HK1021537A1 - 6-O-substituted ketolides having antibacterial activity. - Google Patents

6-O-substituted ketolides having antibacterial activity.

Info

Publication number
HK1021537A1
HK1021537A1 HK00100346A HK00100346A HK1021537A1 HK 1021537 A1 HK1021537 A1 HK 1021537A1 HK 00100346 A HK00100346 A HK 00100346A HK 00100346 A HK00100346 A HK 00100346A HK 1021537 A1 HK1021537 A1 HK 1021537A1
Authority
HK
Hong Kong
Prior art keywords
alkyl
substituted
heteroaryl
aryl
optionally substituted
Prior art date
Application number
HK00100346A
Other languages
English (en)
Inventor
Yat Sur Or
Henkun Ma
Richard F Clark
Daniel T Chu
Jacob J Plattner
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107953&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1021537(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/888,350 external-priority patent/US5866549A/en
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of HK1021537A1 publication Critical patent/HK1021537A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Cephalosporin Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK00100346A 1996-09-04 2000-01-19 6-O-substituted ketolides having antibacterial activity. HK1021537A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US70777696A 1996-09-04 1996-09-04
US08/888,350 US5866549A (en) 1996-09-04 1997-07-03 6-O-substituted ketolides having antibacterial activity
PCT/US1997/015506 WO1998009978A1 (en) 1996-09-04 1997-09-02 6-o-substituted ketolides having antibacterial activity

Publications (1)

Publication Number Publication Date
HK1021537A1 true HK1021537A1 (en) 2000-06-16

Family

ID=27107953

Family Applications (1)

Application Number Title Priority Date Filing Date
HK00100346A HK1021537A1 (en) 1996-09-04 2000-01-19 6-O-substituted ketolides having antibacterial activity.

Country Status (28)

Country Link
US (4) US6075133A (hr)
EP (5) EP1291352B1 (hr)
JP (1) JP4597274B2 (hr)
KR (5) KR100576988B1 (hr)
CN (4) CN100441591C (hr)
AT (5) ATE299508T1 (hr)
BG (1) BG63547B1 (hr)
BR (1) BR9711661A (hr)
CA (1) CA2263972C (hr)
CZ (1) CZ300106B6 (hr)
DE (5) DE69733422T2 (hr)
DK (5) DK1291351T3 (hr)
ES (5) ES2242983T3 (hr)
HK (1) HK1021537A1 (hr)
HR (5) HRP970473B1 (hr)
HU (1) HU230166B1 (hr)
ID (1) ID19406A (hr)
IL (1) IL128681A0 (hr)
NO (1) NO314230B1 (hr)
NZ (1) NZ334274A (hr)
PL (1) PL188173B1 (hr)
PT (5) PT1291351E (hr)
RO (1) RO121473B1 (hr)
RU (1) RU2192427C2 (hr)
SI (1) SI20023B (hr)
SK (5) SK285536B6 (hr)
TR (1) TR199901127T2 (hr)
WO (1) WO1998009978A1 (hr)

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US6495348B1 (en) 1993-10-07 2002-12-17 Regents Of The University Of Minnesota Mitomycin biosynthetic gene cluster
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ATE243219T1 (de) 1998-04-24 2003-07-15 Pfizer Prod Inc 9a, 11b-dehydro derivative von 9-oxime-3-keto-6-0-methylerythromycin
US6265202B1 (en) 1998-06-26 2001-07-24 Regents Of The University Of Minnesota DNA encoding methymycin and pikromycin
JP4573925B2 (ja) * 1998-07-09 2010-11-04 アベンティス・ファーマ・ソシエテ・アノニム 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用
FR2780977B1 (fr) * 1998-07-09 2000-09-01 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
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FR2785612A1 (fr) 1998-11-10 2000-05-12 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
JP4043191B2 (ja) 1998-11-03 2008-02-06 ファイザー・プロダクツ・インク 新規なマクロライド抗生物質
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Also Published As

