CN103450129B - 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法 - Google Patents

吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法 Download PDF

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Publication number
CN103450129B
CN103450129B CN201310414119.9A CN201310414119A CN103450129B CN 103450129 B CN103450129 B CN 103450129B CN 201310414119 A CN201310414119 A CN 201310414119A CN 103450129 B CN103450129 B CN 103450129B
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alkyl
benzyl
solution
benzene
substituted
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CN103450129A (zh
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弗兰克.希梅尔斯巴赫
马赛厄斯.埃克哈特
彼得.艾克尔曼
爱德华.L.巴索米恩
利奥.托马斯
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Boehringer Ingelheim International GmbH
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Priority claimed from DE102004012676A external-priority patent/DE102004012676A1/de
Priority claimed from DE102004040168A external-priority patent/DE102004040168A1/de
Priority claimed from DE102004061145A external-priority patent/DE102004061145A1/de
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CN201310414119.9A 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法 Ceased CN103450129B (zh)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
DE102004012676A DE102004012676A1 (de) 2004-03-16 2004-03-16 Glucopyranosyl-substituierte Phenyle, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
DE102004012676.3 2004-03-16
DE102004040168.3 2004-08-18
DE102004040168A DE102004040168A1 (de) 2004-08-18 2004-08-18 Glucopyranosyl-substituierte Phenyle, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
DE102004061145A DE102004061145A1 (de) 2004-12-16 2004-12-16 Glucopyranosyl-substituierte Benzol-Derivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
DE102004061145.9 2004-12-16
EP05002628.5 2005-02-09
EP05002628 2005-02-09
CNA2005800069449A CN1930141A (zh) 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法

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CN103450129A CN103450129A (zh) 2013-12-18
CN103450129B true CN103450129B (zh) 2015-08-12

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CN201310414119.9A Ceased CN103450129B (zh) 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法
CN2012105151009A Pending CN103030617A (zh) 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法
CN201310368328.4A Ceased CN103467423B (zh) 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法
CN201310379906.4A Ceased CN103435581B (zh) 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法

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CN2012105151009A Pending CN103030617A (zh) 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法
CN201310368328.4A Ceased CN103467423B (zh) 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法
CN201310379906.4A Ceased CN103435581B (zh) 2004-03-16 2005-03-11 吡喃葡萄糖基取代的苯基衍生物、含该化合物的药物、其用途及其制造方法

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US (6) US7579449B2 (enExample)
EP (4) EP2360164A3 (enExample)
JP (3) JP4181605B2 (enExample)
KR (2) KR20120007088A (enExample)
CN (4) CN103450129B (enExample)
AR (3) AR048041A1 (enExample)
AT (1) ATE557013T1 (enExample)
AU (1) AU2005225511C1 (enExample)
BE (1) BE2014C064I2 (enExample)
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DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
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TW200637869A (en) 2005-01-28 2006-11-01 Chugai Pharmaceutical Co Ltd The spiroketal derivatives and the use as therapeutical agent for diabetes of the same
JP5264183B2 (ja) 2005-02-23 2013-08-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング グルコピラノシル置換（（ヘテロ）アリールエチニル−ベンジル）−ベンゼン誘導体及びナトリウム依存性グルコース共輸送体２（ｓｇｌｔ２）インヒビターとしてのそれらの使用
DE602006011453D1 (de) 2005-04-15 2010-02-11 Boehringer Ingelheim Pharma Glucopyranosyl-substituierte (heteroaryloxy-benzyl)-benzen-derivate als sglt-inhibitoren
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US7772191B2 (en) * 2005-05-10 2010-08-10 Boehringer Ingelheim International Gmbh Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
TW200726755A (en) * 2005-07-07 2007-07-16 Astellas Pharma Inc A crystalline choline salt of an azulene derivative
EP1910390B1 (en) 2005-07-27 2010-05-19 Boehringer Ingelheim International GmbH Glucopyranosyl-substituted ((hetero)cycloalyklethynyl-benzyl)-benzene derivatives and use thereof as sodium-dependent glucose cotransporter (sglt) inhibitors
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
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