DK1223933T3 - 5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer - Google Patents
5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorerInfo
- Publication number
- DK1223933T3 DK1223933T3 DK00967988T DK00967988T DK1223933T3 DK 1223933 T3 DK1223933 T3 DK 1223933T3 DK 00967988 T DK00967988 T DK 00967988T DK 00967988 T DK00967988 T DK 00967988T DK 1223933 T3 DK1223933 T3 DK 1223933T3
- Authority
- DK
- Denmark
- Prior art keywords
- heterocycles
- monoamine oxidase
- oxidase inhibitors
- membered derivatives
- membered
- Prior art date
Links
- 229940123685 Monoamine oxidase inhibitor Drugs 0.000 title 1
- 125000000623 heterocyclic group Chemical group 0.000 title 1
- 239000002899 monoamine oxidase inhibitor Substances 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
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- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D277/28—Radicals substituted by nitrogen atoms
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9912643A FR2799461B1 (fr) | 1999-10-11 | 1999-10-11 | Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments |
FR0010151A FR2812546B1 (fr) | 2000-08-01 | 2000-08-01 | Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments |
FR0011169 | 2000-09-01 |
Publications (1)
Publication Number | Publication Date |
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DK1223933T3 true DK1223933T3 (da) | 2007-01-15 |
Family
ID=27248695
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
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DK00967988T DK1223933T3 (da) | 1999-10-11 | 2000-10-10 | 5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer |
DK05076749.0T DK1589007T3 (en) | 1999-10-11 | 2000-10-10 | 5-link heterocycle derivatives, their preparation and use as pharmaceuticals |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
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DK05076749.0T DK1589007T3 (en) | 1999-10-11 | 2000-10-10 | 5-link heterocycle derivatives, their preparation and use as pharmaceuticals |
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Country | Link |
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US (4) | US20070021390A1 (de) |
EP (3) | EP1223933B1 (de) |
JP (1) | JP4972263B2 (de) |
KR (2) | KR100731698B1 (de) |
CN (1) | CN100488506C (de) |
AR (1) | AR029006A1 (de) |
AT (2) | ATE522213T1 (de) |
AU (1) | AU783129B2 (de) |
BR (1) | BR0014649A (de) |
CA (1) | CA2388505C (de) |
CY (1) | CY1106237T1 (de) |
CZ (1) | CZ304331B6 (de) |
DE (1) | DE60030574T2 (de) |
DK (2) | DK1223933T3 (de) |
ES (2) | ES2270873T3 (de) |
HK (1) | HK1049957B (de) |
HU (1) | HU228254B1 (de) |
IL (3) | IL148896A0 (de) |
MX (1) | MXPA02003665A (de) |
MY (1) | MY145388A (de) |
NO (1) | NO331874B1 (de) |
NZ (2) | NZ518304A (de) |
PL (1) | PL215580B1 (de) |
PT (2) | PT1589007E (de) |
RU (1) | RU2271355C2 (de) |
TW (2) | TWI292316B (de) |
WO (1) | WO2001026656A2 (de) |
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US7291641B2 (en) * | 1999-10-11 | 2007-11-06 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | Derivatives of heterocycles with 5 members, their preparation and their use as medicaments |
FR2818978B1 (fr) * | 2000-12-28 | 2003-02-28 | Sod Conseils Rech Applic | Modulateurs de canaux sodiques derives de 2-piperidylimidazoles |
TWI248438B (en) * | 2001-04-10 | 2006-02-01 | Sod Conseils Rech Applic | Derivatives of heterocycles with 5 members, their preparation and their use as medicaments |
FR2825926A1 (fr) * | 2001-06-14 | 2002-12-20 | Sod Conseils Rech Applic | Derives d'imidazoles modulant les canaux sodiques |
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JP2005512975A (ja) | 2001-10-25 | 2005-05-12 | アストラゼネカ アクチボラグ | 抗菌薬として有用なイソキサゾリン誘導体 |
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FR2835254B1 (fr) * | 2002-01-25 | 2006-04-07 | Sod Conseils Rech Applic | Derives de thiazoles dans le traitement de maladies neurologiques |
FR2842808B1 (fr) | 2002-07-25 | 2004-09-10 | Sod Conseils Rech Applic | Nouveaux derives d'arylimidazoles, leur preparation et leurs applications therapeutiques |
JP2006506340A (ja) * | 2002-08-09 | 2006-02-23 | アストラゼネカ アクチボラグ | 代謝調節型グルタミン酸受容体5のモジュレーターとしてのオキサジアゾール |
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MXPA05010945A (es) * | 2003-04-09 | 2005-11-25 | Japan Tobacco Inc | Compuesto pentaciclico heteroaromatico y uso medicinal del mismo. |
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DK2142514T3 (da) | 2007-04-18 | 2015-03-23 | Probiodrug Ag | Thioureaderivater som glutaminylcyclase-inhibitorer |
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EP2542549B1 (de) | 2010-03-03 | 2016-05-11 | Probiodrug AG | Glutaminylcyclase-hemmer |
BR112012022478B1 (pt) | 2010-03-10 | 2021-09-21 | Probiodrug Ag | Inibidores heterocíclicos de glutaminil ciclase (qc, ec 2.3.2.5), seu processo de preparação, e composição farmacêutica |
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2000
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- 2000-10-10 HU HU0203841A patent/HU228254B1/hu not_active IP Right Cessation
- 2000-10-10 EP EP00967988A patent/EP1223933B1/de not_active Expired - Lifetime
- 2000-10-10 DK DK00967988T patent/DK1223933T3/da active
- 2000-10-10 AT AT02076763T patent/ATE522213T1/de not_active IP Right Cessation
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- 2000-10-10 CZ CZ2002-1292A patent/CZ304331B6/cs not_active IP Right Cessation
- 2000-10-10 WO PCT/FR2000/002805 patent/WO2001026656A2/fr active Application Filing
- 2000-10-10 EP EP02076763A patent/EP1228760B1/de not_active Expired - Lifetime
- 2000-10-10 MY MYPI20004725A patent/MY145388A/en unknown
- 2000-10-10 PT PT50767490T patent/PT1589007E/pt unknown
- 2000-10-10 KR KR1020077013941A patent/KR20070068491A/ko active IP Right Grant
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- 2000-10-10 CA CA2388505A patent/CA2388505C/fr not_active Expired - Fee Related
- 2000-10-10 DK DK05076749.0T patent/DK1589007T3/en active
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- 2000-10-10 AT AT00967988T patent/ATE338547T1/de active
- 2000-10-10 RU RU2002112227/15A patent/RU2271355C2/ru not_active IP Right Cessation
- 2000-10-10 BR BR0014649-8A patent/BR0014649A/pt not_active IP Right Cessation
- 2000-10-10 EP EP05076749.0A patent/EP1589007B1/de not_active Expired - Lifetime
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- 2007-02-20 US US11/708,531 patent/US20070179153A1/en not_active Abandoned
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