CA2035155A1 - Pharmaceutical composition for the targeted controlled release of an active principle within the intestine, and particularly within the colon - Google Patents

Pharmaceutical composition for the targeted controlled release of an active principle within the intestine, and particularly within the colon

Info

Publication number
CA2035155A1
CA2035155A1 CA002035155A CA2035155A CA2035155A1 CA 2035155 A1 CA2035155 A1 CA 2035155A1 CA 002035155 A CA002035155 A CA 002035155A CA 2035155 A CA2035155 A CA 2035155A CA 2035155 A1 CA2035155 A1 CA 2035155A1
Authority
CA
Canada
Prior art keywords
active principle
membrane
composition
covered
colon
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002035155A
Other languages
English (en)
French (fr)
Inventor
Massimo Calanchi
Marco Zema
Gabriele Brunetti
Enzo Giorgetti
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GUILIANE SpA
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2035155A1 publication Critical patent/CA2035155A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CA002035155A 1990-04-17 1991-01-29 Pharmaceutical composition for the targeted controlled release of an active principle within the intestine, and particularly within the colon Abandoned CA2035155A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT02005490A IT1246382B (it) 1990-04-17 1990-04-17 Metodo per la cessione mirata e controllata di farmaci nell'intestino e particolarmente nel colon
IT20054A/90 1990-04-17

Publications (1)

Publication Number Publication Date
CA2035155A1 true CA2035155A1 (en) 1991-10-18

Family

ID=11163447

Family Applications (2)

Application Number Title Priority Date Filing Date
CA002035155A Abandoned CA2035155A1 (en) 1990-04-17 1991-01-29 Pharmaceutical composition for the targeted controlled release of an active principle within the intestine, and particularly within the colon
CA002040471A Abandoned CA2040471A1 (en) 1990-04-17 1991-04-15 Controlled release drug formulation

Family Applications After (1)

Application Number Title Priority Date Filing Date
CA002040471A Abandoned CA2040471A1 (en) 1990-04-17 1991-04-15 Controlled release drug formulation

Country Status (20)

Country Link
US (1) US5900252A (enExample)
EP (2) EP0453001A1 (enExample)
JP (2) JP3194974B2 (enExample)
KR (1) KR100196256B1 (enExample)
AT (1) ATE144138T1 (enExample)
AU (1) AU654277B2 (enExample)
CA (2) CA2035155A1 (enExample)
DE (1) DE69122751T2 (enExample)
DK (1) DK0524989T3 (enExample)
ES (1) ES2093097T3 (enExample)
GR (1) GR3021847T3 (enExample)
IE (1) IE911271A1 (enExample)
IT (1) IT1246382B (enExample)
NZ (1) NZ237823A (enExample)
PT (1) PT97370B (enExample)
RU (1) RU2111743C1 (enExample)
SG (1) SG46584A1 (enExample)
TW (1) TW223022B (enExample)
WO (1) WO1991016042A1 (enExample)
ZA (1) ZA912792B (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
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US8580302B2 (en) 2000-11-20 2013-11-12 Warner Chilcott Company, Llc Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures
US8709476B2 (en) 2003-11-04 2014-04-29 Supernus Pharmaceuticals, Inc. Compositions of quaternary ammonium compounds containing bioavailability enhancers

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* Cited by examiner, † Cited by third party
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* Cited by examiner, † Cited by third party
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US8580302B2 (en) 2000-11-20 2013-11-12 Warner Chilcott Company, Llc Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures
US9089492B2 (en) 2000-11-20 2015-07-28 Warner Chilcott Company, Llc Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures
US7759359B2 (en) 2003-11-04 2010-07-20 Supernus Pharmaceuticals, Inc. Method of treating bladder dysfunction with once-a-day trospium salt formulation
US7763635B2 (en) 2003-11-04 2010-07-27 Supermus Pharmaceuticals, Inc. Once daily dosage forms of trospium
US7781449B2 (en) 2003-11-04 2010-08-24 Supernus Pharmaceuticals, Inc. Trospium chloride treatment method
US7781448B2 (en) 2003-11-04 2010-08-24 Supernus Pharmaceuticals, Inc. Once daily dosage forms of trospium
US8709476B2 (en) 2003-11-04 2014-04-29 Supernus Pharmaceuticals, Inc. Compositions of quaternary ammonium compounds containing bioavailability enhancers

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CA2040471A1 (en) 1991-10-18
ZA912792B (en) 1992-12-30
AU654277B2 (en) 1994-11-03
US5900252A (en) 1999-05-04
JPH05506217A (ja) 1993-09-16
GR3021847T3 (en) 1997-02-28
IT9020054A0 (it) 1990-04-17
IT1246382B (it) 1994-11-18
AU7679891A (en) 1991-11-11
IT9020054A1 (enExample) 1991-10-17
PT97370A (pt) 1992-01-31
SG46584A1 (en) 1998-02-20
DE69122751D1 (de) 1996-11-21
IE911271A1 (en) 1991-10-23
PT97370B (pt) 1998-08-31
KR930700077A (ko) 1993-03-13
DE69122751T2 (de) 1997-02-13
TW223022B (enExample) 1994-05-01
WO1991016042A1 (en) 1991-10-31
DK0524989T3 (da) 1996-11-18
JPH04224517A (ja) 1992-08-13
ES2093097T3 (es) 1996-12-16
EP0524989A1 (en) 1993-02-03
ATE144138T1 (de) 1996-11-15
KR100196256B1 (ko) 1999-06-15
NZ237823A (en) 1992-09-25
JP3194974B2 (ja) 2001-08-06
EP0524989B1 (en) 1996-10-16
RU2111743C1 (ru) 1998-05-27
EP0453001A1 (en) 1991-10-23

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