JP2022536979A5 - - Google Patents

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Publication number
JP2022536979A5
JP2022536979A5 JP2021575994A JP2021575994A JP2022536979A5 JP 2022536979 A5 JP2022536979 A5 JP 2022536979A5 JP 2021575994 A JP2021575994 A JP 2021575994A JP 2021575994 A JP2021575994 A JP 2021575994A JP 2022536979 A5 JP2022536979 A5 JP 2022536979A5
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JP
Japan
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JP2021575994A
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Japanese (ja)
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JP2022536979A (ja
JPWO2020257573A5 (https=
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Priority claimed from PCT/US2020/038624 external-priority patent/WO2020257573A1/en
Publication of JP2022536979A publication Critical patent/JP2022536979A/ja
Publication of JP2022536979A5 publication Critical patent/JP2022536979A5/ja
Publication of JPWO2020257573A5 publication Critical patent/JPWO2020257573A5/ja
Withdrawn legal-status Critical Current

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JP2021575994A 2019-06-21 2020-06-19 塩形態のベンペド酸及びそれを使用する方法 Withdrawn JP2022536979A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962864873P 2019-06-21 2019-06-21
US62/864,873 2019-06-21
PCT/US2020/038624 WO2020257573A1 (en) 2019-06-21 2020-06-19 Salt forms of bempedoic acid and methods for using the same

Publications (3)

Publication Number Publication Date
JP2022536979A JP2022536979A (ja) 2022-08-22
JP2022536979A5 true JP2022536979A5 (https=) 2023-06-16
JPWO2020257573A5 JPWO2020257573A5 (https=) 2023-06-16

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ID=71528020

Family Applications (3)

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JP2021575993A Pending JP2022537049A (ja) 2019-06-21 2020-06-19 ベンペド酸の製造方法及びその組成物
JP2021575994A Withdrawn JP2022536979A (ja) 2019-06-21 2020-06-19 塩形態のベンペド酸及びそれを使用する方法
JP2024211105A Pending JP2025032197A (ja) 2019-06-21 2024-12-04 ベンペド酸を含む製薬材料、医薬製剤及び医薬組成物

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JP2021575993A Pending JP2022537049A (ja) 2019-06-21 2020-06-19 ベンペド酸の製造方法及びその組成物

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JP2024211105A Pending JP2025032197A (ja) 2019-06-21 2024-12-04 ベンペド酸を含む製薬材料、医薬製剤及び医薬組成物

Country Status (13)

Country Link
US (10) US12344578B2 (https=)
EP (3) EP3986860A1 (https=)
JP (3) JP2022537049A (https=)
KR (3) KR20250143358A (https=)
CN (3) CN112437766A (https=)
AU (3) AU2020296094B2 (https=)
BR (1) BR112021025964A2 (https=)
CA (3) CA3144372A1 (https=)
ES (1) ES3032779T3 (https=)
HU (1) HUE072061T2 (https=)
IL (3) IL288909A (https=)
MX (2) MX2021015936A (https=)
WO (2) WO2020257571A1 (https=)

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CN112437766A (zh) 2019-06-21 2021-03-02 艾斯柏伦治疗公司 制备贝派地酸及其组合物的方法
CN114746389A (zh) 2019-10-03 2022-07-12 斯索恩有限公司 贝派地酸的晶形
US12516013B2 (en) 2019-12-06 2026-01-06 Synthon B.V. Crystalline forms of sodium salt of Bempedoic acid
CN111559961A (zh) * 2020-05-26 2020-08-21 杭州科巢生物科技有限公司 一种贝派地酸晶型及其制备方法
WO2021255180A1 (en) * 2020-06-19 2021-12-23 Synthon B.V. Salts of bempedoic acid
CN112521282A (zh) * 2020-12-02 2021-03-19 苏州汉德创宏生化科技有限公司 一种贝派地酸中间体及其合成方法
WO2022149161A1 (en) * 2021-01-05 2022-07-14 Dr. Reddy's Laboratories Limited Process for preparation of bempedoic acid and its intermediates
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CN115504914B (zh) * 2021-06-23 2024-05-07 武汉武药科技有限公司 一种贝派地酸中间体的制备方法
CN114436837B (zh) * 2021-12-27 2024-02-20 甘李药业股份有限公司 一种贝派地酸中间体的纯化方法
WO2023187833A1 (en) * 2022-03-30 2023-10-05 Enaltec Labs Private Limited A novel salt of bempedoic acid
CN117551009A (zh) * 2022-08-05 2024-02-13 武汉武药科技有限公司 一种贝派地酸中间体的合成方法
WO2024151311A1 (en) 2023-01-09 2024-07-18 Esperion Therapeutics, Inc. Methods of treatment using bempedoic acid
CN116589341A (zh) * 2023-04-14 2023-08-15 苏州汉德创宏生化科技有限公司 一种抗高血酯药物中间体的制备方法
TW202539678A (zh) 2024-03-20 2025-10-16 瑞典商阿斯特捷利康公司 Pcsk9抑制劑及其使用方法
TW202602886A (zh) 2024-03-20 2026-01-16 瑞典商阿斯特捷利康公司 Pcsk9抑制劑及其使用方法
TW202602866A (zh) 2024-03-20 2026-01-16 瑞典商阿斯特捷利康公司 Pcsk9抑制劑及其使用方法
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CN112437766A (zh) 2019-06-21 2021-03-02 艾斯柏伦治疗公司 制备贝派地酸及其组合物的方法
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