JP3194974B2 - 標的制御釈放薬剤 - Google Patents
標的制御釈放薬剤Info
- Publication number
- JP3194974B2 JP3194974B2 JP02778491A JP2778491A JP3194974B2 JP 3194974 B2 JP3194974 B2 JP 3194974B2 JP 02778491 A JP02778491 A JP 02778491A JP 2778491 A JP2778491 A JP 2778491A JP 3194974 B2 JP3194974 B2 JP 3194974B2
- Authority
- JP
- Japan
- Prior art keywords
- membrane
- active ingredient
- cellulose
- colon
- drug according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT02005490A IT1246382B (it) | 1990-04-17 | 1990-04-17 | Metodo per la cessione mirata e controllata di farmaci nell'intestino e particolarmente nel colon |
| IT20054A/90 | 1990-04-17 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPH04224517A JPH04224517A (ja) | 1992-08-13 |
| JP3194974B2 true JP3194974B2 (ja) | 2001-08-06 |
Family
ID=11163447
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP02778491A Expired - Lifetime JP3194974B2 (ja) | 1990-04-17 | 1991-01-30 | 標的制御釈放薬剤 |
| JP91506876A Pending JPH05506217A (ja) | 1990-04-17 | 1991-04-09 | 制御放出薬剤処方 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP91506876A Pending JPH05506217A (ja) | 1990-04-17 | 1991-04-09 | 制御放出薬剤処方 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US5900252A (enExample) |
| EP (2) | EP0453001A1 (enExample) |
| JP (2) | JP3194974B2 (enExample) |
| KR (1) | KR100196256B1 (enExample) |
| AT (1) | ATE144138T1 (enExample) |
| AU (1) | AU654277B2 (enExample) |
| CA (2) | CA2035155A1 (enExample) |
| DE (1) | DE69122751T2 (enExample) |
| DK (1) | DK0524989T3 (enExample) |
| ES (1) | ES2093097T3 (enExample) |
| GR (1) | GR3021847T3 (enExample) |
| IE (1) | IE911271A1 (enExample) |
| IT (1) | IT1246382B (enExample) |
| NZ (1) | NZ237823A (enExample) |
| PT (1) | PT97370B (enExample) |
| RU (1) | RU2111743C1 (enExample) |
| SG (1) | SG46584A1 (enExample) |
| TW (1) | TW223022B (enExample) |
| WO (1) | WO1991016042A1 (enExample) |
| ZA (1) | ZA912792B (enExample) |
Families Citing this family (422)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6764697B1 (en) | 1991-06-27 | 2004-07-20 | Alza Corporation | System for delaying drug delivery up to seven hours |
| US5160742A (en) * | 1991-12-31 | 1992-11-03 | Abbott Laboratories | System for delivering an active substance for sustained release |
| IT1260505B (it) * | 1992-06-01 | 1996-04-09 | Poli Ind Chimica Spa | Sistemi farmaceutici orali a cessione ritardata per il rilascio specifico nel colon |
| WO1995016451A1 (fr) * | 1992-06-22 | 1995-06-22 | Franck Arno Gouchet | Comprimes a liberation controlee de 4-asa |
| FR2692484B1 (fr) * | 1992-06-22 | 1995-06-30 | Gouchet Franck | Nouvelle forme galenique de 4-asa a liberation controlee. |
| ES2173096T3 (es) * | 1992-08-05 | 2002-10-16 | Faulding F H & Co Ltd | Composicion farmaceutica peletizada. |
| AU670958B2 (en) * | 1992-08-05 | 1996-08-08 | Mayne Pharma International Pty Ltd | Pelletised pharmaceutical composition |
| US5358502A (en) | 1993-02-25 | 1994-10-25 | Pfizer Inc | PH-triggered osmotic bursting delivery devices |
| US5914132A (en) * | 1993-02-26 | 1999-06-22 | The Procter & Gamble Company | Pharmaceutical dosage form with multiple enteric polymer coatings for colonic delivery |
| IT1265092B1 (it) * | 1993-05-31 | 1996-10-30 | Giuliani Spa | Preparato per uso come integratore alimentare, o dietetico,a rilascio mirato nel colon |
| DE4332394A1 (de) * | 1993-09-23 | 1995-03-30 | Falk Pharma Gmbh | Budesonid-Pellets mit kontrolliertem Freigabeprofil und Verfahren zu ihrer Herstellung |
| US5523095A (en) * | 1993-12-15 | 1996-06-04 | Eastman Chemical Company | Controlled release matrix system using cellulose acetate/polyvinylpyrrolidone blends |
| US5536505A (en) * | 1993-12-15 | 1996-07-16 | Eastman Chemical Company | Controlled release matrix system using cellulose acetate/poly-2-ethyl-2-oxazoline blends |
| KR100388569B1 (ko) | 1994-04-22 | 2003-10-11 | 야마노우치세이야쿠 가부시키가이샤 | 결장특이적약물방출용경구약제학적제제 |
| AT403988B (de) * | 1994-05-18 | 1998-07-27 | Lannacher Heilmittel | Festes orales retardpräparat |
| US5686106A (en) * | 1995-05-17 | 1997-11-11 | The Procter & Gamble Company | Pharmaceutical dosage form for colonic delivery |
| KR100542544B1 (ko) * | 1995-12-21 | 2006-05-10 | 파마슈티스크 라보라토리움 페링 에이/에스 | 5-아미노살리실산을함유하는방출제어형경구용약제학적조성물및장질환을치료하는방법 |
| US5840332A (en) * | 1996-01-18 | 1998-11-24 | Perio Products Ltd. | Gastrointestinal drug delivery system |
