ATE522213T1 - Fünfgliedrige-heteroringderivate , ihre herstellung und ihre verwendung als arzneimittel - Google Patents
Fünfgliedrige-heteroringderivate , ihre herstellung und ihre verwendung als arzneimittelInfo
- Publication number
- ATE522213T1 ATE522213T1 AT02076763T AT02076763T ATE522213T1 AT E522213 T1 ATE522213 T1 AT E522213T1 AT 02076763 T AT02076763 T AT 02076763T AT 02076763 T AT02076763 T AT 02076763T AT E522213 T1 ATE522213 T1 AT E522213T1
- Authority
- AT
- Austria
- Prior art keywords
- membed
- heteroring
- derivatives
- production
- medicinal products
- Prior art date
Links
- 229940126601 medicinal product Drugs 0.000 title 1
Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
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- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9912643A FR2799461B1 (fr) | 1999-10-11 | 1999-10-11 | Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments |
FR0010151A FR2812546B1 (fr) | 2000-08-01 | 2000-08-01 | Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments |
FR0011169 | 2000-09-01 |
Publications (1)
Publication Number | Publication Date |
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ATE522213T1 true ATE522213T1 (de) | 2011-09-15 |
Family
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Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
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AT02076763T ATE522213T1 (de) | 1999-10-11 | 2000-10-10 | Fünfgliedrige-heteroringderivate , ihre herstellung und ihre verwendung als arzneimittel |
AT00967988T ATE338547T1 (de) | 1999-10-11 | 2000-10-10 | Fünfgliedrige derivate von heterozyklen und ihre verwendung als monoaminoxidase-inhibitoren |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
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AT00967988T ATE338547T1 (de) | 1999-10-11 | 2000-10-10 | Fünfgliedrige derivate von heterozyklen und ihre verwendung als monoaminoxidase-inhibitoren |
Country Status (27)
Country | Link |
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US (4) | US20070021390A1 (de) |
EP (3) | EP1223933B1 (de) |
JP (1) | JP4972263B2 (de) |
KR (2) | KR20070068491A (de) |
CN (1) | CN100488506C (de) |
AR (1) | AR029006A1 (de) |
AT (2) | ATE522213T1 (de) |
AU (1) | AU783129B2 (de) |
BR (1) | BR0014649A (de) |
CA (1) | CA2388505C (de) |
CY (1) | CY1106237T1 (de) |
CZ (1) | CZ304331B6 (de) |
DE (1) | DE60030574T2 (de) |
DK (2) | DK1223933T3 (de) |
ES (2) | ES2544856T3 (de) |
HK (1) | HK1049957B (de) |
HU (1) | HU228254B1 (de) |
IL (3) | IL148896A0 (de) |
MX (1) | MXPA02003665A (de) |
MY (1) | MY145388A (de) |
NO (1) | NO331874B1 (de) |
NZ (2) | NZ518304A (de) |
PL (1) | PL215580B1 (de) |
PT (2) | PT1589007E (de) |
RU (1) | RU2271355C2 (de) |
TW (2) | TWI283577B (de) |
WO (1) | WO2001026656A2 (de) |
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TWI283577B (en) * | 1999-10-11 | 2007-07-11 | Sod Conseils Rech Applic | Pharmaceutical composition of imidazole derivatives acting as modulators of sodium channels and the use thereof |
FR2823208B1 (fr) * | 2001-04-10 | 2004-03-19 | Sod Conseils Rech Applic | Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments |
FR2818978B1 (fr) * | 2000-12-28 | 2003-02-28 | Sod Conseils Rech Applic | Modulateurs de canaux sodiques derives de 2-piperidylimidazoles |
TWI248438B (en) * | 2001-04-10 | 2006-02-01 | Sod Conseils Rech Applic | Derivatives of heterocycles with 5 members, their preparation and their use as medicaments |
FR2825926A1 (fr) * | 2001-06-14 | 2002-12-20 | Sod Conseils Rech Applic | Derives d'imidazoles modulant les canaux sodiques |
HU228783B1 (en) | 2001-07-26 | 2013-05-28 | Greenearth Cleaning | Dry cleaning apparatus and method capable of utilizing a siloxane solvent |
US6815555B2 (en) | 2001-09-26 | 2004-11-09 | Theravance, Inc. | Substituted phenol compounds useful for anesthesia and sedation |
WO2003035073A1 (en) | 2001-10-25 | 2003-05-01 | Astrazeneca Ab | Isoxazoline derivatives useful as antimicrobials |
WO2003048140A1 (fr) | 2001-12-03 | 2003-06-12 | Japan Tobacco Inc. | Compose azole et utilisation medicinale de celui-ci |
FR2835254B1 (fr) * | 2002-01-25 | 2006-04-07 | Sod Conseils Rech Applic | Derives de thiazoles dans le traitement de maladies neurologiques |
FR2842808B1 (fr) * | 2002-07-25 | 2004-09-10 | Sod Conseils Rech Applic | Nouveaux derives d'arylimidazoles, leur preparation et leurs applications therapeutiques |
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RU2352568C9 (ru) | 2002-08-09 | 2009-06-27 | Астразенека Аб | [1,2,4]оксадиазолы (варианты), способ их получения, фармацевтическая композиция и способ ингибирования активации метаботропных глютаматных рецепторов-5 |
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US7732162B2 (en) | 2003-05-05 | 2010-06-08 | Probiodrug Ag | Inhibitors of glutaminyl cyclase for treating neurodegenerative diseases |
TWI256952B (en) * | 2003-08-27 | 2006-06-21 | Sk Corp | Chroman carboxylic acid derivatives for the treatment of diabetes and lipid disorders |
EP1533295A1 (de) * | 2003-11-24 | 2005-05-25 | Newron Pharmaceuticals S.p.A. | Cyclopentylderivate |
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KR101220182B1 (ko) | 2009-02-25 | 2013-01-11 | 에스케이바이오팜 주식회사 | 치환된 아졸 유도체 화합물, 이를 포함하는 약제학적 조성물 및 이를 이용한 파킨슨씨 병 치료방법 |
EA022007B1 (ru) | 2009-09-11 | 2015-10-30 | Пробиодруг Аг | Гетероциклические производные в качестве ингибиторов глутаминилциклазы |
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