RS62738B1 - Sinteza jedinjenja estra organoborne kiseline i organoborne kiseline - Google Patents

Sinteza jedinjenja estra organoborne kiseline i organoborne kiseline

Info

Publication number
RS62738B1
RS62738B1 RS20211565A RSP20211565A RS62738B1 RS 62738 B1 RS62738 B1 RS 62738B1 RS 20211565 A RS20211565 A RS 20211565A RS P20211565 A RSP20211565 A RS P20211565A RS 62738 B1 RS62738 B1 RS 62738B1
Authority
RS
Serbia
Prior art keywords
synthesis
acid compounds
boronic ester
boronic
ester
Prior art date
Application number
RS20211565A
Other languages
English (en)
Inventor
Fraser I Pickersgill
John Bishop
Young Lo
Fang-Ting Chui
Vithalanand R Kulkarni
Original Assignee
Millennium Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34968044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RS62738(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Millennium Pharm Inc filed Critical Millennium Pharm Inc
Publication of RS62738B1 publication Critical patent/RS62738B1/sr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/04—Esters of boric acids
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Transplantation (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
RS20211565A 2004-03-30 2005-03-24 Sinteza jedinjenja estra organoborne kiseline i organoborne kiseline RS62738B1 (sr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55753504P 2004-03-30 2004-03-30
EP18172486.5A EP3385267B1 (en) 2004-03-30 2005-03-24 Synthesis of boronic ester and acid compounds

Publications (1)

Publication Number Publication Date
RS62738B1 true RS62738B1 (sr) 2022-01-31

Family

ID=34968044

Family Applications (4)

Application Number Title Priority Date Filing Date
RS20110502A RS51983B (sr) 2004-03-30 2005-03-24 Sinteza jedinjenja estra organoborne kiseline i organoborne kiseline
RS20240260A RS65253B1 (sr) 2004-03-30 2005-03-24 Sinteza jedinjenja estra organoborne kiseline i organoborne kiseline
RS20211565A RS62738B1 (sr) 2004-03-30 2005-03-24 Sinteza jedinjenja estra organoborne kiseline i organoborne kiseline
RS20140186A RS53259B (sr) 2004-03-30 2005-03-24 Sinteza bortezomiba

Family Applications Before (2)

Application Number Title Priority Date Filing Date
RS20110502A RS51983B (sr) 2004-03-30 2005-03-24 Sinteza jedinjenja estra organoborne kiseline i organoborne kiseline
RS20240260A RS65253B1 (sr) 2004-03-30 2005-03-24 Sinteza jedinjenja estra organoborne kiseline i organoborne kiseline

Family Applications After (1)

Application Number Title Priority Date Filing Date
RS20140186A RS53259B (sr) 2004-03-30 2005-03-24 Sinteza bortezomiba

Country Status (41)

Country Link
US (14) US7714159B2 (sr)
EP (5) EP1756121B1 (sr)
JP (4) JP4558039B2 (sr)
KR (1) KR100939598B1 (sr)
CN (5) CN1960996B (sr)
AR (3) AR049374A1 (sr)
AT (1) ATE521612T1 (sr)
AU (1) AU2005230930B2 (sr)
BR (1) BRPI0509587A (sr)
CA (4) CA2738706C (sr)
CL (2) CL2010000350A1 (sr)
CR (1) CR8653A (sr)
CY (3) CY1112053T1 (sr)
DK (4) DK3385267T3 (sr)
DO (1) DOP2011000293A (sr)
EA (1) EA012927B1 (sr)
EC (1) ECSP066960A (sr)
ES (3) ES2899606T3 (sr)
FI (1) FI4008721T3 (sr)
HK (4) HK1100004A1 (sr)
HR (4) HRP20212002T1 (sr)
HU (1) HUE056859T2 (sr)
IL (3) IL178250A (sr)
LT (2) LT3385267T (sr)
ME (1) ME01975B (sr)
MX (1) MX367324B (sr)
MY (1) MY145427A (sr)
NL (3) NL1028639C2 (sr)
NO (4) NO338905B1 (sr)
NZ (3) NZ586824A (sr)
PE (3) PE20142402A1 (sr)
PL (4) PL2377869T3 (sr)
PT (4) PT1756121E (sr)
RS (4) RS51983B (sr)
SG (5) SG10201800972PA (sr)
SI (4) SI1756121T1 (sr)
TW (1) TWI386212B (sr)
UA (1) UA90108C2 (sr)
UY (3) UY28830A1 (sr)
WO (1) WO2005097809A2 (sr)
ZA (1) ZA200608689B (sr)