Publication number Publication date
HRP20060275A2 (hr) 2007-10-31
PL332009A1 (en) 1999-08-16
HUP9902869A2 (hu) 2000-02-28
EP1291351A1 (en) 2003-03-12
ATE296308T1 (de) 2005-06-15
KR20050044815A (ko) 2005-05-12
ID19406A (id) 1998-07-09
PL188173B1 (pl) 2004-12-31
CN1237183A (zh) 1999-12-01
HU230166B1 (hu) 2015-09-28
HRP20060277A2 (hr) 2007-10-31
RO121473B1 (ro) 2007-06-29
US6147197A (en) 2000-11-14
DE69733439D1 (de) 2005-07-07
BG103292A (en) 1999-12-30
HRP20060275B1 (hr) 2014-04-11
PT1291351E (pt) 2005-11-30
WO1998009978A1 (en) 1998-03-12
DE69733439T2 (de) 2006-05-04
DE69733723T2 (de) 2006-04-20
USRE39591E1 (en) 2007-04-24
NZ334274A (en) 2001-02-23
SK285536B6 (sk) 2007-03-01
PT1291350E (pt) 2005-09-30
CN100460415C (zh) 2009-02-11
EP1291353A1 (en) 2003-03-12
DE69733422D1 (de) 2005-07-07
KR100610043B1 (ko) 2006-08-08
HRP20060276B1 (hr) 2014-04-25
CN1680420A (zh) 2005-10-12
DE69733370T2 (de) 2006-02-02
ES2242812T3 (es) 2005-11-16
BG63547B1 (bg) 2002-04-30
SK285535B6 (sk) 2007-03-01
CA2263972A1 (en) 1998-03-12
DK1291350T3 (da) 2005-09-26
EP1291351B1 (en) 2005-07-13
HUP9902869A3 (en) 2001-04-28
PT1291353E (pt) 2005-10-31
JP2001500855A (ja) 2001-01-23
EP1291350A1 (en) 2003-03-12
KR20050043993A (ko) 2005-05-11
CN1273475C (zh) 2006-09-06
TR199901127T2 (xx) 1999-07-21
EP1291353B1 (en) 2005-06-01
HRP20060277B1 (hr) 2014-04-11
DE69733422T2 (de) 2006-05-04
AU4178097A (en) 1998-03-26
KR100523679B1 (ko) 2005-10-26
DK1291351T3 (da) 2005-10-24
DE69733369T2 (de) 2006-01-26
EP1291352B1 (en) 2005-05-25
ES2244716T3 (es) 2005-12-16
ATE296831T1 (de) 2005-06-15
DE69733723D1 (de) 2005-08-18
US6028181A (en) 2000-02-22
AU729348B2 (en) 2001-02-01
EP1291350B1 (en) 2005-05-25
IL128681A0 (en) 2000-01-31
CZ68599A3 (cs) 1999-08-11
HRP970473B1 (hr) 2007-02-28
KR100568455B1 (ko) 2006-04-07
EP0929563A1 (en) 1999-07-21
CN100441591C (zh) 2008-12-10
PT929563E (pt) 2005-10-31
DK0929563T3 (da) 2005-10-03
KR100576988B1 (ko) 2006-05-10
NO991022L (no) 1999-05-03
RU2192427C2 (ru) 2002-11-10
KR20050043994A (ko) 2005-05-11
CN1680418A (zh) 2005-10-12
CA2263972C (en) 2008-01-29
SK286181B6 (sk) 2008-04-07
SK285534B6 (sk) 2007-03-01
BR9711661A (pt) 1999-08-24
EP1291352A1 (en) 2003-03-12
HRP20060278B1 (hr) 2014-04-11
NO314230B1 (no) 2003-02-17
SI20023B (en) 2001-02-28
DK1291352T3 (da) 2005-09-19
SK28699A3 (en) 2000-03-13
EP0929563B1 (en) 2005-06-01
ES2242813T3 (es) 2005-11-16
ATE299508T1 (de) 2005-07-15
DE69733370D1 (de) 2005-06-30
CZ300106B6 (cs) 2009-02-11
HRP20060278A2 (hr) 2007-10-31
PT1291352E (pt) 2005-09-30
US6075133A (en) 2000-06-13
HRP20060276A2 (hr) 2007-10-31
DK1291353T3 (da) 2005-10-03
HRP970473A2 (en) 1998-08-31
ATE296832T1 (de) 2005-06-15
SK285533B6 (sk) 2007-03-01
KR20000068435A (ko) 2000-11-25
DE69733369D1 (de) 2005-06-30
ES2242811T3 (es) 2005-11-16
ATE296307T1 (de) 2005-06-15
SI20023A (sl) 2000-02-29
KR20050044816A (ko) 2005-05-12
JP4597274B2 (ja) 2010-12-15
NO991022D0 (no) 1999-03-02
ES2242983T3 (es) 2005-11-16
CN1680419A (zh) 2005-10-12

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