリジン-4-イル]-1h-ピラゾール-4-カルボキサミド一水和物の結晶形態

Country Status (21)

Country Link
US (1) US12269813B2 (https=)
EP (1) EP3927696B1 (https=)
JP (1) JP2022523368A (https=)
KR (1) KR20210131371A (https=)
CN (1) CN113474339B (https=)
AU (1) AU2020226723B2 (https=)
BR (1) BR112021016400A2 (https=)
CA (1) CA3129623A1 (https=)
EA (1) EA202192320A1 (https=)
EC (1) ECSP21067828A (https=)
ES (1) ES2966132T3 (https=)
IL (1) IL285675A (https=)
JO (1) JOP20210227A1 (https=)
MA (1) MA55019A (https=)
MX (1) MX2021010133A (https=)
PE (1) PE20212067A1 (https=)
PH (1) PH12021552018A1 (https=)
SG (1) SG11202108909SA (https=)
TW (1) TW202045495A (https=)
UY (1) UY38592A (https=)
WO (1) WO2020169736A1 (https=)

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Publication number Priority date Publication date Assignee Title
TWI795381B (zh) 2016-12-21 2023-03-11 比利時商健生藥品公司 作為malt1抑制劑之吡唑衍生物
ES2949871T3 (es) 2019-04-11 2023-10-03 Janssen Pharmaceutica Nv Anillos de piridina que contienen derivados como inhibidores de MALT1
JP2023539729A (ja) 2020-08-21 2023-09-19 ヤンセン ファーマシューティカ エヌ.ベー. Malt1阻害剤の非晶質形態及びその製剤
JP2024508890A (ja) 2021-03-03 2024-02-28 ヤンセン ファーマシューティカ エヌ.ベー. 治療有効用量のmalt1阻害剤jnj-67856633(1-(1-オキソ-1,2-ジヒドロイソキノリン-5-イル)-5-(トリフルオロメチル)-n-(2-(トリフルオロメチル)ピリジン-4-イル)-1h-ピラゾール-4-カルボキサミド)を使用して状態を治療する方法
EP4301365A1 (en) 2021-03-03 2024-01-10 Janssen Pharmaceutica NV Combination therapy using a malt1 inhibitor and a btk inhibitor
KR20240046170A (ko) 2021-08-09 2024-04-08 얀센 파마슈티카 엔브이 B-세포 악성종양의 치료에 사용하기 위한 조성물
AU2024357109A1 (en) 2023-10-06 2026-03-12 Ionctura Sa Combination of roginolisib with a malt1-gls inhibitor

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ES2336625T3 (es) * 2006-03-22 2010-04-14 Vertex Pharmaceuticals Incorporated Inhibidores de la proteina quinasa c-met para el tratamiento de trastornos proliferativos.
WO2008092292A1 (en) 2007-01-17 2008-08-07 The Hong Kong University Of Science And Technology Isoquinolone compounds as subtype-selective agonists for melatonin receptors mt1 and mt2
WO2011036885A1 (ja) * 2009-09-25 2011-03-31 武田薬品工業株式会社 複素環化合物
US20120071497A1 (en) 2010-06-03 2012-03-22 Pharmacyclics, Inc. Methods of treating abc-dlbcl using inhibitors of bruton's tyrosine kinase
CN107898791A (zh) 2010-06-03 2018-04-13 药品循环有限责任公司 布鲁顿酪氨酸激酶(btk)抑制剂的应用
JP5984801B2 (ja) 2010-06-22 2016-09-06 ビーエーエスエフ ソシエタス・ヨーロピアBasf Se 4−ヒドロキシピリジン類の製造方法
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ES2738695T3 (es) 2014-05-28 2020-01-24 Novartis Ag Nuevos Derivados de Pirazolo Pirimidina y su uso como inhibidores de MALT1
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US20200009135A1 (en) 2017-02-01 2020-01-09 Medivir Ab Therapeutic applications of malt1 inhibitors
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JP2023539729A (ja) * 2020-08-21 2023-09-19 ヤンセン ファーマシューティカ エヌ.ベー. Malt1阻害剤の非晶質形態及びその製剤

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