EA201270069A1 - Быстрорастворимая оральная пленочная лекарственная форма, содержащая стевиозиды в качестве агента, маскирующего неприятный вкус - Google Patents

Быстрорастворимая оральная пленочная лекарственная форма, содержащая стевиозиды в качестве агента, маскирующего неприятный вкус

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Publication number
EA201270069A1
EA201270069A1 EA201270069A EA201270069A EA201270069A1 EA 201270069 A1 EA201270069 A1 EA 201270069A1 EA 201270069 A EA201270069 A EA 201270069A EA 201270069 A EA201270069 A EA 201270069A EA 201270069 A1 EA201270069 A1 EA 201270069A1
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EA
Eurasian Patent Office
Prior art keywords
steviosid
form containing
oral film
medicine form
quickly soluble
Prior art date
Application number
EA201270069A
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English (en)
Other versions
EA021695B1 (ru
Inventor
Дзин Киу Парк
Вон Сук Янг
Киоунг Тае Дзунг
Original Assignee
Чабайо Энд Дайостек Ко., Лтд.
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43387021&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201270069(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Чабайо Энд Дайостек Ко., Лтд. filed Critical Чабайо Энд Дайостек Ко., Лтд.
Publication of EA201270069A1 publication Critical patent/EA201270069A1/ru
Publication of EA021695B1 publication Critical patent/EA021695B1/ru

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/075Ethers or acetals
    • A61K31/085Ethers or acetals having an ether linkage to aromatic ring nuclear carbon
    • A61K31/09Ethers or acetals having an ether linkage to aromatic ring nuclear carbon having two or more such linkages
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/14Quaternary ammonium compounds, e.g. edrophonium, choline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7007Drug-containing films, membranes or sheets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Inorganic Chemistry (AREA)
  • Zoology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Описана быстрорастворимая оральная пленочная лекарственная форма для маскировки неприятного вкуса, в частности быстрорастворимая оральная пленочная лекарственная форма, содержащая подсластитель на основе стевиозида и высокоэффективный подсластитель в соотношении по массе (мас./мас.) от 1:3 до 3:1, которая может эффективно маскировать горький или неприятный вкус лекарственного средства и может быстро растворяться в ротовой полости без воды, посредством этого улучшая ее послевкусие, таким образом, повышая приемлемость лекарственной формы для пациента.
EA201270069A 2009-06-25 2010-06-22 Быстрорастворимая оральная пленочная лекарственная форма, содержащая ребаудиозид а в качестве усилителя послевкусия и первичный подсластитель в качестве агента, маскирующего вкус EA021695B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR20090057276 2009-06-25
KR1020100057450A KR101074271B1 (ko) 2009-06-25 2010-06-17 불쾌한 맛을 효과적으로 은폐한 경구용 속용 필름
PCT/KR2010/004020 WO2010151020A2 (ko) 2009-06-25 2010-06-22 불쾌한 맛을 효과적으로 은폐한 경구용 속용 필름

Publications (2)

Publication Number Publication Date
EA201270069A1 true EA201270069A1 (ru) 2012-08-30
EA021695B1 EA021695B1 (ru) 2015-08-31

Family

ID=43387021

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201270069A EA021695B1 (ru) 2009-06-25 2010-06-22 Быстрорастворимая оральная пленочная лекарственная форма, содержащая ребаудиозид а в качестве усилителя послевкусия и первичный подсластитель в качестве агента, маскирующего вкус

Country Status (16)

Country Link
US (2) US20120156229A1 (ru)
EP (1) EP2431028B1 (ru)
JP (1) JP5539503B2 (ru)
KR (1) KR101074271B1 (ru)
CN (1) CN102333526B (ru)
AU (1) AU2010263494A1 (ru)
BR (1) BRPI1007804A2 (ru)
CA (1) CA2752865C (ru)
CO (1) CO6470871A2 (ru)
CR (1) CR20110671A (ru)
EA (1) EA021695B1 (ru)
MA (1) MA33439B1 (ru)
MX (1) MX2011008698A (ru)
SG (1) SG176545A1 (ru)
WO (1) WO2010151020A2 (ru)
ZA (1) ZA201106319B (ru)

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MX2011008698A (es) 2011-10-03
JP2012528854A (ja) 2012-11-15
AU2010263494A1 (en) 2011-08-25
CR20110671A (es) 2012-02-13
ZA201106319B (en) 2012-05-30
WO2010151020A3 (ko) 2011-05-19
WO2010151020A2 (ko) 2010-12-29
KR101074271B1 (ko) 2011-10-17
US9492379B2 (en) 2016-11-15
SG176545A1 (en) 2012-01-30
EP2431028B1 (en) 2017-07-12
BRPI1007804A2 (pt) 2016-02-23
KR20100138768A (ko) 2010-12-31
EP2431028A2 (en) 2012-03-21
CN102333526B (zh) 2014-05-28
CN102333526A (zh) 2012-01-25
CA2752865C (en) 2013-11-05
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US20130039932A1 (en) 2013-02-14
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