TWI484962B - 作為jak抑制劑之3-〔4-(7h-吡咯并〔2,3-d〕嘧啶-4-基)-1h-吡唑-1-基〕辛烷或庚腈 - Google Patents

作為jak抑制劑之3-〔4-(7h-吡咯并〔2,3-d〕嘧啶-4-基)-1h-吡唑-1-基〕辛烷或庚腈 Download PDF

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TWI484962B
TWI484962B TW099116415A TW99116415A TWI484962B TW I484962 B TWI484962 B TW I484962B TW 099116415 A TW099116415 A TW 099116415A TW 99116415 A TW99116415 A TW 99116415A TW I484962 B TWI484962 B TW I484962B
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compound
pharmaceutically acceptable
acceptable salt
pyrrolo
pyrimidin
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TW099116415A
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TW201106951A (en
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Yun-Long Li
James D Rodgers
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Incyte Corp
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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TW099116415A 2009-05-22 2010-05-21 作為jak抑制劑之3-〔4-(7h-吡咯并〔2,3-d〕嘧啶-4-基)-1h-吡唑-1-基〕辛烷或庚腈 TWI484962B (zh)

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US18058209P 2009-05-22 2009-05-22

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TW201106951A TW201106951A (en) 2011-03-01
TWI484962B true TWI484962B (zh) 2015-05-21

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