CA2564377A1 - 6-o-substituted ketolides having antibacterial activity - Google Patents

6-o-substituted ketolides having antibacterial activity Download PDF

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Publication number
CA2564377A1
CA2564377A1 CA002564377A CA2564377A CA2564377A1 CA 2564377 A1 CA2564377 A1 CA 2564377A1 CA 002564377 A CA002564377 A CA 002564377A CA 2564377 A CA2564377 A CA 2564377A CA 2564377 A1 CA2564377 A1 CA 2564377A1
Authority
CA
Canada
Prior art keywords
compounds
antibacterial activity
substituted ketolides
iva
ketolides
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002564377A
Other languages
French (fr)
Other versions
CA2564377C (en
Inventor
Yat Sun Or
Zhenkun Ma
Richard F. Clark
Jacob J. Plattner
George Griesgraber
Daniel T. Chu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AbbVie Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/888,350 external-priority patent/US5866549A/en
Application filed by Individual filed Critical Individual
Priority claimed from CA002263972A external-priority patent/CA2263972C/en
Publication of CA2564377A1 publication Critical patent/CA2564377A1/en
Application granted granted Critical
Publication of CA2564377C publication Critical patent/CA2564377C/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

Antimicrobial compounds having formula (IV) or (IVA) as well as pharmaceutically acceptable salts, esters or prodrugs thereof; pharmaceutical compositions comprising such compounds; methods of treating bacterial infections by the administration of such compounds; and processes for the preparation of the compounds. (see formula IV) or (see formula IVA)
CA002564377A 1996-09-04 1997-09-02 6-o-substituted ketolides having antibacterial activity Expired - Lifetime CA2564377C (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US70777696A 1996-09-04 1996-09-04
US08/707,776 1996-09-04
US08/888,350 1997-07-03
US08/888,350 US5866549A (en) 1996-09-04 1997-07-03 6-O-substituted ketolides having antibacterial activity
CA002263972A CA2263972C (en) 1996-09-04 1997-09-02 6-o-substituted ketolides having antibacterial activity

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CA002263972A Division CA2263972C (en) 1996-09-04 1997-09-02 6-o-substituted ketolides having antibacterial activity

Publications (2)

Publication Number Publication Date
CA2564377A1 true CA2564377A1 (en) 1998-03-12
CA2564377C CA2564377C (en) 2009-08-11

Family

ID=37545836

Family Applications (3)

Application Number Title Priority Date Filing Date
CA002563965A Expired - Lifetime CA2563965C (en) 1996-09-04 1997-09-02 6-0-substituted ketolides having antibacterial activity
CA002564020A Expired - Lifetime CA2564020C (en) 1996-09-04 1997-09-02 6-o-substituted ketolides having antibacterial activity
CA002564377A Expired - Lifetime CA2564377C (en) 1996-09-04 1997-09-02 6-o-substituted ketolides having antibacterial activity

Family Applications Before (2)

Application Number Title Priority Date Filing Date
CA002563965A Expired - Lifetime CA2563965C (en) 1996-09-04 1997-09-02 6-0-substituted ketolides having antibacterial activity
CA002564020A Expired - Lifetime CA2564020C (en) 1996-09-04 1997-09-02 6-o-substituted ketolides having antibacterial activity

Country Status (1)

Country Link
CA (3) CA2563965C (en)

Also Published As

Publication number Publication date
CA2564020C (en) 2009-10-27
CA2564377C (en) 2009-08-11
CA2564020A1 (en) 1998-03-12
CA2563965A1 (en) 1998-03-12
CA2563965C (en) 2009-08-25

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Legal Events

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EEER Examination request
MKEX Expiry

Effective date: 20170905