JP5567252B2 - グリコピロレートおよびベータ２アドレナリン受容体アゴニストの組合せ剤 - Google Patents

グリコピロレートおよびベータ２アドレナリン受容体アゴニストの組合せ剤 Download PDF

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JP5567252B2
JP5567252B2 JP2007517074A JP2007517074A JP5567252B2 JP 5567252 B2 JP5567252 B2 JP 5567252B2 JP 2007517074 A JP2007517074 A JP 2007517074A JP 2007517074 A JP2007517074 A JP 2007517074A JP 5567252 B2 JP5567252 B2 JP 5567252B2
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alkyl
hydroxy
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substituted
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JP2007538036A (ja
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スティーブン・ポール・コリングウッド
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ノバルティス アーゲー
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4704—2-Quinolinones, e.g. carbostyril
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/402—1-aryl substituted, e.g. piretanide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Compositions Of Oxide Ceramics (AREA)
JP2007517074A 2004-05-18 2005-05-17 グリコピロレートおよびベータ２アドレナリン受容体アゴニストの組合せ剤 Expired - Lifetime JP5567252B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0411056.5 2004-05-18
GBGB0411056.5A GB0411056D0 (en) 2004-05-18 2004-05-18 Organic compounds
PCT/EP2005/005354 WO2005110402A1 (en) 2004-05-18 2005-05-17 Combinations of glycopyrrolate and beta2 adrenoceptor agonists

Related Child Applications (1)

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JP2012156212A Division JP2012236833A (ja) 2004-05-18 2012-07-12 グリコピロレートおよびベータ２アドレナリン受容体アゴニストの組合せ剤

Publications (2)

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JP2007538036A JP2007538036A (ja) 2007-12-27
JP5567252B2 true JP5567252B2 (ja) 2014-08-06

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JP2007517074A Expired - Lifetime JP5567252B2 (ja) 2004-05-18 2005-05-17 グリコピロレートおよびベータ２アドレナリン受容体アゴニストの組合せ剤
JP2012156212A Pending JP2012236833A (ja) 2004-05-18 2012-07-12 グリコピロレートおよびベータ２アドレナリン受容体アゴニストの組合せ剤

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US (6) US20080267886A1 (cg-RX-API-DMAC7.html)
EP (3) EP2228064B1 (cg-RX-API-DMAC7.html)
JP (2) JP5567252B2 (cg-RX-API-DMAC7.html)
KR (2) KR101360556B1 (cg-RX-API-DMAC7.html)
CN (1) CN1953745A (cg-RX-API-DMAC7.html)
AT (1) ATE521348T1 (cg-RX-API-DMAC7.html)
AU (1) AU2005244439C1 (cg-RX-API-DMAC7.html)
BE (1) BE2020C517I2 (cg-RX-API-DMAC7.html)
BR (1) BRPI0511327B8 (cg-RX-API-DMAC7.html)
CA (1) CA2563302C (cg-RX-API-DMAC7.html)
CY (4) CY1112086T1 (cg-RX-API-DMAC7.html)
DK (2) DK2228064T3 (cg-RX-API-DMAC7.html)
EC (1) ECSP066950A (cg-RX-API-DMAC7.html)
ES (2) ES2370647T3 (cg-RX-API-DMAC7.html)
FR (1) FR20C1018I2 (cg-RX-API-DMAC7.html)
GB (1) GB0411056D0 (cg-RX-API-DMAC7.html)
HU (3) HUE048936T2 (cg-RX-API-DMAC7.html)
IL (1) IL179013A (cg-RX-API-DMAC7.html)
LT (3) LT2228064T (cg-RX-API-DMAC7.html)
LU (1) LUC00155I2 (cg-RX-API-DMAC7.html)
MA (1) MA28598B1 (cg-RX-API-DMAC7.html)
MX (1) MXPA06013382A (cg-RX-API-DMAC7.html)
NO (2) NO334760B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ550369A (cg-RX-API-DMAC7.html)
PL (2) PL1755590T3 (cg-RX-API-DMAC7.html)
PT (2) PT1755590E (cg-RX-API-DMAC7.html)
RU (1) RU2388465C2 (cg-RX-API-DMAC7.html)
SE (1) SE1755590T5 (cg-RX-API-DMAC7.html)
SG (1) SG153836A1 (cg-RX-API-DMAC7.html)
SI (2) SI2228064T1 (cg-RX-API-DMAC7.html)
TN (1) TNSN06377A1 (cg-RX-API-DMAC7.html)
WO (1) WO2005110402A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA200608123B (cg-RX-API-DMAC7.html)

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