KR830001901B1 - 페니실린과 세팔로스포린 이미노할라이드의 제조방법 - Google Patents

페니실린과 세팔로스포린 이미노할라이드의 제조방법 Download PDF

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Publication number
KR830001901B1
KR830001901B1 KR1019800000403A KR800000403A KR830001901B1 KR 830001901 B1 KR830001901 B1 KR 830001901B1 KR 1019800000403 A KR1019800000403 A KR 1019800000403A KR 800000403 A KR800000403 A KR 800000403A KR 830001901 B1 KR830001901 B1 KR 830001901B1
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KR
South Korea
Prior art keywords
mmol
added
solution
reaction mixture
chlorine
Prior art date
Application number
KR1019800000403A
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English (en)
Korean (ko)
Other versions
KR830001943A (ko
Inventor
델로스 하트필드 로우웰
크리스 브라스즈크작 라리
웨인 피셔 잭
Original Assignee
일라이 릴리 앤드 캄파니
아더 알·웨일
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27358615&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR830001901(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US06/008,645 external-priority patent/US4223133A/en
Priority claimed from US06/008,647 external-priority patent/US4226986A/en
Priority claimed from US06/008,470 external-priority patent/US4211702A/en
Application filed by 일라이 릴리 앤드 캄파니, 아더 알·웨일 filed Critical 일라이 릴리 앤드 캄파니
Publication of KR830001943A publication Critical patent/KR830001943A/ko
Application granted granted Critical
Publication of KR830001901B1 publication Critical patent/KR830001901B1/ko

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04Preparation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02Preparation
    • C07D501/04Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D505/00Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
KR1019800000403A 1979-02-01 1980-02-01 페니실린과 세팔로스포린 이미노할라이드의 제조방법 KR830001901B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US06/008,645 US4223133A (en) 1979-02-01 1979-02-01 Cephalosporin reduction process
US8470 1979-02-01
US06/008,647 US4226986A (en) 1979-02-01 1979-02-01 Process for halogenation of β-lactam compounds
US06/008,470 US4211702A (en) 1979-02-01 1979-02-01 Process for preparation of penicillin and cephalosporin imino halides

Publications (2)

Publication Number Publication Date
KR830001943A KR830001943A (ko) 1983-05-19
KR830001901B1 true KR830001901B1 (ko) 1983-09-19

Family

ID=27358615

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019800000403A KR830001901B1 (ko) 1979-02-01 1980-02-01 페니실린과 세팔로스포린 이미노할라이드의 제조방법

Country Status (32)

Country Link
EP (1) EP0014567B1 (US20030199744A1-20031023-C00003.png)
JP (12) JPS55113789A (US20030199744A1-20031023-C00003.png)
KR (1) KR830001901B1 (US20030199744A1-20031023-C00003.png)
AT (1) AT372684B (US20030199744A1-20031023-C00003.png)
AU (1) AU538175B2 (US20030199744A1-20031023-C00003.png)
BE (1) BE881425A (US20030199744A1-20031023-C00003.png)
BG (1) BG35899A3 (US20030199744A1-20031023-C00003.png)
CA (1) CA1133468A (US20030199744A1-20031023-C00003.png)
CH (3) CH656385A5 (US20030199744A1-20031023-C00003.png)
DD (1) DD153374A5 (US20030199744A1-20031023-C00003.png)
DE (1) DE3066119D1 (US20030199744A1-20031023-C00003.png)
DK (2) DK163513C (US20030199744A1-20031023-C00003.png)
ES (1) ES488231A0 (US20030199744A1-20031023-C00003.png)
FI (1) FI74968C (US20030199744A1-20031023-C00003.png)
FR (1) FR2447924A1 (US20030199744A1-20031023-C00003.png)
GB (1) GB2044256B (US20030199744A1-20031023-C00003.png)
GR (1) GR72278B (US20030199744A1-20031023-C00003.png)
IE (1) IE49377B1 (US20030199744A1-20031023-C00003.png)
IL (1) IL59269A (US20030199744A1-20031023-C00003.png)
IT (1) IT1193908B (US20030199744A1-20031023-C00003.png)
LU (1) LU82120A1 (US20030199744A1-20031023-C00003.png)
MA (1) MA18715A1 (US20030199744A1-20031023-C00003.png)
MW (1) MW880A1 (US20030199744A1-20031023-C00003.png)
MY (1) MY8500598A (US20030199744A1-20031023-C00003.png)
NL (1) NL191791C (US20030199744A1-20031023-C00003.png)
NO (1) NO160660C (US20030199744A1-20031023-C00003.png)
NZ (1) NZ192749A (US20030199744A1-20031023-C00003.png)
OA (1) OA06451A (US20030199744A1-20031023-C00003.png)
PH (1) PH15158A (US20030199744A1-20031023-C00003.png)
PL (4) PL129604B1 (US20030199744A1-20031023-C00003.png)
PT (1) PT70744A (US20030199744A1-20031023-C00003.png)
YU (4) YU22580A (US20030199744A1-20031023-C00003.png)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2063129T3 (es) * 1988-06-22 1995-01-01 Lilly Co Eli Intermedio de la 1-carba(detia)cefalosporina.
EP1961636B1 (en) 2007-02-20 2013-04-24 Yamaha Hatsudoki Kabushiki Kaisha Hydraulic master cylinder and vehicle provided with the same
KR101466783B1 (ko) 2012-03-09 2014-11-28 신이치로 다니 트레이닝 래더
WO2014056567A1 (de) * 2012-10-11 2014-04-17 Merck Patent Gmbh Materialien für organische elektrolumineszenzvorrichtungen
JP6202969B2 (ja) * 2013-10-01 2017-09-27 富士電機株式会社 情報処理装置、暗号化方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK118506B (da) * 1963-02-18 1970-08-31 Ciba Geigy Fremgangsmåde til fremstilling af 7-aminocephalosporansyre eller estere deraf.
US3641014A (en) * 1968-10-03 1972-02-08 Lilly Co Eli Reduction of delta**3-cephalosporin sulfoxides
US3925372A (en) * 1973-02-23 1975-12-09 Lilly Co Eli Alpha-aminoacyl-3-halo cephalosporins

