BR0210941A - Terapia de combinação de oxazolidinonas substituìdas - Google Patents

Terapia de combinação de oxazolidinonas substituìdas

Info

Publication number
BR0210941A
BR0210941A BR0210941-7A BR0210941A BR0210941A BR 0210941 A BR0210941 A BR 0210941A BR 0210941 A BR0210941 A BR 0210941A BR 0210941 A BR0210941 A BR 0210941A
Authority
BR
Brazil
Prior art keywords
combination therapy
substituted oxazolidinone
combinations
oxazolidinone
substituted
Prior art date
Application number
BR0210941-7A
Other languages
English (en)
Other versions
BRPI0210941B1 (pt
BRPI0210941B8 (pt
Inventor
Alexander Straub
Thomas Lampe
Josef Pernestorfer
Elisabeth Perzborn
Jens Pohlmann
Susanne Roehrig
Karl-Heinz Schlemmer
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7688824&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR0210941(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of BR0210941A publication Critical patent/BR0210941A/pt
Publication of BRPI0210941B1 publication Critical patent/BRPI0210941B1/pt
Publication of BRPI0210941B8 publication Critical patent/BRPI0210941B8/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

"TERAPIA DE COMBINAçãO DE OXAZOLIDINONAS SUBSTITUìDAS". A presente invenção refere-se a combinações de A) oxazolidinonas da fórmula (I) com B) outras substâncias ativas, a um processo para produção dessas combinações e ao uso das mesmas como medicamento, particularmente para tratamento e/ou profilaxia de doenças tromboembólicas.
BRPI0210941A 2001-06-20 2002-06-07 produto farmacêutico contendo combinações de oxazolidinonas substituídas, seu uso, seu processo de produção, e medicamento BRPI0210941B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10129725A DE10129725A1 (de) 2001-06-20 2001-06-20 Kombinationstherapie substituierter Oxazolidinone
PCT/EP2002/006237 WO2003000256A1 (de) 2001-06-20 2002-06-07 Kombinationstherapie substituierter oxazolidinone

Publications (3)

Publication Number Publication Date
BR0210941A true BR0210941A (pt) 2004-06-08
BRPI0210941B1 BRPI0210941B1 (pt) 2015-09-15
BRPI0210941B8 BRPI0210941B8 (pt) 2021-05-25

Family

ID=7688824

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0210941A BRPI0210941B8 (pt) 2001-06-20 2002-06-07 produto farmacêutico contendo combinações de oxazolidinonas substituídas, seu uso, seu processo de produção, e medicamento

Country Status (33)

Country Link
US (2) US7767702B2 (pt)
EP (1) EP1411932B1 (pt)
JP (1) JP4667744B2 (pt)
KR (1) KR100904138B1 (pt)
CN (1) CN100577162C (pt)
AT (1) ATE457171T1 (pt)
AU (1) AU2002312982B2 (pt)
BG (1) BG66354B1 (pt)
BR (1) BRPI0210941B8 (pt)
CA (1) CA2451258C (pt)
CO (1) CO5550434A2 (pt)
CU (1) CU23366B7 (pt)
CY (1) CY1110019T1 (pt)
CZ (1) CZ303715B6 (pt)
DE (2) DE10129725A1 (pt)
DK (1) DK1411932T3 (pt)
EC (1) ECSP034916A (pt)
EE (1) EE05419B1 (pt)
ES (1) ES2338997T3 (pt)
HK (1) HK1068811A1 (pt)
HR (1) HRP20040042B1 (pt)
HU (1) HU230120B1 (pt)
IL (2) IL159257A0 (pt)
MX (1) MXPA03011519A (pt)
NO (1) NO334821B1 (pt)
NZ (1) NZ530223A (pt)
PL (1) PL206803B1 (pt)
PT (1) PT1411932E (pt)
RU (1) RU2321407C9 (pt)
SI (1) SI1411932T1 (pt)
SK (1) SK287904B6 (pt)
UA (1) UA82986C2 (pt)
WO (1) WO2003000256A1 (pt)

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DE50214206D1 (de) 2010-03-25
SK15302003A3 (sk) 2004-07-07
ATE457171T1 (de) 2010-02-15
HU230120B1 (hu) 2015-08-28
CZ20033451A3 (en) 2004-03-17
NO20035743D0 (no) 2003-12-19
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EP1411932A1 (de) 2004-04-28
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US20040242660A1 (en) 2004-12-02
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HK1068811A1 (en) 2005-05-06
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