DK2114924T3 - Co-krystaller og farmaceutiske sammensætninger omfattende disse - Google Patents

Co-krystaller og farmaceutiske sammensætninger omfattende disse

Info

Publication number
DK2114924T3
DK2114924T3 DK08726147.5T DK08726147T DK2114924T3 DK 2114924 T3 DK2114924 T3 DK 2114924T3 DK 08726147 T DK08726147 T DK 08726147T DK 2114924 T3 DK2114924 T3 DK 2114924T3
Authority
DK
Denmark
Prior art keywords
crystals
pharmaceutical compositions
comprehensive
compositions comprehensive
pharmaceutical
Prior art date
Application number
DK08726147.5T
Other languages
English (en)
Inventor
Patrick R Connelly
Irina Kadiyala
Kathy Stavropolus
Yuegang Zhang
Steve Johnston
Govinda Rao Bhisetti
Valdas Jurkauskas
Peter Rose
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Application granted granted Critical
Publication of DK2114924T3 publication Critical patent/DK2114924T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/07—Tetrapeptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Peptides Or Proteins (AREA)
DK08726147.5T 2007-02-27 2008-02-27 Co-krystaller og farmaceutiske sammensætninger omfattende disse DK2114924T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US90358707P 2007-02-27 2007-02-27
PCT/US2008/002568 WO2008106151A2 (en) 2007-02-27 2008-02-27 Co-crystals and pharmaceutical compositions comprising the same

Publications (1)

Publication Number Publication Date
DK2114924T3 true DK2114924T3 (da) 2012-04-10

Family

ID=39672669

Family Applications (1)

Application Number Title Priority Date Filing Date
DK08726147.5T DK2114924T3 (da) 2007-02-27 2008-02-27 Co-krystaller og farmaceutiske sammensætninger omfattende disse

Country Status (28)

Country Link
US (1) US8759353B2 (da)
EP (3) EP2463284A1 (da)
JP (1) JP2010519330A (da)
KR (1) KR20090115970A (da)
CN (1) CN101687856A (da)
AP (1) AP2009004960A0 (da)
AR (1) AR065498A1 (da)
AT (1) ATE542815T1 (da)
AU (1) AU2008219607B2 (da)
BR (1) BRPI0807907A2 (da)
CA (1) CA2679312A1 (da)
CO (1) CO6220963A2 (da)
CY (1) CY1112865T1 (da)
DK (1) DK2114924T3 (da)
EA (1) EA200970806A1 (da)
EC (1) ECSP099600A (da)
ES (1) ES2379905T3 (da)
GE (1) GEP20125645B (da)
HR (1) HRP20120330T1 (da)
IL (1) IL200616A0 (da)
MX (1) MX2009009182A (da)
NZ (1) NZ579442A (da)
PL (1) PL2114924T3 (da)
PT (1) PT2114924E (da)
RS (1) RS52306B (da)
SI (1) SI2114924T1 (da)
TW (1) TW200846343A (da)
WO (1) WO2008106151A2 (da)

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ITMI20131839A1 (it) * 2013-11-06 2015-05-07 Dipharma Francis Srl Co-cristallo di un farmaco antidepressivo
CN103819379A (zh) * 2014-02-18 2014-05-28 中国科学院上海药物研究所 维生素d3的胆甾烷醇共结晶及其制备方法和应用
CN105696066B (zh) * 2015-10-26 2018-07-03 西北大学 一种压片法制备共晶的方法
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CN113295723B (zh) * 2021-07-27 2021-09-28 西南石油大学 一种岩石中粘土矿物的分子模拟表征方法

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NZ579442A (en) 2012-02-24
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MX2009009182A (es) 2009-09-04
US8759353B2 (en) 2014-06-24
CA2679312A1 (en) 2008-09-04
CO6220963A2 (es) 2010-11-19
WO2008106151A2 (en) 2008-09-04
ECSP099600A (es) 2009-09-29
ES2379905T3 (es) 2012-05-04
KR20090115970A (ko) 2009-11-10
PL2114924T3 (pl) 2012-07-31
CY1112865T1 (el) 2016-04-13
EP2463284A1 (en) 2012-06-13
TW200846343A (en) 2008-12-01
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US20110059987A1 (en) 2011-03-10
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AR065498A1 (es) 2009-06-10
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AU2008219607A1 (en) 2008-09-04
EP2114924A2 (en) 2009-11-11
RS52306B (en) 2012-12-31
EA200970806A1 (ru) 2010-08-30
EP2114924B1 (en) 2012-01-25
CN101687856A (zh) 2010-03-31
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IL200616A0 (en) 2010-05-17
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