HK1068811A1 - Substituted oxazolidinones for combinational therapy - Google Patents
Substituted oxazolidinones for combinational therapyInfo
- Publication number
- HK1068811A1 HK1068811A1 HK05101508.8A HK05101508A HK1068811A1 HK 1068811 A1 HK1068811 A1 HK 1068811A1 HK 05101508 A HK05101508 A HK 05101508A HK 1068811 A1 HK1068811 A1 HK 1068811A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- substituted oxazolidinones
- combinational therapy
- oxazolidinones
- combinations
- combinational
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10129725A DE10129725A1 (de) | 2001-06-20 | 2001-06-20 | Kombinationstherapie substituierter Oxazolidinone |
PCT/EP2002/006237 WO2003000256A1 (de) | 2001-06-20 | 2002-06-07 | Kombinationstherapie substituierter oxazolidinone |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1068811A1 true HK1068811A1 (en) | 2005-05-06 |
Family
ID=7688824
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK05101508.8A HK1068811A1 (en) | 2001-06-20 | 2005-02-23 | Substituted oxazolidinones for combinational therapy |
Country Status (33)
Country | Link |
---|---|
US (2) | US7767702B2 (xx) |
EP (1) | EP1411932B1 (xx) |
JP (1) | JP4667744B2 (xx) |
KR (1) | KR100904138B1 (xx) |
CN (1) | CN100577162C (xx) |
AT (1) | ATE457171T1 (xx) |
AU (1) | AU2002312982B2 (xx) |
BG (1) | BG66354B1 (xx) |
BR (1) | BRPI0210941B8 (xx) |
CA (1) | CA2451258C (xx) |
CO (1) | CO5550434A2 (xx) |
CU (1) | CU23366B7 (xx) |
CY (1) | CY1110019T1 (xx) |
CZ (1) | CZ303715B6 (xx) |
DE (2) | DE10129725A1 (xx) |
DK (1) | DK1411932T3 (xx) |
EC (1) | ECSP034916A (xx) |
EE (1) | EE05419B1 (xx) |
ES (1) | ES2338997T3 (xx) |
HK (1) | HK1068811A1 (xx) |
HR (1) | HRP20040042B1 (xx) |
HU (1) | HU230120B1 (xx) |
IL (2) | IL159257A0 (xx) |
MX (1) | MXPA03011519A (xx) |
NO (1) | NO334821B1 (xx) |
NZ (1) | NZ530223A (xx) |
PL (1) | PL206803B1 (xx) |
PT (1) | PT1411932E (xx) |
RU (1) | RU2321407C9 (xx) |
SI (1) | SI1411932T1 (xx) |
SK (1) | SK287904B6 (xx) |
UA (1) | UA82986C2 (xx) |
WO (1) | WO2003000256A1 (xx) |
Families Citing this family (66)
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DE10129725A1 (de) | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
DE10300111A1 (de) * | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
EP1631560A2 (en) * | 2003-04-25 | 2006-03-08 | 3-Dimensional Pharmaceuticals, Inc. | C-fms kinase inhibitors |
WO2004101552A1 (en) * | 2003-05-14 | 2004-11-25 | Orchid Chemicals & Pharmaceuticals Ltd | Oxazolidinone derivatives as antibacterial agents |
DE10336716A1 (de) | 2003-08-11 | 2005-03-10 | Merck Patent Gmbh | Verfahren zur Herstellung von N-Aryl-morpholinonen |
US7687627B2 (en) * | 2003-09-08 | 2010-03-30 | Wockhardt Limited | Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy |
DE10342570A1 (de) * | 2003-09-15 | 2005-04-14 | Bayer Healthcare Ag | Verfahren zur Herstellung von 4-(4-Aminophenyl)-3-morpholinon |
WO2005027896A1 (ja) * | 2003-09-19 | 2005-03-31 | Kissei Pharmaceutical Co., Ltd. | 併用医薬 |
DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
DE102004002044A1 (de) * | 2004-01-15 | 2005-08-04 | Bayer Healthcare Ag | Herstellverfahren |
US7371743B2 (en) * | 2004-02-28 | 2008-05-13 | Boehringer Ingelheim International Gmbh | Carboxylic acid amides, the preparation thereof and their use as medicaments |
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2001
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2002
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- 2002-06-07 RU RU2004101404/15A patent/RU2321407C9/ru active
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- 2002-06-07 BR BRPI0210941A patent/BRPI0210941B8/pt not_active IP Right Cessation
- 2002-06-07 WO PCT/EP2002/006237 patent/WO2003000256A1/de active IP Right Grant
- 2002-06-07 JP JP2003506901A patent/JP4667744B2/ja not_active Expired - Lifetime
- 2002-06-07 US US10/481,297 patent/US7767702B2/en not_active Expired - Fee Related
- 2002-06-07 KR KR1020037016596A patent/KR100904138B1/ko active IP Right Grant
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- 2002-06-07 ES ES02738154T patent/ES2338997T3/es not_active Expired - Lifetime
- 2002-06-07 CN CN02812411A patent/CN100577162C/zh not_active Expired - Lifetime
- 2002-06-07 HU HU0400240A patent/HU230120B1/hu unknown
- 2002-06-07 DK DK02738154.0T patent/DK1411932T3/da active
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- 2002-06-07 DE DE50214206T patent/DE50214206D1/de not_active Expired - Lifetime
- 2002-06-07 EP EP02738154A patent/EP1411932B1/de not_active Expired - Lifetime
- 2002-06-07 PT PT02738154T patent/PT1411932E/pt unknown
- 2002-06-07 MX MXPA03011519A patent/MXPA03011519A/es active IP Right Grant
- 2002-06-07 AT AT02738154T patent/ATE457171T1/de active
- 2002-06-07 PL PL368079A patent/PL206803B1/pl unknown
- 2002-07-06 UA UA2004010387A patent/UA82986C2/uk unknown
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- 2003-12-12 BG BG108443A patent/BG66354B1/bg unknown
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2004
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- 2004-01-19 HR HRP20040042AA patent/HRP20040042B1/hr not_active IP Right Cessation
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2005
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