AR033985A1 - Peptidos inhibidores de proteasa serina-ns3 del virus de la hepatitis c, composicion farmaceutica que los comprende, un metodo para su preparacion, uso de los mismos para la fabricacion de un medicamento y un metodo de modulacion de la actividad de la proteasa del virus de la hepatitis c - Google Patents

Peptidos inhibidores de proteasa serina-ns3 del virus de la hepatitis c, composicion farmaceutica que los comprende, un metodo para su preparacion, uso de los mismos para la fabricacion de un medicamento y un metodo de modulacion de la actividad de la proteasa del virus de la hepatitis c

Info

Publication number
AR033985A1
AR033985A1 ARP010103450A ARP010103450A AR033985A1 AR 033985 A1 AR033985 A1 AR 033985A1 AR P010103450 A ARP010103450 A AR P010103450A AR P010103450 A ARP010103450 A AR P010103450A AR 033985 A1 AR033985 A1 AR 033985A1
Authority
AR
Argentina
Prior art keywords
conhch
alkyl
present
absent
aryl
Prior art date
Application number
ARP010103450A
Other languages
English (en)
Spanish (es)
Original Assignee
Dendreon Corp
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22822095&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR033985(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dendreon Corp, Schering Corp filed Critical Dendreon Corp
Publication of AR033985A1 publication Critical patent/AR033985A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02—Linear peptides containing at least one abnormal peptide link
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
ARP010103450A 2000-07-21 2001-07-20 Peptidos inhibidores de proteasa serina-ns3 del virus de la hepatitis c, composicion farmaceutica que los comprende, un metodo para su preparacion, uso de los mismos para la fabricacion de un medicamento y un metodo de modulacion de la actividad de la proteasa del virus de la hepatitis c AR033985A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US22010800P 2000-07-21 2000-07-21

Publications (1)

Publication Number Publication Date
AR033985A1 true AR033985A1 (es) 2004-01-21

Family

ID=22822095

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP010103450A AR033985A1 (es) 2000-07-21 2001-07-20 Peptidos inhibidores de proteasa serina-ns3 del virus de la hepatitis c, composicion farmaceutica que los comprende, un metodo para su preparacion, uso de los mismos para la fabricacion de un medicamento y un metodo de modulacion de la actividad de la proteasa del virus de la hepatitis c
ARP080105033A AR069373A2 (es) 2000-07-21 2008-11-19 Peptidos inhibidores de proteasa serina-ns3 del virus de la hepatitis c, y uso de los mismos para la fabricacion de un medicamento

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP080105033A AR069373A2 (es) 2000-07-21 2008-11-19 Peptidos inhibidores de proteasa serina-ns3 del virus de la hepatitis c, y uso de los mismos para la fabricacion de un medicamento

Country Status (31)

Country Link
US (4) US7012066B2 (OSRAM)
EP (1) EP1385870B1 (OSRAM)
JP (3) JP4298289B2 (OSRAM)
KR (2) KR100939155B1 (OSRAM)
CN (3) CN1498224A (OSRAM)
AR (2) AR033985A1 (OSRAM)
AT (1) ATE461207T1 (OSRAM)
AU (2) AU2001276988B2 (OSRAM)
BR (1) BR0112540A (OSRAM)
CA (1) CA2410662C (OSRAM)
CY (2) CY1112267T1 (OSRAM)
CZ (1) CZ303213B6 (OSRAM)
DE (2) DE60141608D1 (OSRAM)
DK (1) DK1385870T3 (OSRAM)
EC (1) ECSP034438A (OSRAM)
ES (1) ES2341534T3 (OSRAM)
HU (1) HU229997B1 (OSRAM)
IL (2) IL153670A0 (OSRAM)
LU (1) LU91910I2 (OSRAM)
MX (1) MXPA03000627A (OSRAM)
MY (2) MY139078A (OSRAM)
NO (2) NO332329B1 (OSRAM)
NZ (1) NZ523782A (OSRAM)
PL (1) PL206255B1 (OSRAM)
PT (1) PT1385870E (OSRAM)
RU (2) RU2355700C9 (OSRAM)
SI (1) SI1385870T1 (OSRAM)
SK (1) SK288064B6 (OSRAM)
TW (1) TWI324611B (OSRAM)
WO (1) WO2002008244A2 (OSRAM)
ZA (1) ZA200210312B (OSRAM)

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* Cited by examiner, † Cited by third party
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