UA78032C2 - Sulfonyl derivatives as histone deacetylase inhibitors - Google Patents

Sulfonyl derivatives as histone deacetylase inhibitors Download PDF

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Publication number
UA78032C2
UA78032C2 UA20041008336A UA20041008336A UA78032C2 UA 78032 C2 UA78032 C2 UA 78032C2 UA 20041008336 A UA20041008336 A UA 20041008336A UA 20041008336 A UA20041008336 A UA 20041008336A UA 78032 C2 UA78032 C2 UA 78032C2
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UA
Ukraine
Prior art keywords
alkyl
amino
valkyl
hydroxyc
dalalkyl
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UA20041008336A
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English (en)
Ukrainian (uk)
Inventor
Brandt Sven Franciscus Ann Van
Marc Gustaaf Celine Verdonck
Oleksii Borysovych Diatkin
Original Assignee
Janssen Pharmaceutica Nv
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Priority claimed from PCT/EP2003/002516 external-priority patent/WO2003076422A1/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of UA78032C2 publication Critical patent/UA78032C2/uk

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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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