FI960155A - Terapeuttisia heterosyklisiä yhdisteitä - Google Patents

Terapeuttisia heterosyklisiä yhdisteitä Download PDF

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Publication number
FI960155A
FI960155A FI960155A FI960155A FI960155A FI 960155 A FI960155 A FI 960155A FI 960155 A FI960155 A FI 960155A FI 960155 A FI960155 A FI 960155A FI 960155 A FI960155 A FI 960155A
Authority
FI
Finland
Prior art keywords
formula
alkyl
hydrogen
heterocyclic compounds
group
Prior art date
Application number
FI960155A
Other languages
English (en)
Swedish (sv)
Other versions
FI960155A0 (fi
FI106262B (fi
Inventor
Alan Duncan Robertson
Alan Peter Hill
Robert Charles Glen
Graeme Richard Martin
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26297174&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI960155(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB909012672A external-priority patent/GB9012672D0/en
Priority claimed from GB919102182A external-priority patent/GB9102182D0/en
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of FI960155A0 publication Critical patent/FI960155A0/fi
Publication of FI960155A publication Critical patent/FI960155A/fi
Application granted granted Critical
Publication of FI106262B publication Critical patent/FI106262B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Steroid Compounds (AREA)
FI960155A 1990-06-07 1996-01-12 Menetelmä terapeuttisesti käyttökelpoisten yhdisteiden valmistamiseksi FI106262B (fi)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
GB9012672 1990-06-07
GB909012672A GB9012672D0 (en) 1990-06-07 1990-06-07 Therapeutic heterocyclic compounds
GB919102182A GB9102182D0 (en) 1991-02-01 1991-02-01 Therapeutic heterocyclic compounds
GB9102182 1991-02-01
GB9100908 1991-06-06
PCT/GB1991/000908 WO1991018897A1 (en) 1990-06-07 1991-06-06 Therapeutic heterocyclic compounds
FI920503A FI105686B (fi) 1990-06-07 1992-02-06 Menetelmä terapeuttisesti käyttökelpoisen yhdisteen ja sen fysiologisesti hyväksyttävien suolojen valmistamiseksi
FI920503 1992-02-06

Publications (3)

Publication Number Publication Date
FI960155A0 FI960155A0 (fi) 1996-01-12
FI960155A true FI960155A (fi) 1996-01-12
FI106262B FI106262B (fi) 2000-12-29

Family

ID=26297174

Family Applications (3)

Application Number Title Priority Date Filing Date
FI920503A FI105686B (fi) 1990-06-07 1992-02-06 Menetelmä terapeuttisesti käyttökelpoisen yhdisteen ja sen fysiologisesti hyväksyttävien suolojen valmistamiseksi
FI960155A FI106262B (fi) 1990-06-07 1996-01-12 Menetelmä terapeuttisesti käyttökelpoisten yhdisteiden valmistamiseksi
FI20001406A FI20001406A (fi) 1990-06-07 2000-06-13 Terapeuttisia heterosyklisiä yhdisteitä

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FI920503A FI105686B (fi) 1990-06-07 1992-02-06 Menetelmä terapeuttisesti käyttökelpoisen yhdisteen ja sen fysiologisesti hyväksyttävien suolojen valmistamiseksi

Family Applications After (1)

Application Number Title Priority Date Filing Date
FI20001406A FI20001406A (fi) 1990-06-07 2000-06-13 Terapeuttisia heterosyklisiä yhdisteitä

Country Status (37)

Country Link
US (3) US5399574A (fi)
EP (2) EP0636623B1 (fi)
JP (1) JP2738461B2 (fi)
KR (1) KR100215627B1 (fi)
AT (2) ATE156823T1 (fi)
AU (1) AU646871B2 (fi)
CA (2) CA2064815C (fi)
CZ (1) CZ288351B6 (fi)
DE (3) DE69127260T2 (fi)
DK (1) DK0486666T3 (fi)
EG (1) EG19650A (fi)
ES (1) ES2104708T3 (fi)
FI (3) FI105686B (fi)
GR (1) GR3024828T3 (fi)
HK (1) HK1000534A1 (fi)
HR (1) HRP940524B1 (fi)
HU (2) HU219974B (fi)
IE (1) IE911931A1 (fi)
IL (3) IL114690A (fi)
LT (1) LT3264B (fi)
LU (1) LU90205I2 (fi)
LV (1) LV10274B (fi)
MC (1) MC2210A1 (fi)
MX (1) MX9203421A (fi)
MY (1) MY110226A (fi)
NL (1) NL980001I2 (fi)
NO (2) NO300634B1 (fi)
NZ (1) NZ238424A (fi)
PL (1) PL166214B1 (fi)
PT (1) PT97888B (fi)
RU (1) RU2160736C2 (fi)
SA (1) SA05260104B1 (fi)
SI (2) SI9111010B (fi)
SK (1) SK281621B6 (fi)
UA (1) UA37178C2 (fi)
WO (1) WO1991018897A1 (fi)
YU (1) YU48855B (fi)

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* Cited by examiner, † Cited by third party
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