JP5951600B2 - キナーゼ調節のための、化合物、組成物および方法 - Google Patents
キナーゼ調節のための、化合物、組成物および方法 Download PDFInfo
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- JP5951600B2 JP5951600B2 JP2013511397A JP2013511397A JP5951600B2 JP 5951600 B2 JP5951600 B2 JP 5951600B2 JP 2013511397 A JP2013511397 A JP 2013511397A JP 2013511397 A JP2013511397 A JP 2013511397A JP 5951600 B2 JP5951600 B2 JP 5951600B2
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/16—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
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| US34737010P | 2010-05-21 | 2010-05-21 | |
| US61/347,370 | 2010-05-21 | ||
| PCT/US2011/037412 WO2011146882A1 (en) | 2010-05-21 | 2011-05-20 | Chemical compounds, compositions and methods for kinase modulation |
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| JP (2) | JP5951600B2 (https=) |
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| CA (1) | CA2799579A1 (https=) |
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| JP2016172744A (ja) * | 2010-05-21 | 2016-09-29 | インフィニティー ファーマシューティカルズ， インコーポレイテッド | キナーゼ調節のための、化合物、組成物および方法 |
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- 2011-05-20 WO PCT/US2011/037412 patent/WO2011146882A1/en not_active Ceased
- 2011-05-20 AU AU2011255218A patent/AU2011255218B2/en not_active Ceased
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2016172744A (ja) * | 2010-05-21 | 2016-09-29 | インフィニティー ファーマシューティカルズ， インコーポレイテッド | キナーゼ調節のための、化合物、組成物および方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| CN103002738A (zh) | 2013-03-27 |
| JP2013526586A (ja) | 2013-06-24 |
| EP2571357B1 (en) | 2016-07-06 |
| US9738644B2 (en) | 2017-08-22 |
| US20120059000A1 (en) | 2012-03-08 |
| CA2799579A1 (en) | 2011-11-24 |
| EP2571357A4 (en) | 2013-11-20 |
| ES2593256T3 (es) | 2016-12-07 |
| JP2016172744A (ja) | 2016-09-29 |
| AU2011255218B2 (en) | 2015-03-12 |
| US9181221B2 (en) | 2015-11-10 |
| EP2571357A1 (en) | 2013-03-27 |
| US20160016957A1 (en) | 2016-01-21 |
| US8604032B2 (en) | 2013-12-10 |
| WO2011146882A1 (en) | 2011-11-24 |
| US20140088099A1 (en) | 2014-03-27 |
| AU2011255218A1 (en) | 2012-12-20 |
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