Also Published As

Publication number Publication date
OA06451A (fr) 1981-07-31
JPH04364187A (ja) 1992-12-16
NO160660C (no) 1989-05-16
JPH0649705B2 (ja) 1994-06-29
NL8000545A (nl) 1980-08-05
BG35899A3 (en) 1984-07-16
DD153374A5 (de) 1982-01-06
JPH089629B2 (ja) 1996-01-31
MW880A1 (en) 1981-09-09
YU18283A (en) 1984-02-29
EP0014567B1 (en) 1984-01-18
CH648318A5 (fr) 1985-03-15
JPH0334984A (ja) 1991-02-14
FI74968B (fi) 1987-12-31
IE800190L (en) 1980-08-01
NL191791C (nl) 1996-08-02
JPH0334983A (ja) 1991-02-14
JPH0372631B2 (US20030199744A1-20031023-C00003.png) 1991-11-19
MY8500598A (en) 1985-12-31
AU538175B2 (en) 1984-08-02
GB2044256B (en) 1983-05-05
NO160660B (no) 1989-02-06
BE881425A (fr) 1980-07-30
IT1193908B (it) 1988-08-31
DK163513B (da) 1992-03-09
DK41480A (da) 1980-08-02
ES8101603A1 (es) 1980-12-16
PT70744A (en) 1980-02-01
IE49377B1 (en) 1985-10-02
JPH0372633B2 (US20030199744A1-20031023-C00003.png) 1991-11-19
PL128595B1 (en) 1984-02-29
DK163513C (da) 1992-07-27
YU44734B (en) 1991-02-28
CH652405A5 (fr) 1985-11-15
IL59269A0 (en) 1980-05-30
JPH0565514B2 (US20030199744A1-20031023-C00003.png) 1993-09-17
JPH0372634B2 (US20030199744A1-20031023-C00003.png) 1991-11-19
JPH0334982A (ja) 1991-02-14
FR2447924A1 (fr) 1980-08-29
DK163667B (da) 1992-03-23
MA18715A1 (fr) 1980-10-01
PH15158A (en) 1982-08-24
JPH0532669A (ja) 1993-02-09
YU16483A (en) 1984-02-29
JPH0372632B2 (US20030199744A1-20031023-C00003.png) 1991-11-19
CA1133468A (en) 1982-10-12
DK163667C (da) 1992-08-17
AT372684B (de) 1983-11-10
DK179991A (da) 1991-10-30
JPH0649706B2 (ja) 1994-06-29
NL191791B (nl) 1996-04-01
CH656385A5 (fr) 1986-06-30
JPH0372231B2 (US20030199744A1-20031023-C00003.png) 1991-11-18
YU22580A (en) 1983-06-30
PL221744A1 (US20030199744A1-20031023-C00003.png) 1980-12-01
ES488231A0 (es) 1980-12-16
FI74968C (fi) 1988-04-11
LU82120A1 (fr) 1980-04-23
PL126947B1 (en) 1983-09-30
JPH0334985A (ja) 1991-02-14
JPH04356490A (ja) 1992-12-10
AU5502980A (en) 1980-08-07
JPH0517483A (ja) 1993-01-26
GB2044256A (en) 1980-10-15
NO800251L (no) 1980-08-04
DE3066119D1 (en) 1984-02-23
GR72278B (US20030199744A1-20031023-C00003.png) 1983-10-11
IL59269A (en) 1984-04-30
JPH0371435B2 (US20030199744A1-20031023-C00003.png) 1991-11-13
FI800303A (fi) 1980-08-02
IT8019609A0 (it) 1980-01-31
JPH054990A (ja) 1993-01-14
NZ192749A (en) 1983-06-17
PL129604B1 (en) 1984-05-31
KR830001943A (ko) 1983-05-19
FR2447924B1 (US20030199744A1-20031023-C00003.png) 1983-10-21
PL129399B1 (en) 1984-05-31
JPH0565513B2 (US20030199744A1-20031023-C00003.png) 1993-09-17
JPH0334981A (ja) 1991-02-14
JPH054991A (ja) 1993-01-14
JPH07121950B2 (ja) 1995-12-25
YU16383A (en) 1984-02-29
ATA50280A (de) 1983-03-15
DK179991D0 (da) 1991-10-30
EP0014567A1 (en) 1980-08-20
JPS55113789A (en) 1980-09-02

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