RU2422450C2 - Новые фосфорсодержащие тиромиметики - Google Patents

Новые фосфорсодержащие тиромиметики Download PDF

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RU2422450C2
RU2422450C2 RU2006117986/04A RU2006117986A RU2422450C2 RU 2422450 C2 RU2422450 C2 RU 2422450C2 RU 2006117986/04 A RU2006117986/04 A RU 2006117986/04A RU 2006117986 A RU2006117986 A RU 2006117986A RU 2422450 C2 RU2422450 C2 RU 2422450C2
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group
alkyl
independently selected
hydrogen
attached
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RU2006117986/04A
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Russian (ru)
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RU2006117986A (ru
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Марк Д. ЭРИОН (US)
Марк Д. ЭРИОН
Хонгджиан ДЖИАНГ (US)
Хонгджиан ДЖИАНГ
Серж Х. БОЙЕР (US)
Серж Х. БОЙЕР
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Метабазис Терапеутикс, Инк.
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    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
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    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
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    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
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    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
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    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
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    • C07F9/40—Esters thereof
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RU2006117986/04A 2003-11-19 2004-11-19 Новые фосфорсодержащие тиромиметики RU2422450C2 (ru)

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Application Number Priority Date Filing Date Title
US52383003P 2003-11-19 2003-11-19
US60/523,830 2003-11-19
US59852404P 2004-08-03 2004-08-03
US60/598,524 2004-08-03

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RU2006117986A RU2006117986A (ru) 2007-12-27
RU2422450C2 true RU2422450C2 (ru) 2011-06-27

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US (3) US7829552B2 (enExample)
EP (2) EP2428516A1 (enExample)
JP (1) JP2007512359A (enExample)
KR (1) KR20060109926A (enExample)
CN (1) CN1882327A (enExample)
AU (1) AU2004293013B2 (enExample)
BR (1) BRPI0416639A (enExample)
CA (1) CA2546601A1 (enExample)
RU (1) RU2422450C2 (enExample)
WO (1) WO2005051298A2 (enExample)

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WO2006128055A2 (en) * 2005-05-26 2006-11-30 Metabasis Therapeutics, Inc. Novel phosphorus-containing thyromimetics
JP2007512359A (ja) 2003-11-19 2007-05-17 メタバシス・セラピューティクス・インコーポレイテッド 新規なリン含有甲状腺ホルモン様物質
WO2005051898A2 (en) * 2003-11-20 2005-06-09 Eli Lilly And Company Vitamin d receptor modulators
EP1687258A2 (en) * 2003-11-20 2006-08-09 Eli Lilly And Company Vitamin d receptor modulators
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EP1689383A4 (en) 2009-02-18
US7514419B2 (en) 2009-04-07
AU2004293013A1 (en) 2005-06-09
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