US20110046076A1 - Pharmaceutical composition, methods for treating and uses thereof - Google Patents
Pharmaceutical composition, methods for treating and uses thereof Download PDFInfo
- Publication number
- US20110046076A1 US20110046076A1 US12/703,988 US70398810A US2011046076A1 US 20110046076 A1 US20110046076 A1 US 20110046076A1 US 70398810 A US70398810 A US 70398810A US 2011046076 A1 US2011046076 A1 US 2011046076A1
- Authority
- US
- United States
- Prior art keywords
- inhibitor
- obesity
- antidiabetic agent
- patient
- glucose
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- AACOGWZOMPLOCZ-ZQGJOIPISA-N CCC1=CC=C(CC2=C(C#N)C=C(C)C([C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)=C2)C=C1 Chemical compound CCC1=CC=C(CC2=C(C#N)C=C(C)C([C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)=C2)C=C1 AACOGWZOMPLOCZ-ZQGJOIPISA-N 0.000 description 1
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Images
Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
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- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid, pantothenic acid
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- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
- A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Molecular Biology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Child & Adolescent Psychology (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US12/703,988 US20110046076A1 (en) | 2009-02-13 | 2010-02-11 | Pharmaceutical composition, methods for treating and uses thereof |
| US13/912,599 US10406172B2 (en) | 2009-02-13 | 2013-06-07 | Pharmaceutical composition, methods for treating and uses thereof |
| US16/452,719 US20200085851A1 (en) | 2009-02-13 | 2019-06-26 | Pharmaceutical composition, methods for treating and uses thereof |
| US17/176,450 US20210346415A1 (en) | 2009-02-13 | 2021-02-16 | Pharmaceutical composition, methods for treating and uses thereof |
| US18/320,462 US20230285432A1 (en) | 2009-02-13 | 2023-05-19 | Pharmaceutical composition, methods for treating and uses thereof |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US15230209P | 2009-02-13 | 2009-02-13 | |
| US12/703,988 US20110046076A1 (en) | 2009-02-13 | 2010-02-11 | Pharmaceutical composition, methods for treating and uses thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| US13/912,599 Continuation US10406172B2 (en) | 2009-02-13 | 2013-06-07 | Pharmaceutical composition, methods for treating and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| US20110046076A1 true US20110046076A1 (en) | 2011-02-24 |
Family
ID=42109921
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| US12/703,988 Abandoned US20110046076A1 (en) | 2009-02-13 | 2010-02-11 | Pharmaceutical composition, methods for treating and uses thereof |
| US13/912,599 Active 2030-06-15 US10406172B2 (en) | 2009-02-13 | 2013-06-07 | Pharmaceutical composition, methods for treating and uses thereof |
| US16/452,719 Abandoned US20200085851A1 (en) | 2009-02-13 | 2019-06-26 | Pharmaceutical composition, methods for treating and uses thereof |
| US17/176,450 Abandoned US20210346415A1 (en) | 2009-02-13 | 2021-02-16 | Pharmaceutical composition, methods for treating and uses thereof |
| US18/320,462 Pending US20230285432A1 (en) | 2009-02-13 | 2023-05-19 | Pharmaceutical composition, methods for treating and uses thereof |
Family Applications After (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| US13/912,599 Active 2030-06-15 US10406172B2 (en) | 2009-02-13 | 2013-06-07 | Pharmaceutical composition, methods for treating and uses thereof |
| US16/452,719 Abandoned US20200085851A1 (en) | 2009-02-13 | 2019-06-26 | Pharmaceutical composition, methods for treating and uses thereof |
| US17/176,450 Abandoned US20210346415A1 (en) | 2009-02-13 | 2021-02-16 | Pharmaceutical composition, methods for treating and uses thereof |
| US18/320,462 Pending US20230285432A1 (en) | 2009-02-13 | 2023-05-19 | Pharmaceutical composition, methods for treating and uses thereof |
Country Status (38)
| Country | Link |
|---|---|
| US (5) | US20110046076A1 (ko) |
| EP (2) | EP2395983B1 (ko) |
| JP (1) | JP5685550B2 (ko) |
| KR (1) | KR101694136B1 (ko) |
| CN (2) | CN102307577A (ko) |
| AP (1) | AP2011005794A0 (ko) |
| AR (1) | AR075421A1 (ko) |
| AU (1) | AU2010212867B2 (ko) |
| BR (1) | BRPI1008560B1 (ko) |
| CA (1) | CA2751834C (ko) |
| CL (1) | CL2011001735A1 (ko) |
| CO (1) | CO6410286A2 (ko) |
| CY (1) | CY1123253T1 (ko) |
| DK (1) | DK2395983T3 (ko) |
| EA (1) | EA022349B1 (ko) |
| EC (1) | ECSP11011277A (ko) |
| ES (1) | ES2797503T3 (ko) |
| GE (1) | GEP20135962B (ko) |
| HK (1) | HK1213820A1 (ko) |
| HR (1) | HRP20200828T1 (ko) |
| HU (1) | HUE050287T2 (ko) |
| IL (1) | IL213746A0 (ko) |
| LT (1) | LT2395983T (ko) |
| MA (1) | MA33046B1 (ko) |
| MX (1) | MX339194B (ko) |
| MY (1) | MY160123A (ko) |
| NZ (1) | NZ594487A (ko) |
| PE (1) | PE20120017A1 (ko) |
| PL (1) | PL2395983T3 (ko) |
| PT (1) | PT2395983T (ko) |
| RS (1) | RS60438B1 (ko) |
| SG (1) | SG173619A1 (ko) |
| SI (1) | SI2395983T1 (ko) |
| TN (1) | TN2011000415A1 (ko) |
| TW (1) | TWI481620B (ko) |
| UA (1) | UA102429C2 (ko) |
| UY (1) | UY32441A (ko) |
| WO (1) | WO2010092125A1 (ko) |
Cited By (52)
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