DK2069352T3 - Bestemte kemiske enheder, sammensætninger og fremgangsmåder - Google Patents

Bestemte kemiske enheder, sammensætninger og fremgangsmåder

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Publication number
DK2069352T3
DK2069352T3 DK07810993.1T DK07810993T DK2069352T3 DK 2069352 T3 DK2069352 T3 DK 2069352T3 DK 07810993 T DK07810993 T DK 07810993T DK 2069352 T3 DK2069352 T3 DK 2069352T3
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DK07810993.1T
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DK2069352T5 (da
Inventor
Alex Muci
Jeffrey T Finer
Pu-Ping Lu
Alan James Russell
Bradley P Morgan
David J Morgans Jr
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Cytokinetics Inc
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Publication of DK2069352T3 publication Critical patent/DK2069352T3/da
Publication of DK2069352T5 publication Critical patent/DK2069352T5/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/04Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/06Anabolic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Pulmonology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Nutrition Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK07810993.1T 2006-08-02 2007-08-01 Bestemte kemiske enheder, sammensætninger og fremgangsmåder DK2069352T5 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US83527206P 2006-08-02 2006-08-02
US92105407P 2007-03-30 2007-03-30
PCT/US2007/017235 WO2008016669A2 (en) 2006-08-02 2007-08-01 Certain chemical entities, compositions and methods

Publications (2)

Publication Number Publication Date
DK2069352T3 true DK2069352T3 (da) 2013-12-02
DK2069352T5 DK2069352T5 (da) 2017-04-03

Family

ID=38997712

Family Applications (2)

Application Number Title Priority Date Filing Date
DK13151376.4T DK2583970T3 (da) 2006-08-02 2007-08-01 Bestemte kemiske enheder, sammensætninger og fremgangsmåder omfattende imidazopyrimidiner
DK07810993.1T DK2069352T5 (da) 2006-08-02 2007-08-01 Bestemte kemiske enheder, sammensætninger og fremgangsmåder

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK13151376.4T DK2583970T3 (da) 2006-08-02 2007-08-01 Bestemte kemiske enheder, sammensætninger og fremgangsmåder omfattende imidazopyrimidiner

Country Status (27)

Country Link
US (3) US7598248B2 (da)
EP (4) EP2666777A1 (da)
JP (4) JP5249217B2 (da)
KR (1) KR101410453B1 (da)
CN (1) CN102993204A (da)
AR (1) AR062196A1 (da)
AU (1) AU2007281468B2 (da)
BR (1) BRPI0714725B1 (da)
CA (1) CA2659336C (da)
CL (1) CL2007002252A1 (da)
CO (1) CO6160237A2 (da)
DK (2) DK2583970T3 (da)
EA (1) EA017925B1 (da)
ES (2) ES2439590T3 (da)
HK (3) HK1131785A1 (da)
HR (1) HRP20160036T1 (da)
HU (1) HUE026571T2 (da)
IL (1) IL196767A (da)
MX (1) MX2009001170A (da)
NZ (1) NZ574888A (da)
PE (1) PE20080524A1 (da)
PL (2) PL2069352T3 (da)
PT (2) PT2583970E (da)
RS (1) RS54542B1 (da)
TW (1) TWI386412B (da)
WO (1) WO2008016669A2 (da)
ZA (1) ZA200900976B (da)

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EP2069352B1 (en) 2013-10-09
JP2013173762A (ja) 2013-09-05
EP2666777A1 (en) 2013-11-27
ZA200900976B (en) 2009-12-30
EP2995619A1 (en) 2016-03-16
JP6538809B2 (ja) 2019-07-03
PL2069352T3 (pl) 2014-03-31
KR20090045303A (ko) 2009-05-07
IL196767A (en) 2013-09-30
EP2069352A4 (en) 2010-10-27
JP5746254B2 (ja) 2015-07-08
BRPI0714725A2 (pt) 2013-10-15
PT2069352E (pt) 2014-01-02
AU2007281468A1 (en) 2008-02-07
CO6160237A2 (es) 2010-05-20
KR101410453B1 (ko) 2014-06-27
PT2583970E (pt) 2016-02-08
WO2008016669A2 (en) 2008-02-07
HK1184446A1 (zh) 2014-01-24
EP2069352B9 (en) 2017-03-15
JP2018058878A (ja) 2018-04-12
EA017925B1 (ru) 2013-04-30
TW200825087A (en) 2008-06-16
US7598248B2 (en) 2009-10-06
BRPI0714725B1 (pt) 2021-05-25
ES2558517T3 (es) 2016-02-04
TWI386412B (zh) 2013-02-21
US7956056B2 (en) 2011-06-07
MX2009001170A (es) 2009-05-21
AU2007281468B2 (en) 2012-12-06
JP5249217B2 (ja) 2013-07-31
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EP2583970A1 (en) 2013-04-24
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