EA200200972A1 - Кристаллическое основание циталопрама - Google Patents

Кристаллическое основание циталопрама

Info

Publication number
EA200200972A1
EA200200972A1 EA200200972A EA200200972A EA200200972A1 EA 200200972 A1 EA200200972 A1 EA 200200972A1 EA 200200972 A EA200200972 A EA 200200972A EA 200200972 A EA200200972 A EA 200200972A EA 200200972 A1 EA200200972 A1 EA 200200972A1
Authority
EA
Eurasian Patent Office
Prior art keywords
salts
base
cytalogue
citalopram
preparations
Prior art date
Application number
EA200200972A
Other languages
English (en)
Inventor
Ханс Петерсен
Клаус Петер Бегесе
Пер Хольм
Original Assignee
Х.Лундбекк А/С
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8159320&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200200972(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Х.Лундбекк А/С filed Critical Х.Лундбекк А/С
Publication of EA200200972A1 publication Critical patent/EA200200972A1/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Laminated Bodies (AREA)
  • Silicates, Zeolites, And Molecular Sieves (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Manufacture Of Macromolecular Shaped Articles (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Данное изобретение относится к кристаллическому основанию хорошо известного антидепрессантного лекарственного средства циталопрама, 1-[3-(диметиламино)пропил]-1-(4-фторфенил)-1,3-дигидро-5-изобензофуранкарбонитрилу, препаратам с указанным основанием, способу получения очищенных солей циталопрама, таких как гидробромид, с использованием основания, солям, полученным указанным способом, и препаратам, содержащим указанные соли.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200200972A 2000-03-13 2001-02-28 Кристаллическое основание циталопрама EA200200972A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA200000402 2000-03-13
DKPCT/DK00/00183 2000-04-13
PCT/DK2001/000137 WO2001068627A1 (en) 2000-03-13 2001-02-28 Crystalline base of citalopram

Publications (1)

Publication Number Publication Date
EA200200972A1 true EA200200972A1 (ru) 2003-02-27

Family

ID=8159320

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200200972A EA200200972A1 (ru) 2000-03-13 2001-02-28 Кристаллическое основание циталопрама

Country Status (42)

Country Link
US (7) US20010031784A1 (ru)
EP (2) EP1227088B1 (ru)
JP (1) JP2003527383A (ru)
KR (1) KR20020080486A (ru)
CN (2) CN1680350A (ru)
AR (1) AR029811A1 (ru)
AT (3) ATE223396T1 (ru)
AU (2) AU746664B2 (ru)
BE (1) BE1013210A3 (ru)
BG (1) BG107065A (ru)
BR (1) BR0109373A (ru)
CA (2) CA2411732A1 (ru)
CH (2) CH691537A5 (ru)
CZ (1) CZ292077B6 (ru)
DE (7) DE20007303U1 (ru)
DK (3) DK173903B1 (ru)
EA (1) EA200200972A1 (ru)
ES (3) ES2173054T3 (ru)
FI (2) FI20010156A0 (ru)
FR (1) FR2806086B1 (ru)
GB (2) GB2357762B (ru)
GR (1) GR1003796B (ru)
HK (1) HK1054750A1 (ru)
HR (1) HRP20020756A2 (ru)
HU (3) HU0001581D0 (ru)
IE (1) IES20010109A2 (ru)
IL (2) IL158072A0 (ru)
IS (1) IS5841A (ru)
IT (2) IT1319645B1 (ru)
MX (1) MXPA02008793A (ru)
NL (2) NL1016435C1 (ru)
NO (2) NO312031B1 (ru)
PL (1) PL360158A1 (ru)
PT (2) PT1169314E (ru)
SE (2) SE517136C2 (ru)
SI (2) SI1227088T1 (ru)
SK (1) SK285528B6 (ru)
TR (1) TR200202185T2 (ru)
UA (1) UA74360C2 (ru)
WO (1) WO2001068627A1 (ru)
YU (1) YU68802A (ru)
ZA (1) ZA200207148B (ru)

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AU2003238676A1 (en) * 2003-04-21 2004-11-19 Podile Khadgapathi An improved process for the preparation of citalopram hydrobromide
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GB0317475D0 (en) 2003-07-25 2003-08-27 Meditab Specialities Pvt Ltd Product
JP4025735B2 (ja) * 2003-08-21 2007-12-26 ローム アンド ハース カンパニー 水性系を処理する方法
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KR101306635B1 (ko) 2005-06-27 2013-10-11 밸리언트 인터내셔널(바베이도스) 에스알엘 부프로피온염의 개질-방출 제형
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RU2503422C2 (ru) 2008-10-13 2014-01-10 ТАЙКО ХЕЛСКЕА ГРУП эЛПи Устройства и способы манипулирования стержнем катетера
WO2010126882A1 (en) 2009-04-29 2010-11-04 Fox Hollow Technologies, Inc. Methods and devices for cutting and abrading tissue
KR101323514B1 (ko) 2009-05-14 2013-10-29 코비디엔 엘피 세척이 용이한 죽상반 절제 카테터 및 사용 방법
RU2526915C2 (ru) 2009-12-02 2014-08-27 ТАЙКО ХЕЛСКЕА ГРУП эЛПи Способы и устройства для срезания ткани
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US10314667B2 (en) 2015-03-25 2019-06-11 Covidien Lp Cleaning device for cleaning medical instrument
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Also Published As

