CO5540368A2 - Composicion de liberacion sostenida y proceso para producirla - Google Patents

Composicion de liberacion sostenida y proceso para producirla

Info

Publication number
CO5540368A2
CO5540368A2 CO03111730A CO03111730A CO5540368A2 CO 5540368 A2 CO5540368 A2 CO 5540368A2 CO 03111730 A CO03111730 A CO 03111730A CO 03111730 A CO03111730 A CO 03111730A CO 5540368 A2 CO5540368 A2 CO 5540368A2
Authority
CO
Colombia
Prior art keywords
sustained release
physiologically active
release composition
composition according
produce
Prior art date
Application number
CO03111730A
Other languages
English (en)
Inventor
Yamamoto Kazumichi
Akiko Yamada
Hata Yoshio
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26617908&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO5540368(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of CO5540368A2 publication Critical patent/CO5540368A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Abstract

1.- Una composición de liberación sostenida que contiene un polímero de ácido láctico-ácido glicólico que tiene una relación de peso molecular medio en peso a pesomolecular medio en número de aproximadamente 1,90 ó menos, o una sal del mismo, y una sustancia fisiológicamente activa.2.- La composición de liberación sostenida de acuerdo con la reivindicación 1, donde la sustancia fisiológicamente activa es un péptido fisiológicamente activo.3.- La composición de liberación sostenida de acuerdo con la. reivindicación 2, donde la sustancia fisiológicamente activa es un derivado de la LH-RH.4.- La composición de liberación sostenida de acuerdo con la reivindicación 1, donde el peso molecular medio en peso de dicho polímero de ácido láctico-ácido glicólico es de aproximadamente 3.000 a aproximadamente 100.000.
CO03111730A 2001-06-29 2003-12-22 Composicion de liberacion sostenida y proceso para producirla CO5540368A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2001199462 2001-06-29
JP2001340980 2001-11-06

Publications (1)

Publication Number Publication Date
CO5540368A2 true CO5540368A2 (es) 2005-07-29

Family

ID=26617908

Family Applications (1)

Application Number Title Priority Date Filing Date
CO03111730A CO5540368A2 (es) 2001-06-29 2003-12-22 Composicion de liberacion sostenida y proceso para producirla

Country Status (32)

Country Link
US (3) US20040241229A1 (es)
EP (2) EP2108363A1 (es)
JP (3) JP5491318B2 (es)
KR (3) KR100988178B1 (es)
CN (1) CN1535141B (es)
AR (1) AR034640A1 (es)
AT (1) ATE429903T1 (es)
AU (1) AU2002311630B2 (es)
BR (1) BR0210572A (es)
CA (1) CA2451718C (es)
CO (1) CO5540368A2 (es)
CY (1) CY1109272T1 (es)
CZ (1) CZ306388B6 (es)
DE (1) DE60232147D1 (es)
DK (1) DK1399133T4 (es)
ES (1) ES2324156T5 (es)
HK (1) HK1061802A1 (es)
HU (1) HU230152B1 (es)
IL (1) IL159060A0 (es)
MX (1) MXPA03011440A (es)
MY (1) MY139606A (es)
NO (1) NO333531B1 (es)
NZ (1) NZ529968A (es)
PE (1) PE20030069A1 (es)
PL (1) PL212531B1 (es)
PT (1) PT1399133E (es)
RU (2) RU2297240C2 (es)
SI (1) SI1399133T2 (es)
SK (1) SK287568B6 (es)
TW (1) TWI225416B (es)
WO (1) WO2003002091A2 (es)
ZA (1) ZA200309153B (es)

