CN1742731B - 治疗雌性性机能障碍的吡唑并嘧啶酮类 - Google Patents
治疗雌性性机能障碍的吡唑并嘧啶酮类 Download PDFInfo
- Publication number
- CN1742731B CN1742731B CN011112603A CN01111260A CN1742731B CN 1742731 B CN1742731 B CN 1742731B CN 011112603 A CN011112603 A CN 011112603A CN 01111260 A CN01111260 A CN 01111260A CN 1742731 B CN1742731 B CN 1742731B
- Authority
- CN
- China
- Prior art keywords
- methyl
- pyl
- pro
- pyrazolo
- pyrimidin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Reproductive Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Gynecology & Obstetrics (AREA)
- Urology & Nephrology (AREA)
- Pregnancy & Childbirth (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Paper (AREA)
- Hydroponics (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Description
Claims (1)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB9311920.4 | 1993-06-09 | ||
GB939311920A GB9311920D0 (en) | 1993-06-09 | 1993-06-09 | Therapeutic agents |
Related Parent Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN94192386A Division CN1071118C (zh) | 1993-06-09 | 1994-05-13 | 用于治疗阳萎的吡唑并嘧啶酮类 |
Publications (2)
Publication Number | Publication Date |
---|---|
CN1742731A CN1742731A (zh) | 2006-03-08 |
CN1742731B true CN1742731B (zh) | 2012-02-01 |
Family
ID=10736901
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN011112603A Expired - Lifetime CN1742731B (zh) | 1993-06-09 | 1994-05-13 | 治疗雌性性机能障碍的吡唑并嘧啶酮类 |
CN94192386A Expired - Lifetime CN1071118C (zh) | 1993-06-09 | 1994-05-13 | 用于治疗阳萎的吡唑并嘧啶酮类 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN94192386A Expired - Lifetime CN1071118C (zh) | 1993-06-09 | 1994-05-13 | 用于治疗阳萎的吡唑并嘧啶酮类 |
Country Status (28)
Country | Link |
---|---|
US (2) | US6469012B1 (zh) |
EP (1) | EP0702555B1 (zh) |
JP (4) | JP2925034B2 (zh) |
KR (2) | KR100262926B1 (zh) |
CN (2) | CN1742731B (zh) |
AT (1) | ATE163852T1 (zh) |
AU (1) | AU676571C (zh) |
CA (1) | CA2163446C (zh) |
CY (1) | CY2099B1 (zh) |
CZ (1) | CZ284946B6 (zh) |
DE (1) | DE69408981T2 (zh) |
DK (1) | DK0702555T3 (zh) |
EC (1) | ECSP941102A (zh) |
ES (1) | ES2113656T3 (zh) |
FI (1) | FI955911A0 (zh) |
GB (2) | GB9301192D0 (zh) |
GR (1) | GR3026520T3 (zh) |
HU (1) | HU227877B1 (zh) |
IL (3) | IL121836A (zh) |
LV (1) | LV12269B (zh) |
MY (1) | MY111446A (zh) |
NO (3) | NO309227B3 (zh) |
NZ (2) | NZ314110A (zh) |
PL (1) | PL311948A1 (zh) |
RU (1) | RU2373938C9 (zh) |
TW (1) | TW292971B (zh) |
WO (1) | WO1994028902A1 (zh) |
ZA (1) | ZA944018B (zh) |
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GB9514464D0 (en) * | 1995-07-14 | 1995-09-13 | Glaxo Lab Sa | Medicaments |
GB9514473D0 (en) * | 1995-07-14 | 1995-09-13 | Glaxo Lab Sa | Chemical compounds |
ATE215950T1 (de) | 1996-05-10 | 2002-04-15 | Icos Corp | Carbolinderivate |
GB9612514D0 (en) * | 1996-06-14 | 1996-08-14 | Pfizer Ltd | Novel process |
DE19642284A1 (de) * | 1996-10-14 | 1998-04-16 | Merck Patent Gmbh | Pyrazolinone zur Behandlung von Potenzstörungen |
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IL132993A0 (en) * | 1997-05-29 | 2001-03-19 | Mochida Pharm Co Ltd | Therapeutic agent for erection failure |
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US20020025969A1 (en) * | 1997-07-09 | 2002-02-28 | Wolf-Georg Forssmann | Use of phosphordiesterase inhibitors in the treatment of prostatic diseases |
US20030077229A1 (en) * | 1997-10-01 | 2003-04-24 | Dugger Harry A. | Buccal, polar and non-polar spray or capsule containing cardiovascular or renal drugs |
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1993
- 1993-06-09 GB GB939301192A patent/GB9301192D0/en active Pending
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1994
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- 1994-05-13 CN CN94192386A patent/CN1071118C/zh not_active Expired - Lifetime
- 1994-05-13 DE DE69408981T patent/DE69408981T2/de not_active Revoked
- 1994-05-13 RU RU96100543/63A patent/RU2373938C9/ru active IP Right Maintenance
- 1994-05-13 US US08/549,792 patent/US6469012B1/en not_active Expired - Lifetime
- 1994-05-13 HU HU9501933A patent/HU227877B1/hu unknown
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- 1994-05-13 ES ES94916236T patent/ES2113656T3/es not_active Expired - Lifetime
- 1994-05-13 CZ CZ953242A patent/CZ284946B6/cs not_active IP Right Cessation
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1995
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- 1995-12-08 KR KR1019950705553A patent/KR960702751A/ko active Search and Examination
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1999
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2002
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EP0526004B1 (en) * | 1991-07-09 | 1997-10-08 | Pfizer Limited | Pyrazolopyrimidinone antianginal agents |
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