| US6245351B1 (en) | 1996-03-07 | 2001-06-12 | Takeda Chemical Industries, Ltd. | Controlled-release composition |
| US8071128B2 (en) | 1996-06-14 | 2011-12-06 | Kyowa Hakko Kirin Co., Ltd. | Intrabuccally rapidly disintegrating tablet and a production method of the tablets |
| AUPO247496A0 (en) | 1996-09-23 | 1996-10-17 | Resmed Limited | Assisted ventilation to match patient respiratory need |
| AU5775398A (en) * | 1996-12-17 | 1998-07-15 | Poli Industria Chimica S.P.A. | Site-specific controlled release dosage formulation for mesalamine |
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| DE60005819T2 (de) | 1999-06-14 | 2004-05-06 | Cosmo S.P.A. | Geschmacksmaskierte orale pharmazeutische zusammensetzungen mit kontrollierter abgabe |
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| US3473490A (en) * | 1966-01-17 | 1969-10-21 | Camillo Corvi Mora | Producing chronoactive pharmaceutical granules |
| GB1468172A (en) * | 1973-03-28 | 1977-03-23 | Benzon As Alfred | Oral drug preparations |
| FR2471186A1 (fr) * | 1979-12-10 | 1981-06-19 | Roussel Uclaf | Nouveaux comprimes a delitescence colique, ainsi que leur procede de preparation |
| JPS57171428A (en) * | 1981-04-13 | 1982-10-22 | Sankyo Co Ltd | Preparation of coated solid preparation |
| DK58983D0 (da) * | 1983-02-11 | 1983-02-11 | Leo Pharm Prod Ltd | Farmaceutisk praeparat |
| US4503030A (en) * | 1983-06-06 | 1985-03-05 | Alza Corporation | Device for delivering drug to certain pH environments |
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-
1990
- 1990-04-17 IT IT02005490A patent/IT1246382B/it active IP Right Grant
-
1991
- 1991-01-29 CA CA002035155A patent/CA2035155A1/en not_active Abandoned
- 1991-01-29 EP EP91200173A patent/EP0453001A1/en not_active Withdrawn
- 1991-01-30 JP JP02778491A patent/JP3194974B2/ja not_active Expired - Lifetime
- 1991-04-09 JP JP91506876A patent/JPH05506217A/ja active Pending
- 1991-04-09 DE DE69122751T patent/DE69122751T2/de not_active Expired - Fee Related
- 1991-04-09 AT AT91907396T patent/ATE144138T1/de not_active IP Right Cessation
- 1991-04-09 RU RU92016377A patent/RU2111743C1/ru active
- 1991-04-09 WO PCT/EP1991/000688 patent/WO1991016042A1/en not_active Ceased
- 1991-04-09 EP EP91907396A patent/EP0524989B1/en not_active Expired - Lifetime
- 1991-04-09 DK DK91907396.5T patent/DK0524989T3/da active
- 1991-04-09 SG SG1996006208A patent/SG46584A1/en unknown
- 1991-04-09 ES ES91907396T patent/ES2093097T3/es not_active Expired - Lifetime
- 1991-04-09 AU AU76798/91A patent/AU654277B2/en not_active Ceased
- 1991-04-09 KR KR1019920702558A patent/KR100196256B1/ko not_active Expired - Fee Related
- 1991-04-15 NZ NZ237823A patent/NZ237823A/en unknown
- 1991-04-15 ZA ZA912792A patent/ZA912792B/xx unknown
- 1991-04-15 PT PT97370A patent/PT97370B/pt not_active IP Right Cessation
- 1991-04-15 CA CA002040471A patent/CA2040471A1/en not_active Abandoned
- 1991-04-16 IE IE127191A patent/IE911271A1/en unknown
- 1991-04-16 TW TW080102920A patent/TW223022B/zh active
-
1992
- 1992-11-06 US US07/972,660 patent/US5900252A/en not_active Expired - Fee Related
-
1996
- 1996-11-29 GR GR960403247T patent/GR3021847T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2111743C1 (ru) | 1998-05-27 |
| IE911271A1 (en) | 1991-10-23 |
| NZ237823A (en) | 1992-09-25 |
| IT9020054A0 (it) | 1990-04-17 |
| WO1991016042A1 (en) | 1991-10-31 |
| ATE144138T1 (de) | 1996-11-15 |
| GR3021847T3 (en) | 1997-02-28 |
| TW223022B (enExample) | 1994-05-01 |
| ES2093097T3 (es) | 1996-12-16 |
| CA2035155A1 (en) | 1991-10-18 |
| SG46584A1 (en) | 1998-02-20 |
| AU7679891A (en) | 1991-11-11 |
| DE69122751D1 (de) | 1996-11-21 |
| KR100196256B1 (ko) | 1999-06-15 |
| JPH04224517A (ja) | 1992-08-13 |
| PT97370A (pt) | 1992-01-31 |
| EP0453001A1 (en) | 1991-10-23 |
| IT9020054A1 (enExample) | 1991-10-17 |
| CA2040471A1 (en) | 1991-10-18 |
| KR930700077A (ko) | 1993-03-13 |
| JPH05506217A (ja) | 1993-09-16 |
| US5900252A (en) | 1999-05-04 |
| EP0524989A1 (en) | 1993-02-03 |
| DK0524989T3 (da) | 1996-11-18 |
| PT97370B (pt) | 1998-08-31 |
| IT1246382B (it) | 1994-11-18 |
| DE69122751T2 (de) | 1997-02-13 |
| ZA912792B (en) | 1992-12-30 |
| EP0524989B1 (en) | 1996-10-16 |
| AU654277B2 (en) | 1994-11-03 |
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