DE3822459C2 - Pharmazeutische Zusammensetzung - Google Patents
Pharmazeutische ZusammensetzungInfo
- Publication number
- DE3822459C2 DE3822459C2 DE3822459A DE3822459A DE3822459C2 DE 3822459 C2 DE3822459 C2 DE 3822459C2 DE 3822459 A DE3822459 A DE 3822459A DE 3822459 A DE3822459 A DE 3822459A DE 3822459 C2 DE3822459 C2 DE 3822459C2
- Authority
- DE
- Germany
- Prior art keywords
- peptide
- water
- composition according
- pharmaceutical composition
- salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A61K9/0024—Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Description
D-Ser (0-tBu)⁶-des Gly¹⁰-Azgly¹⁰-LHRH-Embonsäuresalz
D-Ser (But)⁶ LHRH (1-9) Ethylamid-Embonsäuresalz
D-Leu⁶-des Gly¹⁰-LHRH Ethylamid-Embonsäuresalz
0,04, (1 hr) 7,74, (6 hrs) 0,80, (Tag 2) 0,85, (Tag 4) 0,77, (Tag 7) 0,25, (Tag 11) 0,12, (Tag 14) 0,11, (Tag 18) 0,11, (Tag 21) 0,14, (Tag 25) 0,18.
Claims (11)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB8722134A GB2209937B (en) | 1987-09-21 | 1987-09-21 | Water insoluble polypeptides |
Publications (2)
Publication Number | Publication Date |
---|---|
DE3822459A1 DE3822459A1 (de) | 1989-03-30 |
DE3822459C2 true DE3822459C2 (de) | 1994-07-07 |
Family
ID=10624108
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE3822459A Expired - Lifetime DE3822459C2 (de) | 1987-09-21 | 1988-07-04 | Pharmazeutische Zusammensetzung |
DE122004000023C Active DE122004000023I2 (de) | 1987-09-21 | 1988-07-04 | Pharmazeutische Zusammensetzung |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE122004000023C Active DE122004000023I2 (de) | 1987-09-21 | 1988-07-04 | Pharmazeutische Zusammensetzung |
Country Status (23)
Country | Link |
---|---|
US (2) | US5192741A (de) |
JP (1) | JPH0713023B2 (de) |
AT (1) | AT397035B (de) |
AU (1) | AU611944B2 (de) |
BE (1) | BE1001685A5 (de) |
CA (1) | CA1326438C (de) |
CH (1) | CH675968A5 (de) |
DE (2) | DE3822459C2 (de) |
DK (1) | DK175311B1 (de) |
ES (1) | ES2009346A6 (de) |
FI (1) | FI96919C (de) |
FR (1) | FR2620621B1 (de) |
GB (1) | GB2209937B (de) |
GR (1) | GR1002244B (de) |
IE (1) | IE60608B1 (de) |
IL (1) | IL87790A (de) |
IT (1) | IT1225148B (de) |
LU (1) | LU87340A1 (de) |
NL (1) | NL193818C (de) |
NO (2) | NO178604C (de) |
PT (1) | PT88557B (de) |
SE (1) | SE503406C2 (de) |
ZA (1) | ZA886827B (de) |
Families Citing this family (192)
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1988
- 1988-07-04 DE DE3822459A patent/DE3822459C2/de not_active Expired - Lifetime
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- 1988-09-08 IE IE272788A patent/IE60608B1/en not_active IP Right Cessation
- 1988-09-12 AT AT0223488A patent/AT397035B/de not_active IP Right Cessation
- 1988-09-13 ZA ZA886827A patent/ZA886827B/xx unknown
- 1988-09-13 CA CA000577205A patent/CA1326438C/en not_active Expired - Lifetime
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- 1988-09-16 DK DK198805189A patent/DK175311B1/da active Protection Beyond IP Right Term
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- 1988-09-20 BE BE8801079A patent/BE1001685A5/fr not_active IP Right Cessation
- 1988-09-20 US US07/247,060 patent/US5192741A/en not_active Expired - Lifetime
- 1988-09-20 NL NL8802323A patent/NL193818C/nl not_active IP Right Cessation
- 1988-09-20 IT IT8805213A patent/IT1225148B/it active
- 1988-09-20 SE SE8803321A patent/SE503406C2/sv not_active IP Right Cessation
- 1988-09-20 CH CH3494/88A patent/CH675968A5/fr not_active IP Right Cessation
- 1988-09-20 PT PT88557A patent/PT88557B/pt not_active IP Right Cessation
- 1988-09-21 LU LU87340A patent/LU87340A1/fr unknown
- 1988-09-21 JP JP63238626A patent/JPH0713023B2/ja not_active Expired - Lifetime
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1994
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