Publication number Publication date
IL147339A (en) 2004-09-27
HK1054750A1 (en) 2003-12-12
US20040167210A1 (en) 2004-08-26
AU2001100197A4 (en) 2001-09-20
IT1319645B1 (it) 2003-10-23
SI1169314T1 (en) 2002-12-31
JP2003527383A (ja) 2003-09-16
DE20121240U1 (de) 2002-07-04
SI1227088T1 (en) 2003-12-31
IL158072A0 (en) 2004-03-28
DE1227088T1 (de) 2003-02-06
US20030078442A1 (en) 2003-04-24
AR029811A1 (es) 2003-07-16
EP1169314A1 (en) 2002-01-09
CA2360287A1 (en) 2001-09-20
CH691477A5 (de) 2001-07-31
PT1227088E (pt) 2003-12-31
US20040132808A1 (en) 2004-07-08
BG107065A (bg) 2003-05-30
KR20020080486A (ko) 2002-10-23
NL1016435C1 (nl) 2000-11-06
ES2180471T1 (es) 2003-02-16
FR2806086B1 (fr) 2003-05-09
AU3725201A (en) 2001-09-13
DE60100786T2 (de) 2004-07-15
DE60100022D1 (de) 2002-10-10
ES2180471T3 (es) 2004-05-01
ES2159491A1 (es) 2001-10-01
SI1169314T2 (sl) 2011-08-31
DE20007303U1 (de) 2000-07-27
US20050165244A1 (en) 2005-07-28
NO20010619D0 (no) 2001-02-06
NO20010619L (no) 2001-09-14
ITMI20010406A1 (it) 2002-08-28
UA74360C2 (ru) 2005-12-15
US20050165092A1 (en) 2005-07-28
HU0100450D0 (en) 2001-04-28
DE10108042A1 (de) 2001-10-18
HU0001581D0 (en) 2000-06-28
ZA200207148B (en) 2003-04-23
DE10164687B4 (de) 2006-04-27
YU68802A (sh) 2005-11-28
ATE223396T1 (de) 2002-09-15
GR1003796B (el) 2002-02-08
SE0200730L (sv) 2002-08-29
CN1258530C (zh) 2006-06-07
HU0100531D0 (en) 2001-03-28
MXPA02008793A (es) 2003-02-12
NO315851B1 (no) 2003-11-03
WO2001068627A1 (en) 2001-09-20
ES2173054T3 (es) 2002-12-16
DE60100022T2 (de) 2003-03-06
EP1227088B1 (en) 2003-09-17
ITMI20002425A1 (it) 2002-05-09
AT4364U1 (de) 2001-06-25
BE1013210A3 (fr) 2001-10-02
CZ2001808A3 (cs) 2002-01-16
NO312031B1 (no) 2002-03-04
NO20020356D0 (no) 2002-01-23
NL1017413C1 (nl) 2001-09-13
FR2806086A1 (fr) 2001-09-14
ES2173054T1 (es) 2002-10-16
DK1169314T3 (da) 2002-10-14
DK173903B1 (da) 2002-02-11
AU2001100197B4 (en) 2001-12-06
HUP0100531A3 (en) 2004-04-28
IL147339A0 (en) 2002-08-14
SK13132002A3 (sk) 2003-01-09
US20010031784A1 (en) 2001-10-18
FI20010156A0 (fi) 2001-01-25
BR0109373A (pt) 2002-12-24
HUP0100531A2 (hu) 2002-01-28
DE60100786D1 (de) 2003-10-23
ATE250050T1 (de) 2003-10-15
GB2357762A (en) 2001-07-04
CA2411732A1 (en) 2001-09-20
AU746664B2 (en) 2002-05-02
CN1680350A (zh) 2005-10-12
HRP20020756A2 (en) 2004-12-31
PT1169314E (pt) 2002-11-29
IES20010109A2 (en) 2002-02-20
CA2360287C (en) 2003-09-09
FI109022B (fi) 2002-05-15
GB2357762B (en) 2002-01-30
SE0103046D0 (sv) 2001-09-14
NO20020356L (no) 2001-09-14
US20060247451A1 (en) 2006-11-02
SE0103046L (sv) 2001-11-14
DE60100022T3 (de) 2011-11-17
SE526022C2 (sv) 2005-06-14
CN1429220A (zh) 2003-07-09
SE517136C2 (sv) 2002-04-16
PL360158A1 (en) 2004-09-06
FI20010225A (fi) 2001-09-14
IS5841A (is) 2001-09-14
GB0105982D0 (en) 2001-05-02
TR200202185T2 (tr) 2002-12-23
CZ292077B6 (cs) 2003-07-16
ES2159491B1 (es) 2002-05-01
CH691537A5 (de) 2001-08-15
SK285528B6 (sk) 2007-03-01
EP1169314B2 (en) 2011-06-01
GB0102797D0 (en) 2001-03-21
EP1169314B1 (en) 2002-09-04
EP1227088A1 (en) 2002-07-31
DK1227088T3 (da) 2003-12-22
SE0200730D0 (sv) 2002-03-12
FI20010225A0 (fi) 2001-02-07

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