NO309227B1 - Anvendelse av pyrazolopyrimidioner for fremstilling av et medikament for behandling av impotens - Google Patents

Anvendelse av pyrazolopyrimidioner for fremstilling av et medikament for behandling av impotens

Info

Publication number
NO309227B1
NO309227B1 NO954757A NO954757A NO309227B1 NO 309227 B1 NO309227 B1 NO 309227B1 NO 954757 A NO954757 A NO 954757A NO 954757 A NO954757 A NO 954757A NO 309227 B1 NO309227 B1 NO 309227B1
Authority
NO
Norway
Prior art keywords
alkyl
optionally substituted
cycloalkyl
pyrazolopyrimid
impotence
Prior art date
Application number
NO954757A
Other languages
English (en)
Other versions
NO309227B3 (no
NO954757D0 (no
NO954757L (no
Inventor
Peter Ellis
Nicholas Kenneth Terrett
Original Assignee
Pfizer Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10736901&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO309227(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Res & Dev filed Critical Pfizer Res & Dev
Publication of NO954757D0 publication Critical patent/NO954757D0/no
Publication of NO954757L publication Critical patent/NO954757L/no
Publication of NO309227B1 publication Critical patent/NO309227B1/no
Publication of NO309227B3 publication Critical patent/NO309227B3/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Reproductive Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Urology & Nephrology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Paper (AREA)
  • Hydroponics (AREA)
NO19954757A 1993-06-09 1995-11-24 Anvendelse av 5-[2-etoksy-5-(4-metyl-1-piperazinylsulfonyl)fenyl]-1-metyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-on for fremstilling av et medikament for behandling av erektil dysfunksjon NO309227B3 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB939311920A GB9311920D0 (en) 1993-06-09 1993-06-09 Therapeutic agents
PCT/EP1994/001580 WO1994028902A1 (en) 1993-06-09 1994-05-13 Pyrazolopyrimidinones for the treatment of impotence

Publications (4)

Publication Number Publication Date
NO954757D0 NO954757D0 (no) 1995-11-24
NO954757L NO954757L (no) 1995-11-24
NO309227B1 true NO309227B1 (no) 2001-01-02
NO309227B3 NO309227B3 (no) 2011-02-21

Family

ID=10736901

Family Applications (3)

Application Number Title Priority Date Filing Date
NO19954757A NO309227B3 (no) 1993-06-09 1995-11-24 Anvendelse av 5-[2-etoksy-5-(4-metyl-1-piperazinylsulfonyl)fenyl]-1-metyl-3-n-propyl-1,6-dihydro-7H-pyrazolo[4,3-d]pyrimidin-7-on for fremstilling av et medikament for behandling av erektil dysfunksjon
NO20000703A NO321622B1 (no) 1993-06-09 2000-02-11 Pyrazolopyridmidioner for behandling av kvinnelig seksuell dysfunksjon
NO20000702A NO325558B1 (no) 1993-06-09 2000-02-11 Anvendelse av cGMP PDEv-inhibitorer for fremstilling av medikamenter til behandling av erektil dysfunksjon.

Family Applications After (2)

Application Number Title Priority Date Filing Date
NO20000703A NO321622B1 (no) 1993-06-09 2000-02-11 Pyrazolopyridmidioner for behandling av kvinnelig seksuell dysfunksjon
NO20000702A NO325558B1 (no) 1993-06-09 2000-02-11 Anvendelse av cGMP PDEv-inhibitorer for fremstilling av medikamenter til behandling av erektil dysfunksjon.

Country Status (28)

Country Link
US (2) US6469012B1 (no)
EP (1) EP0702555B1 (no)
JP (4) JP2925034B2 (no)
KR (2) KR100262926B1 (no)
CN (2) CN1071118C (no)
AT (1) ATE163852T1 (no)
AU (1) AU676571C (no)
CA (1) CA2163446C (no)
CY (1) CY2099B1 (no)
CZ (1) CZ284946B6 (no)
DE (1) DE69408981T2 (no)
DK (1) DK0702555T3 (no)
EC (1) ECSP941102A (no)
ES (1) ES2113656T3 (no)
FI (1) FI955911A0 (no)
GB (2) GB9301192D0 (no)
GR (1) GR3026520T3 (no)
HU (1) HU227877B1 (no)
IL (3) IL121836A (no)
LV (1) LV12269B (no)
MY (1) MY111446A (no)
NO (3) NO309227B3 (no)
NZ (2) NZ266463A (no)
PL (1) PL311948A1 (no)
RU (1) RU2373938C9 (no)
TW (1) TW292971B (no)
WO (1) WO1994028902A1 (no)
ZA (1) ZA944018B (no)

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TW292971B (no) 1996-12-11
IL109873A (en) 1998-12-27
CY2099B1 (en) 2002-04-05
US20030027824A1 (en) 2003-02-06
CZ324295A3 (en) 1996-07-17
HU9501933D0 (en) 1995-09-28
HU227877B1 (en) 2012-05-29
NZ314110A (en) 2001-02-23
NO309227B3 (no) 2011-02-21
NO954757D0 (no) 1995-11-24
KR960702751A (ko) 1996-05-23
KR100262926B1 (ko) 2000-09-01
RU2130776C1 (ru) 1999-05-27
CA2163446C (en) 1998-07-07
ECSP941102A (es) 1994-12-15
GB9301192D0 (en) 1993-06-09
CN1742731B (zh) 2012-02-01
ZA944018B (en) 1995-12-08
MY111446A (en) 2000-05-31
AU6797394A (en) 1995-01-03
NZ266463A (en) 1997-03-24
CN1124926A (zh) 1996-06-19
EP0702555A1 (en) 1996-03-27
CN1071118C (zh) 2001-09-19
DE69408981D1 (de) 1998-04-16
JPH11286444A (ja) 1999-10-19
FI955911A (fi) 1995-12-08
HUT73420A (en) 1996-07-29
JPH11263728A (ja) 1999-09-28
NO20000702L (no) 1995-11-24
CA2163446A1 (en) 1994-12-22
CN1742731A (zh) 2006-03-08
NO20000702D0 (no) 2000-02-11
JPH09503996A (ja) 1997-04-22
PL311948A1 (en) 1996-03-18
CZ284946B6 (cs) 1999-04-14
ATE163852T1 (de) 1998-03-15
AU676571B2 (en) 1997-03-13
AU676571C (en) 2004-01-15
DE69408981T2 (de) 1998-07-02
NO321622B1 (no) 2006-06-12
LV12269B (en) 1999-08-20
EP0702555B1 (en) 1998-03-11
WO1994028902A1 (en) 1994-12-22
NO20000703L (no) 1995-11-24
NO954757L (no) 1995-11-24
GB9311920D0 (en) 1993-07-28
IL121836A0 (en) 1998-02-22
US6469012B1 (en) 2002-10-22
ES2113656T3 (es) 1998-05-01
FI955911A0 (fi) 1995-12-08

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