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EA034601B1 (ru) * 2007-08-06 2020-02-25 Милленниум Фармасьютикалз, Инк. Способ получения бороновых кислот
EP2527347A1 (en) * 2007-08-06 2012-11-28 Millennium Pharmaceuticals, Inc. Proteasome inhibitors
US7442830B1 (en) 2007-08-06 2008-10-28 Millenium Pharmaceuticals, Inc. Proteasome inhibitors
AU2016253697A1 (en) * 2007-08-06 2016-11-24 Millennium Pharmaceuticals, Inc. Proteasome inhibitors
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US7838673B2 (en) 2007-10-16 2010-11-23 Millennium Pharmaceuticals, Inc. Proteasome inhibitors
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AU2013204881A1 (en) * 2008-09-29 2013-05-16 Millennium Pharmaceuticals, Inc. Derivatives of 1-amino-2-cyclobutylethylboronic acid
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CN102803271B (zh) * 2009-06-19 2016-03-23 力奇制药公司 氢化卤代烯烃而不脱卤的方法
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Also Published As

Publication number Publication date
US9862745B2 (en) 2018-01-09
NO338905B1 (no) 2016-10-31
SI4008721T1 (sl) 2024-05-31
DK1756121T3 (da) 2012-01-09
ATE521612T1 (de) 2011-09-15
HUE056859T2 (hu) 2022-03-28
HK1164320A1 (en) 2012-10-19
SI2377869T1 (sl) 2014-05-30
US20050240047A1 (en) 2005-10-27
HRP20212002T1 (hr) 2022-04-01
UY28830A1 (es) 2005-09-30
SG10201600029PA (en) 2016-02-26
WO2005097809A3 (en) 2006-02-16
EP4008721A1 (en) 2022-06-08
RS53259B (sr) 2014-08-29
JP2007530687A (ja) 2007-11-01
EP3385267A1 (en) 2018-10-10
US20150038706A1 (en) 2015-02-05
PT4008721T (pt) 2024-03-21
PT1756121E (pt) 2011-11-30
AR097309A2 (es) 2016-03-02
IL219853A (en) 2015-05-31
DOP2011000293A (es) 2011-12-15
JP2010241816A (ja) 2010-10-28
JP2013100378A (ja) 2013-05-23
NL1028639A1 (nl) 2005-10-20
HRP20140339T1 (hr) 2014-05-09
AU2005230930B2 (en) 2011-09-29
US20210171574A1 (en) 2021-06-10
EP3385267B1 (en) 2021-09-29
US8283467B2 (en) 2012-10-09
SG10201800972PA (en) 2018-03-28
ME01975B (me) 2015-05-20
NO343966B1 (no) 2019-07-29
JP5414625B2 (ja) 2014-02-12
ZA200608689B (en) 2007-09-26
EP2377868A1 (en) 2011-10-19
US7714159B2 (en) 2010-05-11
NO20171939A1 (no) 2006-12-22
JP6193960B2 (ja) 2017-09-06
JP2016056180A (ja) 2016-04-21
MY145427A (en) 2012-02-15
TWI386212B (zh) 2013-02-21
NZ586824A (en) 2012-03-30
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