DK174125B1 - Farmaceutisk præparat til parenteral indgivelse indeholdende en somatostatinanalog, mælkesyre og en basisk forbindelse - Google Patents
Farmaceutisk præparat til parenteral indgivelse indeholdende en somatostatinanalog, mælkesyre og en basisk forbindelse Download PDFInfo
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- DK174125B1 DK174125B1 DK198803854A DK385488A DK174125B1 DK 174125 B1 DK174125 B1 DK 174125B1 DK 198803854 A DK198803854 A DK 198803854A DK 385488 A DK385488 A DK 385488A DK 174125 B1 DK174125 B1 DK 174125B1
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- Prior art keywords
- alkyl
- hydrogen
- phe
- lys
- amino
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- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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- A—HUMAN NECESSITIES
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- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/31—Somatostatins
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S930/00—Peptide or protein sequence
- Y10S930/01—Peptide or protein sequence
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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Landscapes
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- Chemical & Material Sciences (AREA)
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK200100558A DK174476B1 (da) | 1987-07-10 | 2001-04-04 | Anvendelse af octreotid til fremstilling af et lægemiddel til behandling af brystkræft |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB878716326A GB8716326D0 (en) | 1987-07-10 | 1987-07-10 | Organic compounds |
| GB878716324A GB8716324D0 (en) | 1987-07-10 | 1987-07-10 | Organic compounds |
| GB8716324 | 1987-07-10 | ||
| GB8716326 | 1987-07-10 |
Publications (3)
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| DK385488D0 DK385488D0 (da) | 1988-07-08 |
| DK385488A DK385488A (da) | 1989-01-11 |
| DK174125B1 true DK174125B1 (da) | 2002-07-01 |
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| Application Number | Title | Priority Date | Filing Date |
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| DK198803854A DK174125B1 (da) | 1987-07-10 | 1988-07-08 | Farmaceutisk præparat til parenteral indgivelse indeholdende en somatostatinanalog, mælkesyre og en basisk forbindelse |
| DK200100558A DK174476B1 (da) | 1987-07-10 | 2001-04-04 | Anvendelse af octreotid til fremstilling af et lægemiddel til behandling af brystkræft |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK200100558A DK174476B1 (da) | 1987-07-10 | 2001-04-04 | Anvendelse af octreotid til fremstilling af et lægemiddel til behandling af brystkræft |
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| CA (1) | CA1328402C (enExample) |
| CH (1) | CH677449A5 (enExample) |
| CS (1) | CS411591A3 (enExample) |
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| FR (1) | FR2617714B1 (enExample) |
| GB (1) | GB2208200B (enExample) |
| GR (1) | GR1000172B (enExample) |
| HK (1) | HK16492A (enExample) |
| HU (1) | HU203480B (enExample) |
| IE (1) | IE61908B1 (enExample) |
| IL (1) | IL87044A0 (enExample) |
| LU (1) | LU87268A1 (enExample) |
| MY (2) | MY103746A (enExample) |
| NL (1) | NL194823C (enExample) |
| NO (1) | NO179359C (enExample) |
| NZ (1) | NZ225340A (enExample) |
| PT (1) | PT87957B (enExample) |
| SE (2) | SE503191C2 (enExample) |
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| GB8813339D0 (en) * | 1988-06-06 | 1988-07-13 | Sandoz Ltd | Improvements in/relating to organic compounds |
| US5538739A (en) * | 1989-07-07 | 1996-07-23 | Sandoz Ltd. | Sustained release formulations of water soluble peptides |
| PH30995A (en) * | 1989-07-07 | 1997-12-23 | Novartis Inc | Sustained release formulations of water soluble peptides. |
| RU2128055C1 (ru) * | 1992-12-07 | 1999-03-27 | Такеда Кемикал Индастриз Лтд. | Фармацевтическая композиция замедленного высвобождения и способ ее получения |
| US5626945A (en) * | 1993-09-28 | 1997-05-06 | International Paper Company | Repulpable, water repellant paperboard |
| US6355613B1 (en) * | 1996-07-31 | 2002-03-12 | Peptor Limited | Conformationally constrained backbone cyclized somatostatin analogs |
| AU3215597A (en) | 1996-08-30 | 1998-03-19 | Biomeasure Incorporated | Method of inhibiting fibrosis with a somatostatin agonist |
| ES2167189B1 (es) * | 1999-12-17 | 2003-04-01 | Lipotec Sa | Formulacion farmaceutica estable para la administracion intravenosa o intramuscular, de principios activos peptidicos |
| US6316414B1 (en) | 2000-07-31 | 2001-11-13 | Dabur Research Foundation | Somatostatin analogs for the treatment of cancer |
| RU2277539C2 (ru) * | 2001-06-08 | 2006-06-10 | Сосьете Де Консей Де Решерш Э Д`Аппликасьон Сьентифик С.А.С. | Химерные аналоги соматостатина-дофамина |
| TWI287986B (en) * | 2001-12-13 | 2007-10-11 | Novartis Ag | Use of Epothilones for the treatment of the carcinoid syndrome |
