TWI319320B - 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions - Google Patents

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

Info

Publication number
TWI319320B
TWI319320B TW092122890A TW92122890A TWI319320B TW I319320 B TWI319320 B TW I319320B TW 092122890 A TW092122890 A TW 092122890A TW 92122890 A TW92122890 A TW 92122890A TW I319320 B TWI319320 B TW I319320B
Authority
TW
Taiwan
Prior art keywords
xanthines
piperidin
amino
preparation
pharmaceutical compositions
Prior art date
Application number
TW092122890A
Other languages
English (en)
Chinese (zh)
Other versions
TW200404542A (en
Inventor
Himmelsbach Frank
Eckhardt Matthias
Langkopf Elke
Mark Michael
Maier Roland
R H Lotz Ralf
Tadayyon Mohammad
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TWI319320(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/de
Priority claimed from DE10312353A external-priority patent/DE10312353A1/de
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of TW200404542A publication Critical patent/TW200404542A/zh
Application granted granted Critical
Publication of TWI319320B publication Critical patent/TWI319320B/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
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TW092122890A 2002-08-21 2003-08-20 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions TWI319320B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (de) 2002-08-21 2002-08-21 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
DE10312353A DE10312353A1 (de) 2003-03-20 2003-03-20 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel

Publications (2)

Publication Number Publication Date
TW200404542A TW200404542A (en) 2004-04-01
TWI319320B true TWI319320B (en) 2010-01-11

Family

ID=31947613

Family Applications (3)

Application Number Title Priority Date Filing Date
TW092122890A TWI319320B (en) 2002-08-21 2003-08-20 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
TW101137343A TWI469783B (zh) 2002-08-21 2003-08-20 ８-〔３-胺基-六氫吡啶-１-基〕-黃嘌呤，其製備方法及作為醫藥組合物之用途
TW098125780A TWI388325B (zh) 2002-08-21 2003-08-20 ８-〔３-胺基-六氫吡啶-１-基〕-黃嘌呤，其製備方法及作為醫藥組合物之用途

Family Applications After (2)

Application Number Title Priority Date Filing Date
TW101137343A TWI469783B (zh) 2002-08-21 2003-08-20 ８-〔３-胺基-六氫吡啶-１-基〕-黃嘌呤，其製備方法及作為醫藥組合物之用途
TW098125780A TWI388325B (zh) 2002-08-21 2003-08-20 ８-〔３-胺基-六氫吡啶-１-基〕-黃嘌呤，其製備方法及作為醫藥組合物之用途

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EP (6) EP2070539A1 (enExample)
JP (6) JP4233524B2 (enExample)
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