MX367324B - Sintesis de compuestos de ester y acido borico. - Google Patents

Sintesis de compuestos de ester y acido borico.

Info

Publication number
MX367324B
MX367324B MX2014005871A MX2014005871A MX367324B MX 367324 B MX367324 B MX 367324B MX 2014005871 A MX2014005871 A MX 2014005871A MX 2014005871 A MX2014005871 A MX 2014005871A MX 367324 B MX367324 B MX 367324B
Authority
MX
Mexico
Prior art keywords
acid compounds
synthesis
boronic ester
boronic
acid
Prior art date
Application number
MX2014005871A
Other languages
English (en)
Inventor
Fraser Pickersgill I
Bishop John
Koellner Christoph
Gomez Jean-Marc
Geiser Achim
Hett Robert
Ammoscato Vince
Munk Stephen
Lo Young
Chui Fang-Ting
R Kulkarni Vithalanand
Original Assignee
Millennium Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34968044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX367324(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Millennium Pharm Inc filed Critical Millennium Pharm Inc
Publication of MX367324B publication Critical patent/MX367324B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/04—Esters of boric acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Transplantation (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

La invención se refiere a la síntesis de compuestos de ácido y éster bóricos. Más particularmente, la invención se refiere a procesos sintéticos mejorados para la producción a gran escala de compuestos de ácido y éster bóricos, incluyendo el bortezomib inhibidor de la proteasoma de ácido bórico péptido.
MX2014005871A 2004-03-30 2005-03-24 Sintesis de compuestos de ester y acido borico. MX367324B (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US55753504P 2004-03-30 2004-03-30

Publications (1)

Publication Number Publication Date
MX367324B true MX367324B (es) 2019-08-15

Family

ID=34968044

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014005871A MX367324B (es) 2004-03-30 2005-03-24 Sintesis de compuestos de ester y acido borico.

Country Status (41)

Country Link
US (14) US7714159B2 (es)
EP (5) EP4008721B1 (es)
JP (4) JP4558039B2 (es)
KR (1) KR100939598B1 (es)
CN (5) CN108329337B (es)
AR (3) AR049374A1 (es)
AT (1) ATE521612T1 (es)
AU (1) AU2005230930B2 (es)
BR (1) BRPI0509587A (es)
CA (4) CA2853272A1 (es)
CL (2) CL2010000350A1 (es)
CR (1) CR8653A (es)
CY (3) CY1112053T1 (es)
DK (4) DK3385267T3 (es)
DO (1) DOP2011000293A (es)
EA (1) EA012927B1 (es)
EC (1) ECSP066960A (es)
ES (3) ES2899606T3 (es)
FI (1) FI4008721T3 (es)
HK (4) HK1100004A1 (es)
HR (4) HRP20212002T1 (es)
HU (1) HUE056859T2 (es)
IL (3) IL178250A (es)
LT (2) LT3385267T (es)
ME (1) ME01975B (es)
MX (1) MX367324B (es)
MY (1) MY145427A (es)
NL (3) NL1028639C2 (es)
NO (4) NO338905B1 (es)
NZ (3) NZ550522A (es)
PE (3) PE20142402A1 (es)
PL (4) PL2377869T3 (es)
PT (4) PT4008721T (es)
RS (4) RS65253B1 (es)
SG (5) SG182999A1 (es)
SI (4) SI1756121T1 (es)
TW (1) TWI386212B (es)
UA (1) UA90108C2 (es)
UY (3) UY28830A1 (es)
WO (1) WO2005097809A2 (es)
ZA (1) ZA200608689B (es)

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Also Published As

Publication number Publication date
CN107474062A (zh) 2017-12-15
US20050240047A1 (en) 2005-10-27
IL219856A0 (en) 2012-06-28
CR8653A (es) 2007-10-23
CY1112053T1 (el) 2015-11-04
CL2010000350A1 (es) 2011-01-28
WO2005097809A3 (en) 2006-02-16
NZ586824A (en) 2012-03-30
US20190330270A1 (en) 2019-10-31
JP2010241816A (ja) 2010-10-28
DK4008721T3 (da) 2024-03-25
TWI386212B (zh) 2013-02-21
NZ550522A (en) 2010-08-27
US20200369722A1 (en) 2020-11-26
SG10201800972PA (en) 2018-03-28
NO20171939A1 (no) 2006-12-22
NL1033190A1 (nl) 2007-04-23
CA2738706A1 (en) 2005-10-20
MY145427A (en) 2012-02-15
DK3385267T3 (da) 2021-11-01
ME01975B (me) 2015-05-20
TW200616646A (en) 2006-06-01
JP5414625B2 (ja) 2014-02-12
CL2014002252A1 (es) 2014-12-05
JP4558039B2 (ja) 2010-10-06
DOP2011000293A (es) 2011-12-15
EP3385267B1 (en) 2021-09-29
SG151322A1 (en) 2009-04-30
US20160362449A1 (en) 2016-12-15
CA2853272A1 (en) 2005-10-20
CN103396427A (zh) 2013-11-20
ECSP066960A (es) 2006-12-20
CN111925385B (zh) 2023-11-21
EP2377869A1 (en) 2011-10-19
AU2005230930A1 (en) 2005-10-20
CA2560886A1 (en) 2005-10-20
NO344610B1 (no) 2020-02-10
HK1246300A1 (zh) 2018-09-07
LT4008721T (lt) 2024-03-25
EA012927B1 (ru) 2010-02-26
IL219853A (en) 2015-05-31
UY28830A1 (es) 2005-09-30
RS53259B (en) 2014-08-29
SI2377869T1 (sl) 2014-05-30
EA200601795A1 (ru) 2007-04-27
HRP20140339T1 (hr) 2014-05-09
CN111925385A (zh) 2020-11-13
PE20110075A1 (es) 2011-02-17
IL178250A0 (en) 2006-12-31
US20100174072A1 (en) 2010-07-08
UA90108C2 (uk) 2010-04-12
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IL178250A (en) 2012-06-28
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