| US20030207811A1 (en) * | 2002-05-03 | 2003-11-06 | Schrier Bruce K. | Method of treating retinopathy of prematurity using somatostatin analogs |
| PE20050285A1 (es) * | 2003-06-24 | 2005-06-09 | Novartis Ag | Composicion farmaceutica que comprende analogos ciclicos de somatostatina |
| GB0428151D0 (en) * | 2004-12-22 | 2005-01-26 | Novartis Ag | Organic compounds |
| PT1787658E (pt) | 2005-11-10 | 2012-06-22 | Chemi Spa | Formulações de libertação sustentada de análogos de somatostatina inibidores da hormona do crescimento |
| JP2009532346A (ja) * | 2006-03-31 | 2009-09-10 | イラスマス・ユニバーシティ・メディカル・センター・ロッテルダム | 腫瘍増殖制御のための新規組成物 |
| US9517240B2 (en) | 2006-09-26 | 2016-12-13 | The Regents Of The University Of California | Methods and compositions for cancer prevention and treatment |
| US20100160275A1 (en) * | 2006-09-26 | 2010-06-24 | Lee Eva Y H P | Methods and compositions for cancer prevention and treatment |
| US20090325863A1 (en) * | 2008-06-13 | 2009-12-31 | Kleinberg David L | Somatostatin analogs and IGF-I inhibition for breast cancer prevention |
| GB201016436D0 (en) | 2010-09-30 | 2010-11-17 | Q Chip Ltd | Method of making solid beads |
| GB201016433D0 (en) | 2010-09-30 | 2010-11-17 | Q Chip Ltd | Apparatus and method for making solid beads |
| US8629103B2 (en) * | 2010-12-02 | 2014-01-14 | New York University | Treatment of non-proliferative cystic disease of the breast |
| BR112013030874B8 (pt) * | 2011-06-02 | 2021-09-14 | Univ California | Uso de uma theta-defensina ou análogo da mesma para tratar uma condição inflamatória crônica |
| TWI523863B (zh) | 2012-11-01 | 2016-03-01 | 艾普森藥品公司 | 體抑素－多巴胺嵌合體類似物 |
| HK1213486A1 (zh) | 2012-11-01 | 2016-07-08 | Ipsen Pharma S.A.S. | 促生长素抑制素类似物及其二聚体 |
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| CH621770A5 (en) * | 1976-02-23 | 1981-02-27 | Sandoz Ag | Process for the preparation of novel peptide compounds |
| IE47421B1 (en) * | 1977-06-08 | 1984-03-07 | Merck & Co Inc | Somatostatin analogs,process for their preparation and pharmaceutical compositions containing them |
| LU78191A1 (de) * | 1977-09-28 | 1979-05-25 | Ciba Geigy Ag | Verfahren zur herstellung von neuen cyclopeptiden |
| US4328214A (en) * | 1979-07-04 | 1982-05-04 | Ciba-Geigy Corporation | Cyclopeptides and pharmaceutical preparations thereof and also processes for their manufacture |
| US4900730A (en) * | 1981-01-14 | 1990-02-13 | Toyo Jozo Co., Ltd. | Preparation which promotes the absorption of peptides |
| IE52535B1 (en) * | 1981-02-16 | 1987-12-09 | Ici Plc | Continuous release pharmaceutical compositions |
| JPS57188526A (en) * | 1981-05-14 | 1982-11-19 | Takeda Chem Ind Ltd | Peptide-containing pharmaceutical preparation |
| US4374060A (en) * | 1981-07-15 | 1983-02-15 | Merck & Co., Inc. | Process for the preparation of cyclic hexapeptide |
| DE3264693D1 (en) * | 1981-12-24 | 1985-08-14 | Ciba Geigy Ag | Cyclic octapeptides and pharmaceutical compositions thereof, and processes for their production and use |
| US4522813A (en) * | 1983-10-27 | 1985-06-11 | Merck & Co., Inc. | Cyclic hexapeptide somatostatin analogs |
| NL8503426A (nl) * | 1984-12-24 | 1986-07-16 | Sandoz Ag | 8alfa-acylamino-ergolinen, werkwijzen voor hun bereiding en farmaceutische preparaten die ze bevatten. |
| US4650787A (en) * | 1985-04-25 | 1987-03-17 | Schally Andrew Victor | Biologically active octapeptides |
| US4725577A (en) * | 1985-04-25 | 1988-02-16 | Administrators Of The Tulane Educational Fund | Biologically active lysine containing octapeptides |
| ZW14486A1 (en) * | 1985-07-29 | 1986-10-22 | Smithkline Beckman Corp | Pharmaceutical dosage unit |
| JPH085913B2 (ja) * | 1985-09-12 | 1996-01-24 | ザ・アドミニストレ−タ−ズ・オブ・ザ・ツ−レイン・エデユケイシヨナル・フアンド | 治療用ソマトスタチン同族体 |
| GR862206B (en) * | 1985-09-12 | 1986-12-31 | Univ Tulane | Therapeutic somatostatin analogs |
| HU198626B (en) * | 1986-05-27 | 1989-11-28 | Sandoz Ag | Process for producing pharmaceutical compositions comprising somatostatin analogues as active ingredient |
| HU906340D0 (en) * | 1986-10-13 | 1991-04-29 | Sandoz Ag | Synthesis in solid phase for producing peptonic alcohols |
| AU639371B2 (en) * | 1987-07-10 | 1993-07-22 | Novartis Ag | Method of treating breast cancer |
| US5187150A (en) * | 1987-10-14 | 1993-02-16 | Debiopharm S.A. | Polyester-based composition for the controlled release of polypeptide medicinal substances |
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1988
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- 1988-07-08 FR FR888809439A patent/FR2617714B1/fr not_active Expired - Lifetime
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1991
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1992
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1993
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1995
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1998
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B1 | Patent granted (law 1993) | ||
| PUP | Patent expired |