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PT1532985T (pt) 2002-06-25 2017-01-20 Takeda Pharmaceuticals Co Processo de produção de uma composição de libertação sustentada
WO2004029129A1 (ja) * 2002-09-24 2004-04-08 Asahi Kasei Chemicals Corporation グリコール酸共重合体及びその製造方法
TW200529890A (en) 2004-02-10 2005-09-16 Takeda Pharmaceutical Sustained-release preparations
TW200613012A (en) * 2004-07-02 2006-05-01 Takeda Pharmaceuticals Co Sustained-release composition, process for producing the same and use of the same
ATE382337T1 (de) * 2005-04-28 2008-01-15 Nipro Corp Bioabsorbierbare pharmazeutische zusammensetzung enthaltend einen plga-copolymer
JP5242415B2 (ja) 2006-01-18 2013-07-24 フォアシーエイサー ファーマシューティカルズ インコーポレイテッド 高い安定性を持つ薬理組成物
EA016176B1 (ru) 2006-12-18 2012-02-28 Такеда Фармасьютикал Компани Лимитед Композиция с замедленным высвобождением и способ её получения
LT3660073T (lt) 2007-02-15 2023-10-10 Tolmar International Limited Poli(laktidas-ko-glikolidas) su lėtu pradiniu atsipalaidavimu
KR101008462B1 (ko) * 2007-07-26 2011-01-14 조남열 치어류 이동용 어도 장치
KR100969641B1 (ko) * 2007-11-12 2010-07-14 민선영 저수지의 제방용 어도
KR100969642B1 (ko) * 2007-11-15 2010-07-12 민선영 하천의 보용 어도
US8641900B2 (en) 2009-11-05 2014-02-04 Taiwan Biotech Co., Ltd Method and device for continuously preparing microspheres, and collection unit thereof
TWI477266B (zh) * 2009-11-05 2015-03-21 Taiwan Biotech Co Ltd 連續製備微粒的方法、裝置及其收集單元
EP2697361A1 (en) * 2011-04-11 2014-02-19 Cellcura Asa Protein-free culture media products for manufacturing viral-based vaccines
JP6246712B2 (ja) 2012-07-12 2017-12-13 武田薬品工業株式会社 マイクロカプセル粉末の製造方法
RU2572992C2 (ru) * 2012-08-28 2016-01-20 Федеральное государственное бюджетное образовательное учреждение высшего образования "Курская государственная сельскохозяйственная академия имени И.И. Иванова" Способ получения микрокапсул водорастворимых препаратов пестицидов
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RU2537248C1 (ru) * 2013-05-24 2014-12-27 Екатерина Евгеньевна Быковская Способ получения микрокапсул гетероциклических соединений триазинового ряда
RU2537173C1 (ru) * 2013-05-24 2014-12-27 Александр Александрович Кролевец Способ получения микрокапсул гетероциклических соединений триазинового ряда
WO2015088990A1 (en) 2013-12-09 2015-06-18 Durect Corporation Pharmaceutically active agent complexes, polymer complexes, and compositions and methods involving the same
CN106456704A (zh) 2014-04-16 2017-02-22 Veyx-药物有限公司 兽药组合物和其应用
TW201618783A (zh) 2014-08-07 2016-06-01 艾森塔製藥公司 以布魯頓(Bruton)氏酪胺酸激酶(BTK)佔據和BTK再合成速率為基礎之治療癌症、免疫和自體免疫疾病及發炎性疾病之方法
CN104224731A (zh) * 2014-09-11 2014-12-24 北京天晟泰丰医药科技有限公司 一种不含致敏性辅料的九肽微球的制备方法
JP5938762B1 (ja) 2015-09-01 2016-06-22 日揮株式会社 マイクロカプセル製剤及びその製造方法
CN110856690A (zh) * 2018-08-22 2020-03-03 深圳善康医疗健康产业有限公司 一种植入剂包膜及干燥装置
WO2021234731A1 (en) * 2020-05-18 2021-11-25 Dr Reddy's Institute Of Life Sciences Sustained release compositions

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PT1532985T (pt) * 2002-06-25 2017-01-20 Takeda Pharmaceuticals Co Processo de produção de uma composição de libertação sustentada

Also Published As

Publication number Publication date
ZA200309153B (en) 2005-01-26
IL159060A0 (en) 2004-05-12
PT1399133E (pt) 2009-06-05
ES2324156T5 (es) 2012-07-23
EP1399133A2 (en) 2004-03-24
CN1535141B (zh) 2013-04-24
JP2012136530A (ja) 2012-07-19
RU2006143104A (ru) 2008-06-20
SK15612003A3 (sk) 2004-07-07
PL212531B1 (pl) 2012-10-31
HK1061802A1 (en) 2004-10-08
JP5860300B2 (ja) 2016-02-16
HUP0400382A3 (en) 2010-01-28
WO2003002091A3 (en) 2003-07-24
EP1399133B1 (en) 2009-04-29
KR20090096755A (ko) 2009-09-14
DK1399133T3 (da) 2009-08-03
CZ20033492A3 (cs) 2005-01-12
US20080108778A1 (en) 2008-05-08
JP5931147B2 (ja) 2016-06-08
EP1399133B2 (en) 2012-05-02
US8258252B2 (en) 2012-09-04
NO20035737L (no) 2004-02-20
SK287568B6 (sk) 2011-02-04
CZ306388B6 (cs) 2017-01-04
CY1109272T1 (el) 2014-07-02
BR0210572A (pt) 2004-08-03
ATE429903T1 (de) 2009-05-15
SI1399133T2 (sl) 2012-08-31
EP2108363A1 (en) 2009-10-14
PL367491A1 (en) 2005-02-21
CA2451718C (en) 2011-03-15
MXPA03011440A (es) 2004-07-01
US20120295848A1 (en) 2012-11-22
JP2010280703A (ja) 2010-12-16
WO2003002091A2 (en) 2003-01-09
PE20030069A1 (es) 2003-03-17
ES2324156T3 (es) 2009-07-31
HUP0400382A2 (hu) 2004-12-28
TWI225416B (en) 2004-12-21
CN1535141A (zh) 2004-10-06
NO333531B1 (no) 2013-07-01
US20040241229A1 (en) 2004-12-02
AU2002311630B2 (en) 2007-07-19
HU230152B1 (hu) 2015-09-28
RU2434644C2 (ru) 2011-11-27
NO20035737D0 (no) 2003-12-19
DK1399133T4 (da) 2012-07-23
DE60232147D1 (de) 2009-06-10
MY139606A (en) 2009-10-30
SI1399133T1 (sl) 2009-10-31
CA2451718A1 (en) 2003-01-09
NZ529968A (en) 2005-08-26
AR034640A1 (es) 2004-03-03
RU2297240C2 (ru) 2007-04-20
KR20040018401A (ko) 2004-03-03
RU2004102503A (ru) 2005-03-10
KR100988178B1 (ko) 2010-10-18
JP2015007120A (ja) 2015-01-15
JP5491318B2 (ja) 2014-05-14
KR20090108640A (ko) 2009-10-15

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