AU2010275754B2 - Tamper-resistant dosage form for oxidation-sensitive opioids - Google Patents

Tamper-resistant dosage form for oxidation-sensitive opioids Download PDF

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Publication number
AU2010275754B2
AU2010275754B2 AU2010275754A AU2010275754A AU2010275754B2 AU 2010275754 B2 AU2010275754 B2 AU 2010275754B2 AU 2010275754 A AU2010275754 A AU 2010275754A AU 2010275754 A AU2010275754 A AU 2010275754A AU 2010275754 B2 AU2010275754 B2 AU 2010275754B2
Authority
AU
Australia
Prior art keywords
dosage form
pharmaceutical dosage
acid
opioid
form according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU2010275754A
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English (en)
Other versions
AU2010275754A1 (en
Inventor
Johannes Bartholomaus
Ulrike Bertram
Fatima Bicane
Anja Geissler
Kornelia Griessmann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gruenenthal GmbH
Original Assignee
Gruenenthal GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41263602&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2010275754(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gruenenthal GmbH filed Critical Gruenenthal GmbH
Publication of AU2010275754A1 publication Critical patent/AU2010275754A1/en
Application granted granted Critical
Publication of AU2010275754B2 publication Critical patent/AU2010275754B2/en
Ceased legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
AU2010275754A 2009-07-22 2010-07-21 Tamper-resistant dosage form for oxidation-sensitive opioids Ceased AU2010275754B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09009480 2009-07-22
EP09009480.6 2009-07-22
PCT/EP2010/004460 WO2011009603A1 (en) 2009-07-22 2010-07-21 Tamper-resistant dosage form for oxidation-sensitive oploids

Publications (2)

Publication Number Publication Date
AU2010275754A1 AU2010275754A1 (en) 2011-12-15
AU2010275754B2 true AU2010275754B2 (en) 2014-05-15

Family

ID=41263602

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2010275754A Ceased AU2010275754B2 (en) 2009-07-22 2010-07-21 Tamper-resistant dosage form for oxidation-sensitive opioids
AU2010275755A Ceased AU2010275755B2 (en) 2009-07-22 2010-07-21 Oxidation-stabilized tamper-resistant dosage form

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU2010275755A Ceased AU2010275755B2 (en) 2009-07-22 2010-07-21 Oxidation-stabilized tamper-resistant dosage form

Country Status (26)

Country Link
US (7) US20110020451A1 (es)
EP (4) EP2456424B1 (es)
JP (2) JP2012533585A (es)
KR (2) KR101747156B1 (es)
CN (2) CN102573806B (es)
AR (1) AR077420A1 (es)
AU (2) AU2010275754B2 (es)
BR (2) BR112012001244A2 (es)
CA (2) CA2767888C (es)
CL (2) CL2011002969A1 (es)
CO (2) CO6470798A2 (es)
EC (2) ECSP12011590A (es)
ES (3) ES2560210T3 (es)
HK (3) HK1216296A1 (es)
HU (1) HUE042987T2 (es)
IL (3) IL216522A (es)
MX (2) MX2012000369A (es)
NZ (2) NZ596666A (es)
PE (2) PE20120631A1 (es)
PL (2) PL2456424T3 (es)
PT (1) PT2456424E (es)
RU (3) RU2015138422A (es)
SI (1) SI2456424T1 (es)
TW (1) TWI473628B (es)
WO (2) WO2011009604A1 (es)
ZA (2) ZA201109446B (es)

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