DE60110263D1 - Oxybenzamidderivate als faktor-xa-inhibitoren - Google Patents

Oxybenzamidderivate als faktor-xa-inhibitoren

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Publication number
DE60110263D1
DE60110263D1 DE60110263T DE60110263T DE60110263D1 DE 60110263 D1 DE60110263 D1 DE 60110263D1 DE 60110263 T DE60110263 T DE 60110263T DE 60110263 T DE60110263 T DE 60110263T DE 60110263 D1 DE60110263 D1 DE 60110263D1
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Germany
Prior art keywords
factor
compounds
formula
heteroaryl
factor viia
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Expired - Lifetime
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DE60110263T
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English (en)
Other versions
DE60110263T2 (de
Inventor
Marc Nazare
William Will
Anuschirwan Peyman
Hans Matter
Gerhard Zoller
Uwe Gerlach
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Sanofi Aventis Deutschland GmbH
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Aventis Pharma Deutschland GmbH
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Publication of DE60110263D1 publication Critical patent/DE60110263D1/de
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Publication of DE60110263T2 publication Critical patent/DE60110263T2/de
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/40—Acylated substituent nitrogen atom
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    • C07C2601/00—Systems containing only non-condensed rings
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